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Wiley电子期刊(47)	NATURE电子期刊(5)	ACS电子期刊(580)
SpringerLink电子期刊(212)	Elsevier电子期刊(1472)

在“Elsevier电子期刊”中，命中：1,472条，耗时：0.0709668 秒

在所有数据库中总计命中：2,316条

1.Synthesis and antiproliferative activity of monocationic arylthiophene derivatives

作者：Mohamed A. Ismail^a ; ^b ; ^{ismail_158@yahoo.com} ; ^{mismail@mans.edu.eg} ; Magdy M. Youssef^a ; ^b ; Reem K. Arafa^c ; Shar S. Al-Shihry^a ; Wael M. El-Sayed^d ; ^{waelelhalawany@hotmail.com} ; ^{wael_farag@sci.asu.edu.eg}

关键词：Monocationic arylthiophenes ; Suzuki coupling ; Antiproliferative activity ; DNA affinity ; tyrosine kinase inhibition

刊名：European Journal of Medicinal Chemistry

出版年：2017

2.New derivatives of 7-chloroquinolin-4-amine with antiprotozoal activity

作者：Johanna Faist^a ; ^{johanna.faist@uni-graz.at} ; Clemens Hinteregger^a ; Werner Seebacher^a ; Robert Saf^b ; Pascal Mä ; ser^c ; Marcel Kaiser^c ; Robert Weis^a

关键词：Amines ; Antiplasmodial activity ; Heterocycles ; NMR spectroscopy ; Nucleophilic substitutions ; Quinoline

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

3.Novel dabigatran derivatives with a fluorine atom at the C-2 position of the terminal benzene ring: Design, synthesis and anticoagulant activity evaluation

作者：Haoran Yang ; Qianqian Liu ; Xiaodong Gao ; Yujie Ren ; ^{clab@sit.edu.cn} ; Yonghong Gao

关键词：Anticoagulant activity ; Fluorinated dabigatran derivatives ; Molecular docking ; Synthesis

刊名：European Journal of Medicinal Chemistry

出版年：2017

4.Synthesis, characterization and antineoplastic activity of bis-aziridinyl dimeric naphthoquinone - A novel class of compounds with potent activity against acute myeloid leukemia cells

作者：Brandon A. Carter-Cooper^a ; Steven Fletcher^b ; Dana Ferraris^c ; Eun Yong Choi^a ; Dahlia Kronfli^a ; Smaraki Dash^a ; Phuc Truong^c ; Edward A. Sausville^a ; Rena G. Lapidus^a ; Ashkan Emadi^a ; ^{aemadi@umm.edu}

关键词：Naphthoquinone ; Acute myeloid leukemia ; DNA damage ; Reactive oxygen species ; Aziridine

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

5.Discovery of new nanomolar inhibitors of GPa: Extension of 2-oxo-1,2-dihydropyridinyl-3-yl amide-based GPa inhibitors

作者：Wendy A. Loughlin^a ; ^{w.loughlin@griffith.edu.au} ; Ian D. Jenkins^b ; N. David Karis^b ; Peter C. Healy^a ; ^c

关键词：Glycogen phosphorylase inhibitors ; Pyridone amides ; Dimer ; Structure activity relationship ; Type 2 diabetes

刊名：European Journal of Medicinal Chemistry

出版年：2017

6.Syntheses and antibacterial activity of soluble 9-bromo substituted indolizinoquinoline-5,12-dione derivatives

作者：Hui Yang^a ; ¹ ; Hao-Wen Wang^a ; ¹ ; Teng-Wei Zhu^a ; ¹ ; Le-Mao Yu^a ; Jian-Wen Chen^a ; Lu-Xia Wang^b ; Lei Shi^b ; Ding Li^a ; Lian-Quan Gu^a ; Zhi-Shu Huang^a ; Lin-Kun An^a ; ^{lssalk@mail.sysu.edu.cn}

关键词：Indolizinoquinolinedione ; Quinone ; Antibacterial ; Methicillin-resistant Staphylococcus aureus ; Multi-drug resistance

刊名：European Journal of Medicinal Chemistry

出版年：2017

7.Design, synthesis and biological evaluation of alkylamino biphenylamides as Hsp90 C-terminal inhibitors

作者：Gaurav Garg ; Huiping Zhao ; Brian S.J. Blagg ; ^{bblagg@ku.edu}

关键词：Heat shock protein 90 ; Hsp90 C-terminal inhibitors ; Alkylamino biphenylamides ; Structure-activity relationship ; Breast cancer

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

8.Structure-activity relationship studies on a Trp dendrimer with dual activities against HIV and enterovirus A71. Modifications on the amino acid

作者：Belé ; n Martí ; nez-Gualda^a ; Liang Sun^b ; Eva Rivero-Buceta^a ; ¹ ; Aida Flores^a ; ² ; Ernesto Quesada^a ; Jan Balzarini^b ; Sam Noppen^b ; Sandra Liekens^b ; Dominique Schols^b ; Johan Neyts^b ; Pieter Leyssen^b ; Carmen Mirabelli^b ; Marí ; a-José ; Camarasa^a ; Ana San-Fé ; lix^a ; ^{anarosa@iqm.csic.es}

关键词：Antiviral agents ; AIDS ; HFMD ; HIV ; EV71 ; Tryptophan

刊名：Antiviral Research

出版年：2017

9.5-Substituted-benzylsulfanyl-thiophene-2-sulfonamides with effective carbonic anhydrase inhibitory activity: Solution and crystallographic investigations

作者：Jekaterīna Ivanova^a ; ^b ; Agnese Balode^a ; ^b ; Raivis Žalubovskis^a ; ^{raivis@osi.lv} ; Janis Leitans^c ; Andris Kazaks^c ; Daniela Vullo^d ; Kaspars Tars^c ; ^e ; Claudiu T. Supuran^f ; ^{claudiu.supuran@unifi.it}

关键词：Carbonic anhydrase ; Thiophene-2-sulfonamide ; Mercaptan ; Inhibitor

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

10.Structural optimization of diphenylpyrimidine derivatives (DPPYs) as potent Bruton's tyrosine kinase (BTK) inhibitors with improved activity toward B leukemia cell lines

作者：Dan Zhao^a ; Shanshan Huang^a ; Menghua Qu^a ; Changyuan Wang^a ; Zhihao Liu^a ; Zhen Li^a ; Jinyong Peng^a ; Kexin Liu^a ; Yanxia Li^b ; Xiaodong Ma^a ; ^{xiaodong.ma@139.com} ; Xiaohong Shu^a ; ^{xiaohong_shu@dmu.edu.cn}

关键词：Leukemia ; BTK ; Pyrimidine ; Synthesis ; Inhibitor

刊名：European Journal of Medicinal Chemistry

出版年：2017

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