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SpringerLink电子期刊(2)
Elsevier电子期刊(6)
ACS电子期刊(8)
在“
Elsevier电子期刊
”中,
命中:
6
条,耗时:0.0409815 秒
在所有数据库中总计命中:
16
条
1.
Design, synthesis, and biological activity of novel, potent, and highly selective fused pyrimidine-2-carboxamide-4-one-based matrix metalloproteinase (MMP)-13 zinc-binding inhibitors
作者:
Hiroshi Nara
;
Kenjiro Sato
;
Akira Kaieda
;
Hideyuki Oki
;
Haruhiko Kuno
;
Takashi Santou
;
Naoyuki
Kanzaki
;
Jun Terauchi
;
Osamu Uchikawa
;
Masakuni Kori
关键词:
Matrix metalloproteinase
;
MMP-13
;
Fused pyrimidine-2-carboxamide
;
Zinc-binding group
;
Structure-based drug design
;
Osteoarthritis
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
2.
Design, synthesis, and biological evaluation of 3-aryl-3-hydroxy-1-phenylpyrrolidine derivatives as novel androgen receptor antagonists
作者:
Satoshi Yamamoto
;
satoshi.yamamoto@takeda.com
;
Hiromi Kobayashi
;
Tomohiro Kaku
;
Katsuji Aikawa
;
Takahito Hara
;
Masuo Yamaoka
;
Naoyuki
Kanzaki
;
Atsushi Hasuoka
;
Atsuo Baba
;
Mitsuhiro Ito
关键词:
PC
;
prostate cancer
;
AR
;
androgen receptor
;
CRPC
;
castration-resistant prostate cancer
;
CAB
;
combined androgen blockade
;
PSA
;
prostate-specific antigen
;
DHT
;
dihydrotestosterone
;
SAR
;
structure&ndash
;
activity relationship
;
EDC
;
N-[3-(dimethylamino)propyl]
刊名:Bioorganic and Medicinal Chemistry
出版年:2013
3.
Novel triple reuptake inhibitors with low risk of CAD associated liabilities: Design, synthesis and biological activities of 4-[(1S)-1-(3,4-dichlorophenyl)-2-methoxyethyl]piperidine and related compounds
作者:
Yuji Ishichi
;
Eiji Kimura
;
Eiji Honda
;
Masato Yoshikawa
;
Takashi Nakahata
;
Yasuko Terao
;
Atsuko Suzuki
;
Takayuki Kawai
;
Yuuichi Arakawa
;
Hiroyuki Ohta
;
Naoyuki
Kanzaki
;
Hideyuki Nakagawa
;
Jun Terauchi
关键词:
Monoamine reuptake inhibition
;
Piperidine compounds
;
Cationic amphiphilic drug (CAD)
;
CYP2D6
;
hERG
;
PLsis
;
Tail suspension test
;
Antidepressant
刊名:Bioorganic and Medicinal Chemistry
出版年:2013
4.
Seasonal and spatial variation of nitrogen dynamics in the litter and surface soil layers on a tropical dry evergreen forest slope
作者:
Naoyuki
Yamashita
;
Seiichi Ohta
;
Hiroyuki Sase
;
Jesada Luangjame
;
Thiti Visaratana
;
Bopit Kievuttinon
;
Hathairatana Garivait
;
Mamoru
Kanzaki
关键词:
Tropical dry forest
;
Nitrogen dynamics
;
Nitrate leaching
;
Ion exchange resin
;
Litterfall
刊名:Forest Ecology and Management
出版年:2010
5.
Orally active CCR5 antagonists as anti-HIV-1 agents. Part 3: Synthesis and biological activities of 1-benzazepine derivatives containing a sulfoxide moiety
作者:
Seto
;
Masaki
;
Miyamoto
;
Naoki
;
Aikawa
;
Katsuji
;
Aramaki
;
Yoshio
;
Kanzaki
;
Naoyuki
;
Iizawa
;
Yuji
;
et. al.
关键词:
CCR5 antagonist
;
HIV-1
;
Sulfoxide
;
S-isomer
;
1-Benzazepine
刊名:Bioorganic and Medicinal Chemistry
出版年:2005
6.
T140 analogs as CXCR4 antagonists identified as anti-metastatic agents in the treatment of breast cancer
作者:
Tamamura
;
Hirokazu
;
Hori
;
Akira
;
Kanzaki
;
Naoyuki
;
Hiramatsu
;
Kenichi
;
Mizumoto
;
Makiko
;
Nakashima
;
Hideki
;
et. al.
关键词:
CXCR4 antagonist
;
Pulmonary metastasis
;
T140
;
Breast cancer
刊名:FEBS Letters
出版年:2003
1
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作者(6)
按出版年细分(6)
2016年(1)
2013年(2)
2010年(1)
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2003年(1)
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