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SpringerLink电子期刊(26)
NATURE电子期刊(1)
Elsevier电子期刊(53)
ACS电子期刊(6)
在“
Elsevier电子期刊
”中,
命中:
53
条,耗时:0.0129961 秒
在所有数据库中总计命中:
86
条
1.
New insights into the SAR and drug combination synergy of 2-(quinolin-4-yloxy)acetamides against Mycobacterium tuberculosis
作者:
Bruno Couto Giacobbo
a
;
b
;
Kenia Pissinate
a
;
Valnê
;
s Rodrigues-Junior
a
;
Anne Drumond Villela
a
;
Estê
;
vã
;
o Silveira Grams
a
;
Bruno Lopes Abbadi
a
;
b
;
Fernanda Teixeira Subtil
a
;
b
;
Nathalia Sperotto
a
;
c
;
Rogé
;
rio Valim Trindade
a
;
b
;
Davi Fernando Back
d
;
Maria Martha Campos
a
;
b
;
c
;
Luiz Augusto Basso
a
;
b
;
c
;
Pablo Machado
a
;
b
;
pablo.machado@pucrs.br
;
Dió
;
genes Santiago Santos
a
;
b
;
diogenes@pucrs.br
关键词:
Tuberculosis
;
Intracellular activity
;
Synergism
;
Drug-resistant strains
刊名:European Journal of Medicinal Chemistry
出版年:2017
2.
The Non-Linear Child: Ontogeny,
Isoniazid
Concentration, and NAT2 Genotype Modulate Enzyme Reaction Kinetics and
Metabolism
作者:
Zoe Rogers
a
;
Hiwot Hiruy
b
;
Jotam G. Pasipanodya
c
;
Chris Mbowane
d
;
John Adamson
a
;
Lihle Ngotho
a
;
Farina Karim
a
;
Prakash Jeena
d
;
William Bishai
b
;
e
;
Tawanda Gumbo
c
;
f
;
tawanda.gumbo@baylorhealth.edu" class="auth_mail" title="E-mail the corresponding author
关键词:
NAT2 reaction kinetics
;
Isoniazid
concentration
;
Maturation
;
NAT2 genotype
;
Artificial intelligence
刊名:EBioMedicine
出版年:2016
3.
Metabolism
of
isoniazid
by neutrophil myeloperoxidase leads to
isoniazid
-NAD
+
adduct formation: A comparison of the reactivity of
isoniazid
with its known human metabolites
作者:
Saifur R. Khan
a
;
Andrew G.M. Morgan
a
;
Karim Michail
a
;
Nutan Srivastava
a
;
Randy M. Whittal
b
;
Naif Aljuhani
a
;
c
;
Arno G. Siraki
a
;
siraki@ualberta.ca" class="auth_mail" title="E-mail the corresponding author
关键词:
Isoniazid
;
Myeloperoxidase
;
Neutrophil
;
INH-NAD+
;
Free radicals
刊名:Biochemical Pharmacology
出版年:2016
4.
Isoniazid
metabolism
and hepatotoxicity
作者:
Pengcheng Wang
a
;
Komal Pradhan
a
;
Xiao-bo Zhong
b
;
Xiaochao Ma
a
;
mxiaocha@pitt.edu" class="auth_mail" title="E-mail the corresponding author
关键词:
AcHz
;
acetylhydrazine
;
AcINH
;
acetyl
isoniazid
;
ALP
;
alkaline phosphatase
;
ALT
;
alanine aminotransferase
;
DiAcHz
;
diacetylhydrazine
;
GSH
;
glutathione
;
GST
;
glutathione S-transferase
;
Hz
;
hydrazine
;
INA
;
isonicotinic acid
;
INH
;
isoniazid
;
MPO
;
myeloperoxidase
;
NAD+
;
nicotinamide adenine dinucleotide
;
NAT
;
N-acetyltransferase
;
P450
;
cytochrome P450
;
R.M.
;
reactive metabolite
;
TB
;
tuberculosis
刊名:Acta Pharmaceutica Sinica B
出版年:2016
5.
Effects of repeated administration of rifampicin and
isoniazid
on vitamin D
metabolism
in mice
作者:
Li Sheng
a
;
Ying Xue
a
;
Xin He
a
;
Yungui Zhu
a
;
Huande Li
a
;
lihuande1953@126.com" class="auth_mail" title="E-mail the corresponding author
;
Yanqin Wu
a
;
Ruili Dang
a
;
b
;
Mimi Tang
a
;
Pei Jiang
b
;
jpoet89@126.com" class="auth_mail" title="E-mail the corresponding author
关键词:
Vitamin D
metabolism
;
Tuberculosis
;
Rifampicin
;
Isoniazid
刊名:Steroids
出版年:2015
6.
New agents for the treatment of drug-resistant Mycobacterium tuberculosis
作者:
Daniel T. Hoagland
a
;
b
;
Jiuyu Liu
a
;
Robin B. Lee
a
;
Richard E. Lee
a
;
richard.lee@stjude.org" class="auth_mail" title="E-mail the corresponding author
关键词:
Mtb
;
Mycobacterium tuberculosis
;
TB
;
Tuberculosis
;
MDR-TB
;
Multidrug-resistant tuberculosis
;
RIF
;
Rifampicin
;
INH
;
Isoniazid
;
PZA
;
Pyrazinamide
;
ETH
;
Ethambutol
;
WHO
;
World Health Organization
;
CYP
;
Cytochrome P450
;
ADME
;
Absorption
;
distribution
;
metabolism
;
and excretion
;
HIV
;
Human immunodeficiency virus
;
XDR-TB
;
Extensively drug-resistant tuberculosis
;
TDR-TB
;
Totally drug-resistant tuberculosis
;
PK
;
Pharmacokinetic
;
PD
;
Pharmacodynamic
;
EMA
;
European medicines agency
;
FDA
;
Food and drug adm
刊名:Advanced Drug Delivery Reviews
出版年:2016
7.
Pyrazinamide resistance in Mycobacterium tuberculosis: Review and update
作者:
Moses Njire
a
;
1
;
Yaoju Tan
b
;
1
;
Julius Mugweru
a
;
Changwei Wang
a
;
Jintao Guo
a
;
WingWai Yew
c
;
Shouyong Tan
b
;
tanshyo@tom.com" class="auth_mail" title="E-mail the corresponding author
;
Tianyu Zhang
a
;
zhang_tianyu@gibh.ac.cn" class="auth_mail" title="E-mail the corresponding author
关键词:
Tuberculosis
;
MDR
;
XDR
;
Pyrazinamide
;
Drug resistance
刊名:Advances in Medical Sciences
出版年:2016
8.
Study of mechanism of interaction of truncated
isoniazid
-nicotinamide adenine dinucleotide adduct against multiple enzymes of Mycobacterium tuberculosis by a computational approach
作者:
Lingaraja Jena
;
Shraddha Deshmukh
;
Pranita Waghmare
;
Satish Kumar
;
Bhaskar C. Harinath
;
bc_harinath@yahoo.com" class="auth_mail" title="E-mail the corresponding author
;
info@jbtdrc.org" class="auth_mail" title="E-mail the corresponding author
关键词:
Catalytic triad
;
Docking
;
Isoniazid
;
Truncated INH&ndash
;
NAD adduct
刊名:International Journal of Mycobacteriology
出版年:2015
9.
Pharmacokinetics, tissue distribution and relative bioavailability of
isoniazid
-solid lipid nanoparticles
作者:
Rohit Bhandari
;
Indu Pal Kaur
;
indupalkaur@yahoo.com
关键词:
Solid lipid nanoparticles
;
Isoniazid
;
Pharmacokinetics
;
Bioavailability
;
Tuberculosis
刊名:International Journal of Pharmaceutics
出版年:2013
10.
Synthesis and bioevaluation of some new
isoniazid
derivatives
作者:
Lilia Matei
;
Coralia Bleotu
;
Ion Baciu
;
Constantin Draghici
;
Petre Ionita
;
Anca Paun
;
Mariana Carmen Chifiriuc
;
Adriana Sbarcea
;
Irina Zarafu
关键词:
Isoniazid
;
Thioamides
;
Synthesis
;
Biological evaluation
;
Antitubercular activity
刊名:Bioorganic and Medicinal Chemistry
出版年:2013
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