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Wiley电子期刊(2)
NATURE电子期刊(1)
ACS电子期刊(11)
SpringerLink电子期刊(13)
Elsevier电子期刊(115)
在“
Elsevier电子期刊
”中,
命中:
115
条,耗时:小于0.01 秒
在所有数据库中总计命中:
142
条
1.
Novel Zebrafish EAE model: A quick in vivo screen for multiple sclerosis
作者:
Pushkar Kulkarni
a
;
b
;
1
;
pushkark@drils.org
;
kk.pushkar@gmail.com
;
Swapna Yellanki
b
;
1
;
Raghavender Medishetti
b
;
Dharmarajan Sriram
a
;
Uday Saxena
b
;
c
;
Perumal
Yogeeswari
a
;
pyogee@hyderabad.bits-pilani.ac.in
;
pyogee.sriram@gmail.com
关键词:
Zebrafish
;
Experimental autoimmune encephalomyelitis (EAE)
;
Multiple Sclerosis (MS)
;
Myelin oligodendrocyte glycoprotein (MOG)
;
Fingolimod (Gilenya)
;
Drug Discovery
刊名:Multiple Sclerosis and Related Disorders
出版年:2017
2.
Design, development of new synthetic methodology, and biological evaluation of substituted quinolines as new anti-tubercular leads
作者:
Babita Tanwar
a
;
Asim Kumar
a
;
Perumal
Yogeeswari
b
;
Dharmarajan Sriram
b
;
Asit K. Chakraborti
a
;
akchakraborti@niper.ac.in
关键词:
Anti-mycobacterial agents
;
Substituted quinolines
;
New synthetic methodology
;
Water
;
DBSA
;
Catalyst
;
Structural activity relationship
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
3.
Engineering another class of anti-tubercular lead: Hit to lead optimization of an intriguing class of gyrase ATPase inhibitors
作者:
Variam Ullas Jeankumar
1
;
Rudraraju Srilakshmi Reshma
1
;
Rahul Vats
;
Renuka Janupally
;
Shalini Saxena
;
Perumal
Yogeeswari
;
Dharmarajan Sriram
;
dsriram@hyderabad.bits-pilani.ac.in" class="auth_mail" title="E-mail the corresponding author
关键词:
Medium throughput virtual screening
;
Mycobacterium tuberculosis
;
DNA gyrase
;
Differential scanning fluorimetry
刊名:European Journal of Medicinal Chemistry
出版年:2016
4.
Synthesis and antimycobacterial screening of new N-(4-(5-aryl-3-(5-methyl-1,3,4-oxadiazol-2-yl)-1H-pyrazol-1-yl)phenyl)-4-amide derivatives
作者:
Nagabhushana Nayak
a
;
Jurupula Ramprasad
a
;
Udayakumar Dalimba
a
;
udayaravi80@gmail.com" class="auth_mail" title="E-mail the corresponding author
;
Perumal
Yogeeswari
b
;
Dharmarajan Sriram
b
关键词:
Pyrazole-oxadiazole hybrids
;
Antitubercular activity
;
SC-XRD analysis
;
In vitro cytotoxicity
刊名:Chinese Chemical Letters
出版年:2016
5.
Click-based synthesis and antitubercular evaluation of novel dibenzo[b,d]thiophene-1,2,3-triazoles with piperidine, piperazine, morpholine and thiomorpholine appendages
作者:
Lokesh Pulipati
a
;
Perumal
Yogeeswari
b
;
Dharmarajan Sriram
b
;
Srinivas Kantevari
a
;
c
;
kantevari@yahoo.com" class="auth_mail" title="E-mail the corresponding author
;
kantevari@gmail.com" class="auth_mail" title="E-mail the corresponding author
关键词:
Dibenzothiophene
;
Triazole
;
Piperidine
;
Piperazine
;
Antitubercular agents
;
Click chemistry
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
6.
Anti-tubercular activities of 5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidin-4-amine analogues endowed with high activity toward non-replicative Mycobacterium tuberculosis
作者:
Ganesh Samala
;
Parthiban Brindha Devi
;
Shalini Saxena
;
Saritha Gunda
;
Perumal
Yogeeswari
;
Dharmarajan Sriram
;
dsriram@hyderabad.bits-pilani.ac.in" class="auth_mail" title="E-mail the corresponding author
关键词:
Tuberculosis
;
Dormant tuberculosis
;
l-Alanine dehydrogenase
;
Tetrahydrobenzo[4
;
5]thieno[2
;
3-d]pyrimidin-4-amine analogues
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
7.
Design, synthesis and biological evaluation of imidazo[2,1-b]thiazole and benzo[d]imidazo[2,1-b]thiazole derivatives as Mycobacterium tuberculosis pantothenate synthetase inhibitors
作者:
Ganesh Samala
;
Parthiban Brindha Devi
;
Shalini Saxena
;
Nikhila Meda
;
Perumal
Yogeeswari
;
Dharmarajan Sriram
;
dsriram@hyderabad.bits-pilani.ac.in" class="auth_mail" title="E-mail the corresponding author
关键词:
Tuberculosis
;
Pantothenate synthetase
;
Imidazo[2
;
1-b]thiazole
;
Benzo[d]imidazo[2
;
1-b]thiazole
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
8.
Replacement of cardiotoxic aminopiperidine linker with piperazine moiety reduces cardiotoxicity? Mycobacterium tuberculosis novel bacterial topoisomerase inhibitors
作者:
Karyakulam Andrews Bobesh
a
;
&dagger
;
;
Janupally Renuka
a
;
&dagger
;
;
Rudraraju Reshma Srilakshmi
a
;
Swapna Yellanki
b
;
c
;
Pushkar Kulkarni
b
;
c
;
Perumal
Yogeeswari
a
;
Dharmarajan Sriram
a
;
dsriram@hyderabad.bits-pilani.ac.in" class="auth_mail" title="E-mail the corresponding author
关键词:
DNA gyrase
;
Topoisomerase
;
Tuberculosis
;
1
;
5-Naphthyridin-2(1H)-one
;
zERG toxicity
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
9.
Synthesis of new spirooxindole derivatives through 1,3-dipolar cycloaddition of azomethine ylides and their antitubercular activity
作者:
Fadwa Rouatbi
a
;
Moheddine Askri
a
;
moheddine.askri@fsm.rnu.tn" class="auth_mail" title="E-mail the corresponding author
;
Frederic Nana
b
;
Gilbert Kirsch
b
;
Dharmarajan Sriram
c
;
Perumal
Yogeeswari
c
关键词:
(E
;
E)-1
;
3-Bis(arylidene)indan-2-one
;
1
;
3-Dipolar cycloaddition
;
Azomethine ylide
;
Mycobacterium tuberculosis
刊名:Tetrahedron Letters
出版年:2016
10.
Synthesis, biological evaluation and structure-activity relationship of 2-styrylquinazolones as anti-tubercular agents
作者:
Pradeep S. Jadhavar
a
;
Tejas M. Dhameliya
a
;
Maulikkumar D. Vaja
a
;
Dinesh Kumar
a
;
Jonnalagadda Padma Sridevi
b
;
Perumal
Yogeeswari
b
;
Dharmarajan Sriram
b
;
Asit K. Chakraborti
a
;
akchakraborti@niper.ac.in" class="auth_mail" title="E-mail the corresponding author
;
akchakraborti@rediffmail.com" class="auth_mail" title="E-mail the corresponding author
关键词:
Tuberculosis
;
2-Styrylquinazolone
;
Anti-TB agents
;
H37Rv strain
;
SAR
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
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