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ACS电子期刊(619)
Wiley电子期刊(307)
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Elsevier电子期刊(1621)
在“
Elsevier电子期刊
”中,
命中:
1,621
条,耗时:0.0199895 秒
在所有数据库中总计命中:
4,353
条
1.
Synthesis, characterization, crystal structure and biological studies of silver(I) complexes derived from coumarin-tethered N-
heterocyclic
carbene ligands
作者:
Gautam Achar
a
;
1
;
K. Uppendranath
a
;
1
;
V.C. Ramya
a
;
Andrea Biffis
b
;
Rangappa S. Keri
a
;
Srinivasa Budagumpi
a
;
b.srinivasa@jainuniversity.ac.in
;
dr.sinuvb@gmail.com
关键词:
Antibacterial agent
;
E. coli
;
N-
heterocyclic
carbene
;
Silver complex
;
X-ray diffraction
刊名:Polyhedron
出版年:2017
2.
Therapeutic evolution of benzimidazole
derivative
s in the last quinquennial period
作者:
Wasim Akhtar
a
;
Mohemmed Faraz Khan
a
;
Garima Verma
a
;
M. Shaquiquzzaman
a
;
M.A. Rizvi
b
;
Syed Hassan Mehdi
b
;
Mymoona Akhter
a
;
M. Mumtaz Alam
a
;
drmmalam@gmail.com
关键词:
Heterocyclic
;
Benzimidazole
;
Biological activity
;
Anti-inflammatory and analgesic
;
Anti-cancer
;
Antiviral
刊名:European Journal of Medicinal Chemistry
出版年:2017
3.
Design and synthesis of novel 2-substituted 11-keto-boswellic acid
heterocyclic
derivative
s as anti-prostate cancer agents with Pin1 inhibition ability
作者:
Kun Li
a
;
Lei Li
b
;
Shuxiang Wang
a
;
Xiaojing Li
a
;
Tianyi Ma
a
;
Dan Liu
a
;
sammyld@163.com
;
Yongkui Jing
b
;
yongkjing@yahoo.com
;
Linxiang Zhao
a
;
linxiang.zhao@vip.sina.com
关键词:
Acetyl-11-keto-β-boswellic acid
;
Anti-proliferative activity
;
Cyclin D1
;
Cell cycle
;
Pin1
刊名:European Journal of Medicinal Chemistry
出版年:2017
4.
Stereoselective synthesis of diazaspiro[5.5]undecane
derivative
s via base promoted [5+1] double Michael addition of N,N-dimethylbarbituric acid to diaryliedene acetones
作者:
Mohammad Shahidul Islam
a
;
1
;
mislam@ksu.edu.sa
;
Assem Barakat
a
;
b
;
1
;
ambarakat@ksu.edu.sa
;
Abdullah Mohammed Al-Majid
a
;
1
;
Hazem A Ghabbour
c
;
1
;
Hoong-Kun Fun
c
;
d
;
1
;
M. Rafiq Siddiqui
a
;
1
关键词:
Cascade [5+1] cycloaddition
;
Double Michael reaction
;
Diethylamine catalysis
;
Diazaspiro[5.5]undecane
;
N
;
N-Dimethylbarbituric acid diaryliedene acetone
刊名:Arabian Journal of Chemistry
出版年:2017
5.
Design and synthesis of 4,5,6,7‐tetrahydro‐1H‐1,2‐diazepin‐7‐one
derivative
s as a new series of Phosphodiesterase 4 (PDE4) inhibitors
作者:
Sara Guariento
a
;
Anna Karawajczyk
b
;
James A. Bull
b
;
Gessica Marchini
c
;
Martyna Bielska
b
;
Xenia Iwanowa
b
;
Olga Bruno
a
;
Paola Fossa
a
;
Fabrizio Giordanetto
b
;
fabrizio.giordanetto@deshawresearch.com
关键词:
Phosphodiesterase 4
;
PDE4 inhibitors
;
Diazepinone
derivative
s
;
Compound library
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
6.
A betulinic acid
derivative
SH479 inhibits collagen-induced arthritis by modulating T cell differentiation and cytokine balance
作者:
Shijie Chen
a
;
b
;
1
;
Yang Bai
a
;
1
;
Zhen Li
a
;
1
;
Kunhang Jia
a
;
Yunyun Jin
a
;
Bei He
a
;
Wen-Wei Qiu
c
;
Changsheng Du
d
;
Stefan Siwko
e
;
Huaqing Chen
a
;
hqchen@bio.ecnu.edu.cn
;
Mingyao Liu
a
;
e
;
myliu@bio.ecnu.edu.cn
;
Jian Luo
a
;
jluo@bio.ecnu.edu.cn
关键词:
Betulinic acid
;
SH479
;
Collagen-induced arthritis
;
Th17 cell differentiation
;
STAT3 signaling
刊名:Biochemical Pharmacology
出版年:2017
7.
New N- and O-arylpiperazinylalkyl pyrimidines and 2-methylquinazolines
derivative
s as 5-HT
7
and 5-HT
1A
receptor ligands: Synthesis, structure-activity relationships, and molecular modeling studies
作者:
Sebastiano Intagliata
a
;
1
;
s.intagliata@studium.unict.it
;
Maria N. Modica
a
;
1
;
Valeria Pittalà
;
a
;
Loredana Salerno
a
;
Maria A. Siracusa
a
;
Alfredo Cagnotto
b
;
Mario Salmona
b
;
Rafał Kurczab
c
;
Giuseppe Romeo
a
关键词:
5-HT7 receptor ligands
;
5-HT1A receptor ligands
;
Long-chain arylpiperazines
;
Molecular modeling
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
8.
Structure-activity relationship (SAR) study and design strategies of nitrogen-containing
heterocyclic
moieties for their anticancer activities
作者:
Jawaid Akhtar
;
Ahsan Ahmed Khan
;
Zulphikar Ali
;
Rafi Haider
;
M. Shahar Yar
;
msyar@rediffmail.com
关键词:
Anticancer
;
Cytotoxic
;
SARs
;
N-Heterocycles
刊名:European Journal of Medicinal Chemistry
出版年:2017
9.
Toxicity evaluation of the photoprotective compound LQFM048: Eye irritation, skin toxicity and genotoxic endpoints
作者:
Renato Ivan de Á
;
vila
a
;
1
;
Marcelo de Sousa Vieira
a
;
1
;
Marilisa Pedroso Nogueira Gaeti
b
;
Larissa Cleres Moreira
a
;
Laí
;
s de Brito Rodrigues
a
;
Gisele Augusto Rodrigues de Oliveira
a
;
Aline Carvalho Batista
c
;
Daniela Cristina Vinhal
d
;
Ricardo Menegatti
d
;
Marize Campos Valadares
a
;
marizeufg@gmail.com
关键词:
Alternative methods
;
Eye irritation
;
Genotoxicity
;
Heterocyclic
derivative
;
Phototoxicity
;
Skin sensitization
刊名:Toxicology
出版年:2017
10.
Preparation of novel ring-A fused azole
derivative
s of betulin and evaluation of their cytotoxicity
作者:
Victoria V. Grishko
a
;
grishvic@gmail.com
;
Irina A. Tolmacheva
a
;
Vladimir O. Nebogatikov
a
;
Natalia V. Galaiko
a
;
Alexei V. Nazarov
a
;
Maxim V. Dmitriev
b
;
Irena B. Ivshina
b
;
c
关键词:
Betulin
;
Heterocycles
;
Azoles
;
Tumor cells
;
MTT assay
;
Apoptosis
刊名:European Journal of Medicinal Chemistry
出版年:2017
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6
7
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