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内部出版物
Wiley电子期刊(1)
SpringerLink电子期刊(5)
Elsevier电子期刊(62)
ACS电子期刊(4)
在“
Elsevier电子期刊
”中,
命中:
62
条,耗时:0.0419777 秒
在所有数据库中总计命中:
72
条
1.
Discovery of a potent and dissociated non-steroidal glucocorticoid
receptor
agonist containing an alkyl carbinol pharmacophore
作者:
Hossein Razavi
a
;
hossein.razavi@boehringer-ingelheim.com" class="auth_mail
;
Doris Riether
a
;
Christian Harcken
b
;
Jö
;
rg Bentzien
a
;
Roger M. Dinallo
a
;
Donald Souza
b
;
Richard M. Nelson
a
;
Alison Kukulka
a
;
Tazmeen N. Fadra-Khan
a
;
Edward J. Pack Jr.
a
;
Ljiljana Zuvela-Jelaska
b
;
Josephine Pelletier
b
;
Mark Panzenbeck
b
;
Carol A. Torcellini
b
;
John R. Proudfoot
a
;
Gerald H. Nabozny
b
;
David S. Thomson
a
关键词:
Nuclear hormone
receptor
s
;
Glucocorticoids
;
Non-steroidal
;
Dissociated
;
Agonist
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:15 April, 2014
2.
Evolution of hormone
selectivity
in glucocorticoid and mineralocorticoid
receptor
s
作者:
Michael E. Baker
;
John W. Funder
;
Stephanie R. Kattoula
关键词:
Corticosteroid
receptor
evolution
;
Mineralocorticoid
receptor
;
Glucocorticoid
receptor
;
Lamprey
;
Sharks
;
Coelacanths
;
Helix 3&ndash
;
helix 5 contact
刊名:The Journal of Steroid Biochemistry and Molecular Biology
出版年:2013
3.
Role of phosphorylation in
progesterone
receptor
signaling and specificity
作者:
Christy R. Hagan
;
Andrea R. Daniel
;
Gwen E. Dressing
;
Carol A. Lange
;
Lange047@umn.edu
关键词:
Progesterone
receptor
;
Phosphorylation
;
Breast cancer
;
Promoter
selectivity
;
Growth factors
;
Kinase
刊名:Molecular and Cellular Endocrinology
出版年:2012
4.
Design, synthesis, and structure-activity relationships of dihydrofuran-2-one and dihydropyrrol-2-one derivatives as novel benzoxazin-3-one-based mineralocorticoid
receptor
antagonists
作者:
Tomoaki Hasui
;
Taiichi Ohra
;
Norio Ohyabu
;
Kouhei Asano
;
Hideki Matsui
;
Atsushi Mizukami
;
Noriyuki Habuka
;
Satoshi Sogabe
;
Satoshi Endo
;
Christopher S. Siedem
;
Tony P. Tang
;
Cass
;
ra Gauthier
;
Lisa A. De Meese
;
Steven A. Boyd
;
Shoji Fukumoto
关键词:
Mineralocorticoid
receptor
;
MR
;
Nonsteroidal
;
Aldosterone
刊名:Bioorganic and Medicinal Chemistry
出版年:2013
5.
Substituted phenyl as a steroid A-ring mimetic: Providing agonist activity to a class of arylsulfonamide nonsteroidal glucocorticoid ligands
作者:
Darren DiSalvo
;
Daniel Kuzmich
;
J枚rg Bentzien
;
John Regan
;
Alison Kukulka
;
Tazmeen Fadra-Khan
;
Richard Nelson
;
Christian Harcken
;
David Thomson
;
Gerald Nabozny
关键词:
Glucocorticoids
;
Glucocorticoid
receptor
;
Nuclear hormone
receptor
;
Mineralocorticoid
receptor
;
Progesterone
receptor
;
Glucocorticoid
receptor
agonist
;
Arylsulfonamide
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:15 December, 2013
6.
Aromatic β-amino-ketone derivatives as novel selective non-steroidal
progesterone
receptor
antagonists
作者:
Yongli Du
;
Qunyi Li
;
Bing Xiong
;
Xin Hui
;
Xin Wang
;
Yang Feng
;
Tao Meng
;
Dingyu Hu
;
Datong Zhang
;
Mingwei Wang
;
Jingkang Shen
关键词:
Progesterone
receptor
(PR)
;
Progesterone
receptor
antagonist
;
Non-steroidal
progesterone
receptor
antagonist
;
Aromatic β
;
-amino-ketone
;
Mannich reaction
刊名:Bioorganic and Medicinal Chemistry
出版年:2010
7.
Signaling inputs to
progesterone
receptor
gene regulation and promoter
selectivity
作者:
Andrea R. Daniel
;
Todd P. Knutson
;
Carol A. Lange
关键词:
Progesterone
receptor
(PR)
;
Phosphorylation
;
Sumoylation
;
Promoter
selectivity
;
Transcription
刊名:Molecular and Cellular Endocrinology
出版年:2009
8.
Synthesis and biological effect of halogen substituted phenyl acetic acid derivatives of
progesterone
as potent
progesterone
receptor
antagonists
作者:
Marisa Cabeza
;
Eugene Bratoeff
;
Georgina Gó
;
mez
;
Ivonne Heuze
;
Arely Rojas
;
Martha Ochoa
;
Miguel Angel Palomino
;
Cristina Revilla
关键词:
Novel 5-halogen phenyl acidic derivatives of
progesterone
;
Progesterone
receptor
selectivity
;
Anti-progestin effect
;
Inhibitors of ovulation
;
Antagonist of the
progesterone
receptor
s
刊名:The Journal of Steroid Biochemistry and Molecular Biology
出版年:2008
9.
Selectivity
and potency of the retro
progesterone
dydrogesterone in vitro
作者:
Tea Laniš
;
nik Riž
;
ner
a
;
Petra Brož
;
ič
;
a
;
Christopher Doucette
b
;
Tammy Turek-Etienne
b
;
Ursula Mü
;
ller-Vieira
c
;
Edwin Sonneveld
d
;
1
;
Bart van der Burg
d
;
Christiane Bö
;
cker
e
;
Bettina Husen
e
;
Bettina.Husen@abbott.com
关键词:
Dydrogesterone
;
Steroid
receptor
s
;
Pre-
receptor
metabolism
;
17β
;
-Hydroxysteroid dehydrogenase type 5 (AKR1C3)
;
17β
;
-Hydroxysteroid dehydrogenase type 3
;
5α
;
-Reductase type 2
刊名:Steroids
出版年:2011
10.
Synthesis and antihormonal properties of novel 11¦Â-benzoxazole-substituted steroids
作者:
Chunyang Jin
;
cjin@rti.org
;
Scott E. Fix
;
John A. Kepler
;
C. Edgar Cook
?/sup>
关键词:
Glucocorticoid
receptor
;
Progesterone
receptor
;
Antagonist
;
11¦Â-Arylsteroids
;
Mifepristone
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2012
1
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3
4
5
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