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Wiley电子期刊(2)
SpringerLink电子期刊(27)
Elsevier电子期刊(18)
ACS电子期刊(7)
在“
Elsevier电子期刊
”中,
命中:
18
条,耗时:小于0.01 秒
在所有数据库中总计命中:
54
条
1.
In silico investigation of medicinal spectrum of
imidazo
-
azines
from the perspective of multitarget screening against malaria, tuberculosis and Chagas disease
作者:
Manoj Kumar
;
Barnita Makhal
;
Vinod Kumar Gupta
;
Anuj Sharma
;
anujsharma.mcl@gmail.com" class="auth_mail
关键词:
Docking
;
Imidazo
-
azines
;
Ligand efficiency
;
Multitarget screening
;
Lead-likeness
刊名:Journal of Molecular Graphics and Modelling
出版年:May 2014
2.
Regioselective synthesis of
imidazo
[1,2-a][1,3,5]tri
azines
and 3,4-dihydro
imidazo
[1,2-a][1,3,5]tri
azines
from [1,3,5]triazin-2,4-diamines
作者:
Pascal Dao
;
Christiane Garbay
;
Huixiong Chen
;
huixiong.chen@parisdescartes.fr
关键词:
Nitrogen heterocycles
;
Cyclization
;
Regioselectivity
;
Reaction mechanisms
刊名:Tetrahedron
出版年:2013
3.
Synthesis and structure of new
imidazo
- and pyrazolo[5,1-d][1,2,3,5]thiatri
azines
based on the reaction of diazoazoles with acyl isothiocyanates controlled by S?O interaction
作者:
Elena V. Sadchikova
;
Vasiliy A. Bakulev
;
Julia O. Subbotina
;
Darya L. Privalova
;
Wim Dehaen
;
Kristof Van Hecke
;
Koen Robeyns
;
Luc Van Meervelt
;
Vladimir S. Mokrushin
关键词:
Cycloaddition
;
Diazoazoles
;
Thiatri
azines
;
Nonbonded S?O interaction
;
Covalence ratio factor
刊名:Tetrahedron
出版年:2013
4.
1-Arylamino
imidazo
le-2-thiones as intermediates in the synthesis of
imidazo
[2,1-b][1,3,4]thiadi
azines
作者:
Constantinos Neochoritis
;
Constantinos A. Tsoleridis
;
Julia Stephanidou-Stephanatou
关键词:
Imidazo
lethiadi
azines
;
Imidazo
lone
;
Methylation
;
Selectivity
;
S
-Vinyl
imidazo
les
刊名:Tetrahedron
出版年:2008
5.
Pyrazolo[1,5-a]pyrimidines, triazolo[1,5-a]pyrimidines and their tricyclic derivatives as corticotropin-releasing factor 1 (CRF
1
) receptor antagonists
作者:
Tetsuji
;
Saito
;
;
;
te.saitou@ono.co.jp
;
Tetsuo
;
Obitsu
;
Chiaki
;
Minamoto
;
Tsuneyuki
;
Sugiura
;
Naoya
;
Matsumura
;
Sonoko
;
Ueno
;
Akihiro
;
Kishi
;
Seishi
;
Katsumata
;
Hisao
;
Nakai
;
Masaaki
;
Toda
关键词:
Corticotrophin-releasing factor 1 receptor
;
Antagonist
刊名:Bioorganic and Medicinal Chemistry
出版年:2011
6.
Antinociceptive activity of new
imidazo
lidine carbonyl derivatives.: Part 4. Synthesis and pharmacological activity of 8-aryl-3,4-dioxo-2H,8H-6,7-dihydro
imidazo
[2,1-c] [1,2,4]tri
azines
作者:
Krzysztof Sztanke
;
Sylwia Fidecka
;
Ewa Kę
;
dzierska
;
Zbigniew Karczmarzyk
;
Kalevi Pihlaja
;
Dariusz Matosiuk
关键词:
CNS activity
;
Opioid-like analgesics
;
Antinociception
;
Imidazo
[2
;
1-
c
] [1
2 ;
4]tri
azines
;
Molecular structure
;
Amido-imido tautomerism
刊名:European Journal of Medicinal Chemistry
出版年:2005
7.
Imidazo
[1,2-b][1,2,4]tri
azines
as α2/α3 subtype selective GABA
A
agonists for the treatment of anxiety
作者:
Andrew S.R. Jennings
;
Richard T. Lewis
;
Michael G.N. Russell
;
David J. Hallett
;
Leslie J. Street
;
José
;
L. Castro
;
John R. Atack
;
Susan M. Cook
;
Rachael Lincoln
;
Joanna Stanley
et al.
关键词:
Imidazo
[
1 ;
2-
a
]
;
pyrimidines
;
Imidazo
[
1 ;
2-
b
]
;
[
12 ;
4]
;
tri
azines
;
GABAA receptors
;
α
;
2/α
;
3 subtype selective
;
Anxiolytic
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2006
8.
Reaction between isocyanides and dialkyl acetylenedicarboxylates in the presence of 4,5-diphenyl-1,3-dihydro-2H-
imidazo
l-2-one. One-pot synthesis of 5H-
imidazo
[2,1-b][1,3]oxazine derivatives
作者:
Adib
;
Mehdi
;
Ghanbary
;
Khadijeh
;
Mostofi
;
Manizheh
;
Reza Bijanzadeh
;
Hamid
关键词:
Isocyanides
;
Acetylenic esters
;
4
;
5-Diphenyl-1
;
3-dihydro-2
H
-
imidazo
l-2-one
;
Three-component reactions
;
2
;
3-Diphenyl-5
H
-
imidazo
[2
;
1-
b
][1
;
3]ox
azines
刊名:Tetrahedron
出版年:2005
9.
Efficient highly diastereoselective synthesis of 1,8a-dihydro-7H-
imidazo
[2,1-b][1,3]ox
azines
作者:
Mehdi Adib
;
Esmaeil Sheibani
;
Manizheh Mostofi
;
Khadijeh Ghanbary and Hamid Reza Bijanzadeh
关键词:
Diastereoselective synthesis
;
Pyridine carboxaldehydes
;
Acetylenic esters
;
1-Alkyl
imidazo
les
;
1
;
8a-Dihydro-7
H
-
imidazo
[
2 ;
1-
b
]
;
[
1 ;
3]
;
ox
azines
刊名:Tetrahedron
出版年:2006
10.
Synthesis and antitubercular activity of 7-(R)- and 7-(S)-methyl-2-nitro-6-(S)-(4-(trifluoromethoxy)benzyloxy)-6,7-dihydro-5H-
imidazo
[2,1-b][1,3]ox
azines
, analogues of PA-824
作者:
Xiaojin Li
;
Ujjini H. Manjunatha
;
Michael B. Goodwin
;
John E. Knox
;
Christopher A. Lipinski
;
Thomas H. Keller
;
Clifton E. Barry III
;
Cynthia S. Dowd
关键词:
Mycobacterium tuberculosis
;
PA-824
;
Solubility
;
Water solubility
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2008
1
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