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在“
Elsevier电子期刊
”中,
命中:
666
条,耗时:0.0289876 秒
在所有数据库中总计命中:
1,202
条
1.
Design and synthesis of new RAF kinase-inhibiting antiproliferative
quinoline
derivatives
. Part 2: Diarylurea
derivatives
作者:
Mohammed I. El-Gamal
a
;
b
;
c
;
Mohammad Ashrafuddin Khan
d
;
e
;
Hamadeh Tarazi
a
;
b
;
Mohammed S. Abdel-Maksoud
d
;
e
;
f
;
Mahmoud M. Gamal El-Din
d
;
e
;
f
;
Kyung Ho Yoo
g
;
Chang-Hyun Oh
d
;
e
;
choh@kist.re.kr
关键词:
Antiproliferative activity
;
C-RAF kinase
;
Diarylurea
;
Molecular docking
;
Quinoline
刊名:European Journal of Medicinal Chemistry
出版年:2017
2.
N-(2-(arylmethylimino)ethyl)-7-chloroquinolin-4-amine
derivatives
, synthesized by thermal and ultrasonic means, are endowed with anti-Zika virus activity
作者:
Giselle Barbosa-Lima
a
;
b
;
c
;
1
;
Ligia S. da Silveira Pinto
d
;
1
;
Carlos R. Kaiser
d
;
James L. Wardell
e
;
f
;
Caroline S. De Freitas
a
;
b
;
Yasmine R. Vieira
a
;
b
;
c
;
Andressa Marttorelli
a
;
b
;
José
;
Cerbino Neto
c
;
Patrí
;
cia T. Bozza
a
;
Solange M.S.V. Wardell
g
;
Marcus V.N. de Souza
d
;
e
;
2
;
marcos_souza@far.fiocruz.br
;
Thiago M.L. Souza
a
;
b
;
c
;
2
关键词:
Zika virus
;
Quinoline
derivatives
;
Sonochemical method
刊名:European Journal of Medicinal Chemistry
出版年:2017
3.
Synthesis, identification and in vitro biological evaluation of some novel
quinoline
incorporated 1,3-thiazinan-4-one
derivatives
作者:
S. Umamatheswari
a
;
C. Sankar
b
;
sankschem@gmail.com
关键词:
Tuberculosis
;
Quinoline
;
Thiazinan-4-one
;
Antimalarial
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
4.
Molecular docking, discovery, synthesis, and pharmacological properties of new 6-substituted-2-(3-phenoxyphenyl)-4-phenyl
quinoline
derivatives
; an approach to developing potent DNA gyrase inhibitors/antibacterial agents
作者:
Manikandan Alagumuthu
;
Sivakumar Arumugam
;
mailtomicromani@gmail.com
关键词:
Phenoxyphenyl
quinoline
s
;
Antibacterial
;
DNA gyrase A
;
Molecular docking
;
Drug discovery
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
5.
New quinolinic
derivatives
as melatonergic ligands: Synthesis and pharmacological evaluation
作者:
Elodie Landagaray
a
;
1
;
Mohamed Ettaoussi
a
;
1
;
m.ettaoussi@yahoo.fr
;
Marouan Rami
a
;
Jean A. Boutin
b
;
Daniel-Henri Caignard
c
;
Philippe Delagrange
c
;
Patricia Melnyk
a
;
d
;
Pascal Berthelot
a
;
d
;
Saï
;
d Yous
a
;
d
;
said.yous@univ-lille2.fr
关键词:
Melatonin
;
Quinoline
derivatives
;
MT1
;
MT2-Selectivity
;
Agonist
刊名:European Journal of Medicinal Chemistry
出版年:2017
6.
New
derivatives
of 7-chloroquinolin-4-amine with antiprotozoal activity
作者:
Johanna Faist
a
;
johanna.faist@uni-graz.at
;
Clemens Hinteregger
a
;
Werner Seebacher
a
;
Robert Saf
b
;
Pascal Mä
;
ser
c
;
Marcel Kaiser
c
;
Robert Weis
a
关键词:
Amines
;
Antiplasmodial activity
;
Heterocycles
;
NMR spectroscopy
;
Nucleophilic substitutions
;
Quinoline
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
7.
Synthesis, characterization, and in vitro SAR evaluation of N,N′-bis(arylmethyl)-C
2
-alkyl substituted imidazolium salts
作者:
Michael A. DeBord
;
Patrick O. Wagers
;
Steven R. Crabtree
;
Claire A. Tessier
;
Matthew J. Panzner
;
mjp9@uakron.edu
;
Wiley J. Youngs
;
youngs@uakron.edu
关键词:
Imidazolium salt
;
Anti-cancer
;
Anti-tumor
;
Non-small cell lung cancer
;
Quinoline
;
Naphthalene
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
8.
New donor-acceptor-donor molecules based on
quinoline
acceptor unit with Schiff base bridge: synthesis and characterization
作者:
Sonia Kotowicz
a
;
Mariola Siwy
b
;
Michal Filapek
a
;
Jan G. Malecki
a
;
Karolina Smolarek
c
;
Justyna Grzelak
c
;
Sebastian Mackowski
c
;
Aneta Slodek
a
;
aneta.slodek@us.edu.pl
;
a.slodek@wp.pl
;
Ewa Schab-Balcerzak
a
;
b
;
ewa.schab-balcerzak@us.edu.pl
;
ebalcerzak@cmpw-pan.edu.pl
关键词:
Quinolone
derivatives
;
Schiff bases
;
Bithiophene
;
Donor-acceptor-donor
;
Plasmonic enhancement
刊名:Journal of Luminescence
出版年:2017
9.
2,8-bis(trifluoromethyl)
quinoline
analogs show improved anti-Zika virus activity, compared to mefloquine
作者:
Giselle Barbosa-Lima
a
;
b
;
c
;
Adriana M. Moraes
d
;
e
;
Adriele da S. Araú
;
jo
d
;
Emerson T. da Silva
d
;
Caroline S. de Freitas
a
;
b
;
Yasmine R. Vieira
a
;
b
;
c
;
Andressa Marttorelli
a
;
b
;
José
;
Cerbino Neto
c
;
Patrí
;
cia T. Bozza
a
;
Marcus V.N. de Souza
d
;
e
;
marcos_souza@far.fiocruz.br
;
Thiago Moreno. L. Souza
a
;
b
;
c
关键词:
Zika virus
;
Quinoline
derivatives
;
Mefloquine
;
Antiviral
刊名:European Journal of Medicinal Chemistry
出版年:2017
10.
Design, synthesis and biological evaluation of 7-(aryl)-2,3-dihydro-[1,4]dioxino[2,3-g]
quinoline
derivatives
as potential Hsp90 inhibitors and anticancer agents
作者:
Sina Omid Malayeri
a
;
b
;
Khalil Abnous
c
;
Atefeh Arab
d
;
Maryam Akaberi
e
;
Soghra Mehri
c
;
Afshin Zarghi
f
;
Razieh Ghodsi
a
;
b
;
ghodsir@mums.ac.ir
关键词:
Quinoline
s
;
Heat Shock Protein 90
;
Anti-cancer activity
;
Her2
;
Molecular docking
;
Hsp90 inhibitor
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
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