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内部出版物
Elsevier电子期刊(3)
ACS电子期刊(4)
在“
Elsevier电子期刊
”中,
命中:
3
条,耗时:小于0.01 秒
在所有数据库中总计命中:
7
条
1.
Difluorocyclobutylacetylenes as positive allosteric modulators of mGluR5 with reduced bioactivation potential
作者:
Andrew P. Degnan
;
andrew.degnan@bms.com
;
Darrell Maxwell
;
Anand Balakrishnan
;
Jeffrey M. Brown
;
Amy Easton
;
Michael Gulianello
;
Umesh Hanumegowda
;
Melissa
Hill
-
Drzewi
;
Regina Miller
;
Kenneth S. Santone
;
Arun Senapati
;
Eric E. Shields
;
Digavalli V. Sivarao
;
Ryan Westphal
;
Valerie J. Whiterock
;
Xiaoliang Zhuo
;
Joanne J. Bronson
;
John E. Macor
关键词:
mGluR5
;
PAMs
;
Cognition
;
Schizophrenia
;
Bioactivation
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
2.
SAR studies of non-zinc-chelating MMP-13 inhibitors: Improving selectivity and metabolic stability
作者:
Donghong Amy Gao
;
Zhaoming Xiong
;
Alex
;
er Heim-Riether
;
Laura Amodeo
;
E. Michael August
;
Xianhua Cao
;
Leonard Ciccarelli
;
Br
;
on K. Collins
;
Kyle Harrington
;
Kathleen Haverty
;
Melissa
Hill
-
Drzewi
;
Xian
关键词:
MMP-13
;
Non-Zn-chelating inhibitor
;
SAR
;
Selectivity
;
Metabolic stability
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
3.
Improving potency and selectivity of a new class of non-Zn-chelating MMP-13 inhibitors
作者:
Alex
;
er Heim-Riether
;
Steven J. Taylor
;
Shuang Liang
;
Donghong Amy Gao
;
Zhaoming Xiong
;
E. Michael August
;
Br
;
on K. Collins
;
Bennett T. Farmer II
;
Kathleen Haverty
;
Melissa
Hill
-
Drzewi
;
Hans-Dieter Ju
关键词:
MMP-13
;
Non-Zn-chelating inhibitor
;
SAR
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
1
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