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内部出版物
Wiley电子期刊(2)
Elsevier电子期刊(5)
ACS电子期刊(1)
在“
Elsevier电子期刊
”中,
命中:
5
条,耗时:小于0.01 秒
在所有数据库中总计命中:
8
条
1.
Synthesis and preliminary in vitro kinase inhibition evaluation of new diversely substituted pyrido[3,4-g]quinazoline derivatives
作者:
Wael Zeinyeh
a
;
b
;
Yannick J. Esvan
a
;
b
;
Lionel Nauton
a
;
b
;
Nadè
;
ge Loaë
;
c
c
;
Laurent
Meijer
c
;
Vincent Thé
;
ry
a
;
b
;
Fabrice Anizon
a
;
b
;
Francis Giraud
a
;
b
;
Francis.GIRAUD@univ-bpclermont.fr" class="auth_mail" title="E-mail the corresponding author
;
Pascale Moreau
a
;
b
;
Pascale.MOREAU@univ-bpclermont.fr" class="auth_mail" title="E-mail the corresponding author
关键词:
Pyrido[3
;
4-g]quinazoline
;
Protein kinase inhibition
;
CLK1
;
DYRK1A
;
CDK5
;
GSK3
;
CK1
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
2.
Discovery of pyrido[3,4-g]quinazoline derivatives as CMGC family protein kinase inhibitors: Design, synthesis, inhibitory potency and X-ray co-crystal structure
作者:
Yannick J. Esvan
a
;
b
;
1
;
Wael Zeinyeh
a
;
b
;
1
;
Thibaut Boibessot
a
;
b
;
Lionel Nauton
a
;
b
;
Vincent Thé
;
ry
a
;
b
;
Stefan Knapp
c
;
d
;
Apirat Chaikuad
c
;
d
;
Nadè
;
ge Loaë
;
c
e
;
Laurent
Meijer
e
;
Fabrice Anizon
a
;
b
;
Francis Giraud
a
;
b
;
Francis.GIRAUD@univ-bpclermont.fr" class="auth_mail" title="E-mail the corresponding author
;
Pascale Moreau
a
;
b
;
Pascale.MOREAU@univ-bpclermont.fr" class="auth_mail" title="E-mail the corresponding author
关键词:
Pyrido[3
;
4-g]quinazoline
;
Kinase inhibitors
;
Ser/Thr kinases
;
CMGC family
;
CLK1 binding mode
刊名:European Journal of Medicinal Chemistry
出版年:2016
3.
Synthesis and optimization of an original V-shaped collection of 4-7-disubstituted Pyrido[3,2-d]pyrimidines as CDK5 and DYRK1A inhibitors
作者:
Oussama Dehbi
a
;
b
;
Abdellatif Tikad
a
;
b
;
Sté
;
phane Bourg
a
;
Pascal Bonnet
a
;
Olivier Lozach
c
;
Laurent
Meijer
c
;
1
;
Mina Aadil
b
;
Mohammed Akssira
b
;
Gé
;
rald Guillaumet
a
;
gerald.guillaumet@univ-orleans.fr" class="auth_mail
;
Sylvain Routier
a
;
sylvain.routier@univ-orleans.fr" class="auth_mail
关键词:
Pyridopyrimidine
;
CDK5
;
DYRK1A
;
Synthesis
;
SAR
;
Molecular modelling
刊名:European Journal of Medicinal Chemistry
出版年:10 June 2014
4.
Synthesis and biological evaluation of N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amines and their pyrido and pyrazino analogues as Ser/Thr kinase inhibitors
作者:
Yvonnick Loidreau
a
;
Pascal Marchand
b
;
Carole Dubouilh-Benard
a
;
Marie-René
;
e Nourrisson
b
;
Muriel Duflos
b
;
Olivier Lozach
c
;
Nadè
;
ge Loaë
;
c
c
;
d
;
Laurent
Meijer
d
;
Thierry Besson
a
;
thierry.besson@univ-rouen.fr
关键词:
Microwave-assisted chemistry
;
Dimroth rearrangement
;
Thieno[3
;
2-d]pyrimidine
;
Dimethylformamide dimethylacetal
;
Kinase inhibitor
;
Alzheimer's disease
刊名:European Journal of Medicinal Chemistry
出版年:2012
5.
Dipyrido[3,2-a:2′,3′-c]quinolino[3,2-j]phenazine (dpqp-OH) – Synthesis, characterization and DNA interaction of the corresponding Ru(II) complex
作者:
Laurent
Bouffier
;
Martine Demeunynck
;
Pascal Dumy
;
Cé
;
cile Moucheron
;
André
;
e Kirsch-De Mesmaeker
关键词:
Ruthenium ligand
;
Polyazaaromatic
;
DNA binding
;
Phenanthroline
刊名:Inorganica Chimica Acta
出版年:2007
1
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2012年(1)
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2000年及以前(1)
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