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SpringerLink电子期刊(1)
Elsevier电子期刊(10)
ACS电子期刊(3)
在“
Elsevier电子期刊
”中,
命中:
10
条,耗时:小于0.01 秒
在所有数据库中总计命中:
14
条
1.
Insights into the molecular basis of action of the AT
1
antagonist losartan using a combined NMR spectroscopy and computational approach
作者:
Maria Zervou
;
Zoe Cournia
;
Constantinos Potamitis
;
George Patargias
;
Serdar Durdagi
;
Simona
Golic
Grdadolnik
;
Thomas Mavromoustakos
关键词:
Losartan
;
SDS micelles
;
NMR (DOSY
;
NOESY/ROESY)
;
Spin labels
;
Molecular dynamics in micelles
;
Molecular dynamics in phospholipid bilayers with embedded AT1 receptor
刊名:Biochimica et Biophysica Acta (BBA)/Biomembranes
出版年:March, 2014
2.
Rational design, efficient syntheses and biological evaluation of N,N¡ä-symmetrically bis-substituted butylimidazole analogs as a new class of potent Angiotensin II receptor blockers
作者:
George Agelis
a
;
l
;
1
;
aggelisgeorge@hotmail.com
;
Amalia Resvani
a
;
l
;
1
;
Catherine Koukoulitsa
b
;
Tereza T?mová
;
c
;
Ji?ina Slaninová
;
c
;
Dimitra Kalavrizioti
d
;
Katerina Spyridaki
e
;
Antreas Afantitis
f
;
Georgia Melagraki
f
;
Athanasia Siafaka
g
;
Eleni Gkini
g
;
Grigorios Megariotis
h
;
Simona
Golic
Grdadolnik
i
;
j
;
Manthos G. Papadopoulos
h
;
Demetrios Vlahakos
k
;
Michael Maragoudakis
d
;
George Liapakis
e
;
Thomas Mavromoustakos
b
;
John Matsoukas
a
;
l
;
imats@upatras.gr
关键词:
AT1 receptor blockers
;
N
;
N&prime
;
-Bis-alkylated butylimidazole analogs
;
Synthesis
;
Wittig reaction
;
Hydroxymethylation
;
Structure elucidation
;
Docking studies
;
Molecular dynamics
;
Biological evaluation
刊名:European Journal of Medicinal Chemistry
出版年:2013
3.
Conformational analysis of two novel cytotoxic C2-substituted pyrrolo[2,3-f]quinolines in aqueous media, organic solvents, membrane bilayers and at the putative active site
作者:
Nicole Varvarigou
;
Grigorios Megariotis
;
Georgios Leonis
;
Eleni Vrontaki
;
Antigoni-Margarita Maniati
;
Marilena Vlachou
;
Aphrodite Eikosipentaki
;
Rodanthi Kompogennitaki
;
Manthos G. Papadopoulos
;
Simona
Golic
Grdadolnik
;
Dimitri Komiotis
;
Thomas Mavromoustakos
;
Andrew Tsotinis
关键词:
Cytotoxic agents
;
Conformational analysis
;
NMR spectroscopy
;
Molecular dynamics
;
Molecular docking
;
Lipid bilayers
刊名:Bioorganic and Medicinal Chemistry
出版年:2012
4.
Corrigendum to ¡°Thermal, dynamic and structural properties of drug AT
1
antagonist olmesartan in lipid bilayers?[Biochim. Biophys. Acta 1808 (2011) 2995-3006]
作者:
Dimitrios Ntountaniotis
a
;
b
;
Gregor Mali
c
;
e
;
Simona
Golic
Grdadolnik
d
;
e
;
Maria Halabalaki
f
;
Alexios-Leandros Skaltsounis
f
;
Constantinos Potamitis
b
;
Eleni Siapi
b
;
Petros Chatzigeorgiou
g
;
Michael Rappolt
h
;
michael.rappolt@elettra.trieste.it
;
Thomas Mavromoustakos
i
;
tmavrom@chem.uoa.gr
刊名:Biochimica et Biophysica Acta (BBA)/Biomembranes
出版年:2012
5.
Thermal, dynamic and structural properties of drug AT
1
antagonist olmesartan in lipid bilayers
作者:
Dimitrios
;
Ntountaniotis
a
;
;
b
;
Gregor
;
Mali
c
;
;
e
;
Simona
Golic
;
Grdadolnik
d
;
;
e
;
Halabalaki
;
Maria
f
;
Alexios-Leandros
;
Skaltsounis
f
;
Constantinos
;
Potamitis
b
;
Eleni
;
Siapi
b
;
Petros
;
Chatzigeorgiou
g
;
Michael
;
Rappolt
h
;
;
michael.rappolt@elettra.trieste.it
;
Thomas
;
Mavromoustakos
i
;
;
tmavrom@chem.uoa.gr
关键词:
Olmesartan
;
Dipalmitoyl-phosphatidylcholine bilayer
;
Small-angle and wide angle X-ray scattering
;
Raman spectroscopy
;
Differential scanning calorimetry
;
Solid state NMR spectroscopy
刊名:Biochimica et Biophysica Acta (BBA)/Biomembranes
出版年:2011
6.
Structure elucidation and conformational study of V8: A novel synthetic non peptide AT
1
antagonist
作者:
Panagiotis Zoumpoulakis
;
Aggeliki Politi
;
Simona
Golic
Grdadolnik
;
John Matsoukas and Thomas Mavromoustakos
关键词:
Synthetic angiotensin II antagonists
;
Conformational properties
;
Molecular modeling
;
NMR
;
Losartan
刊名:Journal of Pharmaceutical and Biomedical Analysis
出版年:2006
7.
Structural elucidation and conformational properties of the toxin paralysin β-Ala–Tyr
作者:
Kyrikou
;
Ioanna
;
Grdadolnik
;
Simona
Golic
;
Tatari
;
Maria
;
Poulos
;
Constantine
;
Mavromoustakos
;
Thomas
关键词:
Paralysins
;
β
;
-alanine&ndash
;
tyrosine
;
NMR
;
Molecular modeling
;
Neobelleria Bullata
刊名:Journal of Pharmaceutical and Biomedical Analysis
出版年:2003
8.
Structure elucidation and conformational properties of eprosartan a non peptide Angiotensin II AT
1
antagonist
作者:
Zoumpoulakis
;
Panagiotis
;
Grdadolnik
;
Simona
Golic
;
Matsoukas
;
John
;
Mavromoustakos
;
Thomas
关键词:
Antihypertensives
;
Eprosartan
;
Losartan
;
AT
1
antagonists
;
NMR
;
Molecular modeling
刊名:Journal of Pharmaceutical and Biomedical Analysis
出版年:2002
9.
Structure elucidation and conformational properties of a novel bioactive clerodane diterpene using a combination of high field NMR spectroscopy, computational analysis and X-ray diffraction
作者:
Kolocouris
;
Antonios
;
Mavromoustakos
;
Thomas
;
Demetzos
;
Costas
;
Terzis
;
Aris
;
Grdadolnik
;
Simona
Golic
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2001
10.
Synthesis and study of a cyclic angiotensin II antagonist analogue reveals the role of π*–π* interactions in the C-terminal aromatic residue for agonist activity and its structure rese
作者:
Polevaya
;
Ludmila
;
Mavromoustakos
;
Thomas
;
Zoumboulakis
;
Panagiotis
;
Grdadolnik
;
Simona
Golic
;
et. al.
刊名:Bioorganic and Medicinal Chemistry
出版年:2001
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