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SpringerLink电子期刊(1)
Elsevier电子期刊(20)
ACS电子期刊(1)
在“
Elsevier电子期刊
”中,
命中:
20
条,耗时:小于0.01 秒
在所有数据库中总计命中:
22
条
1.
Discovery of novel phenethylpyridone derivatives as potent melanin-concentrating hormone 1 receptor antagonists
作者:
Makoto Ando
;
Etsuko Sekino
;
Yuji Haga
;
Minoru Moriya
;
Masahiko Ito
;
Junko Ito
;
Hisashi Iwaasa
;
Akane Ishihara
;
Akio Kanatani
;
Norikazu
Ohtake
关键词:
Melanin-concentrating hormone 1 receptor antagonist
;
Phenethylpyridone
;
Anti-obesity
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
2.
Discovery of pyridone-containing imidazolines as potent and selective inhibitors of neuropeptide Y Y5 receptor
作者:
Makoto Ando
;
Nagaaki Sato
;
Tsuyoshi Nagase
;
Keita Nagai
;
Shiho Ishikawa
;
Hirobumi Takahashi
;
Norikazu
Ohtake
;
Junko Ito
;
Mioko Hirayama
;
Yuko Mitobe
;
Hisashi Iwaasa
;
Akira Gomori
;
Hiroko Matsushita
;
K
关键词:
Neuropeptide Y Y5 receptor
;
Anti-obesity
;
Y5 antagonist
;
Imidazoline class
刊名:Bioorganic and Medicinal Chemistry
出版年:2009
3.
Melanin-concentrating hormone 1-receptor antagonist suppresses body weight gain correlated with high receptor occupancy levels in diet-induced obesity mice
作者:
Masahiko Ito
;
Akane Ishihara
;
Akira Gomori
;
Shinichiro Egashira
;
Hiroko Matsushita
;
Satoshi Mashiko
;
Junko Ito
;
Makoto Ito
;
Kazuho Nakase
;
Yuji Haga
;
Hisashi Iwaasa
;
Takao Suzuki
;
Norikazu
Ohtake
;
Min
关键词:
Melanin-concentrating hormone 1-receptor Antagonist
;
Receptor occupancy
;
Obesity
刊名:European Journal of Pharmacology
出版年:2009
4.
Syntheses and structure–activity relationships of novel, potent, and selective trans
作者:
Yoshio Ogino
;
Norikazu
Ohtake
;
Yoshikazu Nagae
;
Kenji Matsuda
;
Makoto Ishikawa
;
Minoru Moriya
;
Maki Kanesaka
;
Yuko Mitobe
;
Junko Ito
;
Tetsuya Kanno
;
Akane Ishihara
;
Hisashi Iwaasa
;
Tomoyuki Ohe
;
Akio
关键词:
Neuropeptide Y
;
Y5 receptor
;
Antagonist
;
Anti-obesity
;
Benzimidazole
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2008
5.
Design, syntheses, and structure–activity relationships of novel NPY Y5 receptor antagonists: 2-{3-Oxospiro[isobenzofuran-1(3H
作者:
Yoshio Ogino
;
Norikazu
Ohtake
;
Yoshikazu Nagae
;
Kenji Matsuda
;
Minoru Moriya
;
Takuya Suga
;
Makoto Ishikawa
;
Maki Kanesaka
;
Yuko Mitobe
;
Junko Ito
;
Tetsuya Kanno
;
Akane Ishihara
;
Hisashi Iwaasa
;
Tomoyu
关键词:
Neuropeptide Y
;
Y5 receptor
;
Antagonist
;
Anti-obesity
;
Benzimidazole
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2008
6.
Structure–activity relationships of a novel class of endothelin receptor selective antagonists; 6-carboxy-2-isopropylamino-5,7-diarylcyclopenteno[1,2-b]pyridines
作者:
Takahashi
;
Hirobumi
;
Ohtake
;
Norikazu
;
Sakamoto
;
Toshihiro
;
Iino
;
Tomoharu
;
Kawanishi
;
Nobuhiko
;
et. al.
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2004
7.
Potent and orally active ET
A
selective antagonists with 5,7-diarylcyclopenteno[1,2-b]pyridine-6-carboxylic acid structures
作者:
Yoshizumi
;
Takashi
;
Takahashi
;
Hirobumi
;
Ohtake
;
Norikazu
;
Jona
;
Hideki
;
Sato
;
Yoshiyuki
;
Kishino
;
Hiroyuki
;
et. al.
刊名:Bioorganic and Medicinal Chemistry
出版年:2004
8.
N-
Acyl 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline: The first orexin-2 receptor selective non-peptidic antagonist
作者:
Hirose
;
Masaaki
;
Egashira
;
Shin-ichiro
;
Goto
;
Yasuhiro
;
Hashihayata
;
Takashi
;
Ohtake
;
Norikazu
;
et. al.
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2003
9.
Muscarinic M
3
receptor antagonists with (2R)-2-[(1R)-3,3-Difluorocyclopentyl]-2-hydroxyphenylacetamide Structures. Part 2
作者:
Ogino
;
Yoshio
;
Ohtake
;
Norikazu
;
Kobayashi
;
Kensuke
;
Kimura
;
Toshifumi
;
Fujikawa
;
Toru
;
Hasegawa
;
Takuro
;
et. al.
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2003
10.
N-Acyl 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline: The first orexin-2 receptor selective non-peptidic antagonist
作者:
Hirose
;
Masaaki
;
Egashira
;
Shin-ichiro
;
Goto
;
Yasuhiro
;
Hashihayata
;
Takashi
;
Ohtake
;
Norikazu
;
et. al.
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2003
1
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