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Wiley电子期刊(8)	NATURE电子期刊(7)	ACS电子期刊(151)
SpringerLink电子期刊(181)	Elsevier电子期刊(797)

在“Elsevier电子期刊”中，命中：797条，耗时：0.0749627 秒

在所有数据库中总计命中：1,144条

1.Identification of novel small molecule inhibitors against NS2B/NS3 serine protease from Zika virus

作者：Hyun Lee^a ; Jinhong Ren^b ; Salvatore Nocadello^d ; Amy J. Rice^b ; ^c ; Isabel Ojeda^b ; ^c ; Samuel Light^d ; George Minasov^d ; Jason Vargas^b ; ^c ; Dhanapalan Nagarathnam^e ; Wayne F. Anderson^d ; Michael E. Johnson^a ; ^{mssjohnson@novalextherapeutics.com}

关键词：Zika flavivirus ; NS2B/NS3 serine protease ; Small molecule inhibitor ; apo ZIKV NS2B-NS3pro structure

刊名：Antiviral Research

出版年：2017

2.Structure-activity relationships of 4-hydroxy-4-biaryl-proline acylsulfonamide tripeptides: A series of potent NS3 protease inhibitors for the treatment of hepatitis C virus

作者：Alan Xiangdong Wang^a ; ^{alan.wang@bms.com} ; Jie Chen^a ; Qian Zhao^a ; Li-Qiang Sun^a ; Jacques Friborg^b ; Fei Yu^b ; Dennis Hernandez^b ; Andrew C. Good^c ; Herbert E. Klei^c ; Ramkumar Rajamani^c ; Kathy Mosure^d ; Jay O. Knipe^d ; Danshi Li^d ; Jialong Zhu^d ; Paul C. Levesque^d ; Fiona McPhee^b ; Nicholas A. Meanwell^a ; Paul M. Scola^a ;

关键词：HCV NS3/4A serine protease inhibitors ; Tripeptide acylsulfonamides ; C4 aryl ; C4 hydroxy-proline ; Potent and orally bioavailable ; Cardiovascular profiles

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

3.The solution structure of the kallikrein-related peptidases inhibitor SPINK6

作者：Sascha Jung^a ; Jan Fischer^b ; Bjö ; rn Spudy^a ; Tim Kerkow^a ; Frank D. Sö ; nnichsen^c ; Li Xue^d ; Alexandre M.J.J. Bonvin^d ; Peter Goettig^e ; Viktor Magdolen^f ; Ulf Meyer-Hoffert^b ; Joachim Grö ; tzinger^a ; ^{jgroetzinger@biochem.uni-kiel.de" class="auth_mail" title="E-mail the corresponding author}

关键词：SPINK6 ; Kallikrein-related peptidase 4 ; KLK4 ; Structure ; Model protease &ndash ; inhibitor complex ; Nuclear magnetic resonance

刊名：Biochemical and Biophysical Research Communications

出版年：2016

4.Insights into the serine protease mechanism based on structural observations of the conversion of a peptidyl serine protease inhibitor to a substrate

作者：Longguang Jiang^a ; ^b ; ; Lisbeth Moreau Andersen^b ; ^c ; ; Peter A. Andreasen^b ; ^c ; ; Liqing Chen^d ; Mingdong Huang^a ; ^b ; ^{mhuang@fjirsm.ac.cn" class="auth_mail" title="E-mail the corresponding author} ;

关键词：uPA ; urokinase-type plasminogen activator ; uPA16&ndash ; 244 ; serine protease domain of uPA (residues 16&ndash ; 244) ; KD ; equilibrium dissociation constant ; Ki ; equilibrium inhibition constant ; PAB ; p-aminobenzamidine

刊名：Biochimica et Biophysica Acta (BBA) - General Subjects

出版年：2016

5.Design and synthesis of a series of serine derivatives as small molecule inhibitors of the SARS coronavirus 3CL protease

作者：Hiroyuki Konno^a ; ^{konno@yz.yamagata-u.ac.jp" class="auth_mail" title="E-mail the corresponding author} ; Masaki Wakabayashi^a ; Daiki Takanuma^a ; Yota Saito^a ; Kenichi Akaji^b ; ^{akaji@mb.kyoto-phu.ac.jp" class="auth_mail" title="E-mail the corresponding author}

关键词：SARS CoV ; SARS 3CL protease ; Serine derivative ; Docking simulation ; Cathepsin B ; Cytotoxicity

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

6.Structural basis of specific inhibition of tissue-type plasminogen activator by plasminogen activators inhibitor-1

作者：Lihu Gong^a ; ^b ; Min Liu^a ; ^b ; Tu Zeng^a ; Xiaoli Shi^a ; Cai Yuan^a ; Peter A. Andreasen^c ; Mingdong Huang^a ; ^b ; ^{mhuang@fjirsm.ac.cn" class="auth_mail" title="E-mail the corresponding author}

关键词：Tpa ; Serine protease ; PAI-1 ; Serpin ; Michaë ; lis complex ; Crystal structure ; Fibrinolysis ; Thrombolytic agents ; Structural biology

刊名：Data in Brief

出版年：2016

7.Drosophila melanogaster clip-domain serine proteases: Structure, function and regulation

作者：Florian Veillard^a ; ^{f.veillard@ibmc-cnrs.unistra.fr" class="auth_mail" title="E-mail the corresponding author} ; Laurent Troxler^a ; Jean-Marc Reichhart^b

关键词：Chymotrypsin ; Insect ; Immunity ; Melanization ; Serpin ; Toll

刊名：Biochimie

出版年：2016

8.Structure-based design, synthesis, and biological evaluation of Leu-Arg dipeptide analogs as novel hepsin inhibitors

作者：Hongmok Kwon ; YunHye Kim ; Kieung Park ; Soo An Choi ; Sang-Hyun Son ; ^{shson@korea.ac.kr" class="auth_mail" title="E-mail the corresponding author} ; Youngjoo Byun ; ^{yjbyun1@korea.ac.kr" class="auth_mail" title="E-mail the corresponding author}

关键词：Hepsin ; Prostate cancer ; Dipeptides ; Serine protease

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

9.How Dextran Sulfate Affects C1-inhibitor Activity: A Model for Polysaccharide Potentiation

作者：Madelon Dijk¹ ; Jolande Holkers² ; Patrick Voskamp¹ ; Bruno M. Giannetti² ; Willem-Jan Waterreus¹ ; Harrie A. van Veen² ; ^{h.vanveen@pharming.com} ; Navraj S. Pannu¹ ; ³ ; ^{raj@chem.leidenuniv.nl}

关键词：serine protease inhibitor ; C1-inhibitor ; polysaccharide potentiation ; complement system ; contact system

刊名：Structure

出版年：2016

10.Biology of rhomboid proteases in infectious diseases

作者：Sunil Kumar Dogga ; ^{Sunil.Dogga@unige.ch} ; Dominique Soldati-Favre

关键词：Rhomboid proteases ; Intramembrane proteolysis ; Apicomplexa ; Mycobacteria ; Adhesins ; Protozoan pathogens ; Parasites

刊名：Seminars in Cell & Developmental Biology

出版年：2016

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