搜索页_+Radioligand

设为首页

收藏本站

网站地图 | English | 公务邮箱

About the library

Background
History
Leadership
Organization

Readers' Guide

Opening Hours
Collections
Help Via Email

Publications

Electronic Information Resources

外文资源

Elsevier电子期刊(3351)

在“Elsevier电子期刊”中，命中：3,351条，耗时：0.0150223 秒

在所有数据库中总计命中：3,351条

1.In vivo evaluation of [¹⁸F]FECIMBI-36, an agonist 5-HT_2A/2C receptor PET radioligand in nonhuman primate

作者：Jaya Prabhakaran^a ; ^b ; Kiran Kumar Solingapuram Sai^c ; Francesca Zanderigo^a ; ^b ; Harry Rubin-Falcone^a ; Matthew J. Jorgensen^d ; Jay R. Kaplan^d ; Katharine I. Tooke^a ; Akiva Mintz^c ; J. John Mann^a ; ^b ; J.S. Dileep Kumar^b ; ^{kumardi@nyspi.columbia.edu}

关键词：5-HT ; 5-HT2A/2CR ; Agonist ; PET ; Radiotracer

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

2.Characterization of P2X4 receptor agonists and antagonists by calcium influx and radioligand binding studies

作者：Aliaa Abdelrahman^a ; Vigneshwaran Namasivayam^a ; ^c ; Sonja Hinz^a ; Anke C. Schiedel^a ; Meryem Kö ; se^a ; Maggi Burton^b ; Ali El-Tayeb^a ; ¹ ; Michel Gillard^b ; Jü ; rgen Bajorath^c ; Marc de Ryck^b ; Christa E. Mü ; ller^a ; ^{christa.mueller@uni-bonn.de}

关键词：Ap3A ; diadenosine triphosphate ; Ap4A ; diadenosine tetraphosphate ; Ap5A ; diadenosine pentaphosphate ; AR-C67085MX ; 2-propylthio-β ; γ-dichloromethylene-ATP ; PSB0412 ; 2-propargylthio-β ; γ-dichloromethylene-ATP ; 5-BDBD ; 5-(3-bromophenyl)-1 ; 3-dihydro-2H-benzofuro[3 ; 2-e]-1 ; 4-diazepin-2-one ; BzATP ; 2&prime ; (3&prime ; )-O-(4-benzoylbenzoyl)adenosine 5&prime ; -triphosphate ; CHO-K1 cells ; Chinese hamster ovary cells ; HBSS ; Hank&rsquo ; s balanced salt solution ; HEPES ; 4-(2-hydroxyethyl)-1-piperazine ethanesulfoni

刊名：Biochemical Pharmacology

出版年：2017

3.Development of [¹¹C]/[³H]THK-5351 - A potential novel carbon-11 tau imaging PET radioligand

作者：Vladimir Stepanov^a ; ^{vladimir.stepanov@ki.se} ; Marie Svedberg^a ; Zhisheng Jia^a ; Raisa Krasikova^a ; Laetitia Lemoine^b ; Nobujuki Okamura^c ; Shozo Furumoto^c ; Nicholas Mitsios^d ; Jan Mulder^d ; Bengt Lå ; ngströ ; m^e ; Agneta Nordberg^b ; Christer Halldin^a

关键词：Tau imaging ; Pet ; Carbon-11 ; Proteinopathy ; Autoradiography ; Tritium

刊名：Nuclear Medicine and Biology

出版年：2017

4.Cocaine self-administration, extinction training and drug-induced relapse change metabotropic glutamate mGlu5 receptors expression: Evidence from radioligand binding and immunohistochemistry assays

作者：Lucyna Pomierny-Chamiolo^a ; ^{lpomiern@cm-uj.krakow.pl} ; Joanna Miszkiel^b ; Malgorzata Frankowska^b ; Beata Bystrowska^a ; Malgorzata Filip^b

关键词：Cocaine self-administration ; Extinction training ; Drug-induced relapse ; MGlu5 receptor binding ; MGlu5 receptor immunohistochemistry

刊名：Brain Research

出版年：2017

5.New potent A₁ adenosine receptor radioligands for positron emission tomography

作者：Sabrina Kreft ; Dirk Bier ; ^{d.bier@fz-juelich.de} ; Marcus H. Holschbach ; Annette Schulze ; Heinz H. Coenen

关键词：CPFPX ; 8-cyclopentyl-3-(3-fluoropropyl)-1-propylxanthine ; PET ; positron-emission-tomography ; CBCPM ; 8-cyclobutyl-1-cyclopropymethyl-3-(3-fluoropropyl)xanthine ; CPMMCB ; 1-cyclopropylmethyl-3-(3-fluoropropyl)-8-(1-methylcyclobutyl)xanthine ; GPCR ; G-protein-coupled receptors ; CNS ; central nervous system ; DPCPX ; 1 ; 3-dipropyl-8-cyclopentylxanthine ; NMR ; nuclear magnetic resonance ; TLC ; thin layer chromatography ; CHO ; Chinese hamster ovary ; POM ; pivaloyloxymethyl ; DMB ; 2 ; 4-dimethoxybenzyl ; HPLC ; high

刊名：Nuclear Medicine and Biology

出版年：2017

6.Tactics for preclinical validation of receptor-binding radiotracers

作者：Susan Z. Lever^a ; ^b ; ^{levers@missouri.edu} ; Kuo-Hsien Fan^a ; John R. Lever^c ; ^d ; ^{leverj@health.missouri.edu}

关键词：Imaging ; Validation ; Radiopharmaceutical ; Radiotracer ; Radiopharmacology ; Sigma receptor

刊名：Nuclear Medicine and Biology

出版年：2017

7.In vivo evaluation of IGF1R/IR PET ligand [¹⁸F]BMS-754807 in rodents

作者：Jaya Prabhakaran^a ; ^b ; Stephen L. Dewey^c ; Richard McClure^d ; ^e ; Norman R. Simpson^b ; Mohammed N. Tantawy^d ; J. John Mann^a ; ^b ; Wellington Pham^d ; ^e ; J.S. Dileep Kumar^b ; ^{kumardi@nyspi.columbia.edu}

关键词：IGF1R ; IR ; Insulin ; Radiotracer ; MicroPET

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

8.High affinity binding of the peptide agonist TIP-39 to the parathyroid hormone 2 (PTH₂) receptor requires the hydroxyl group of Tyr-318 on transmembrane helix 5

作者：Richard E. Weaver^a ; Juan C. Mobarec^c ; Mark J. Wigglesworth^b ; ¹ ; Christopher A. Reynolds^c ; Dan Donnelly^a ; ^{d.donnelly@leeds.ac.uk}

关键词：Parathyroid hormone ; PTH ; GPCR ; Agonist ; Receptor ; TIP39

刊名：Biochemical Pharmacology

出版年：2017

9.Approaches to improve metabolic stability of a statine-based GRP receptor antagonist

作者：Ilinca Popp^a ; Luigi Del Pozzo^a ; ^b ; ^c ; Beatrice Waser^d ; Jean Claude Reubi^d ; Philipp T. Meyer^a ; ^b ; ^c ; Helmut R. Maecke^a ; Eleni Gourni^a ; ^b ; ^c ; ^{eleni.gourni@medisin.uio.no}

关键词：Gastrin-releasing peptide receptor antagonists ; Metabolic stability ; 68Ga ; PET-imaging

刊名：Nuclear Medicine and Biology

出版年：2017

10.Preliminary evidence that negative symptom severity relates to multilocus genetic profile for dopamine signaling capacity and D2 receptor binding in healthy controls and in schizophrenia

作者：Sarah A. Eisenstein^a ; ^b ; ^{seisens@wustl.edu} ; Ryan Bogdan^c ; ^{rbogdan@wustl.edu} ; Ling Chen^d ; ^{lingchen@wustl.edu} ; Stephen M. Moerlein^b ; ^e ; ^{moerleins@mir.wustl.edu} ; Kevin J. Black^a ; ^b ; ^f ; ^g ; ^{kevin@wustl.edu} ; Joel S. Perlmutter^b ; ^e ; ^h ; ^{joel@wustl.edu} ; Tamara Hershey^a ; ^b ; ^c ; ^f ; ^{tammy@wustl.edu} ; Deanna M. Barch^a ; ^b ; ^c ; ^{dbarch@wustl.edu}

关键词：Schizophrenia ; Negative symptoms ; Anhedonia ; Genetic profile ; Dopamine ; PET

刊名：Journal of Psychiatric Research

出版年：2017

按检索点细分(3351)

题名(532)

关键词(491)

文摘(2919)