设为首页
收藏本站
网站地图
|
English
|
公务邮箱
About the library
Background
History
Leadership
Organization
Readers' Guide
Opening Hours
Collections
Help Via Email
Publications
Electronic Information Resources
常用资源
电子图书
期刊论文
学位会议
外文资源
特色专题
内部出版物
SpringerLink电子期刊(2)
Elsevier电子期刊(12)
ACS电子期刊(3)
在“
Elsevier电子期刊
”中,
命中:
12
条,耗时:小于0.01 秒
在所有数据库中总计命中:
17
条
1.
Synthesis and evaluation o
f
carbamate and aryl ether substituted pyrazinones as corticotropin releasing
f
actor-1 (CRF
1
) receptor antagonists
作者:
Vijay T. Ahuja
;
vijay.ahuja@bms.com" class="auth_mail" title="E-mail the corresponding author
;
Richard A. Hartz
;
Thaddeus
F
.
Molski
;
Gail K. Mattson
;
Kimberley A. Lentz
;
James E. Grace Jr.
;
Nicholas J. Lodge
;
Joanne J. Bronson
;
John E. Macor
关键词:
CR
F
1 receptor antagonists
;
CR
F
;
Depression
;
Neuroscience
;
Pyrazinones
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
2.
Con
f
ormationally restricted homotryptamines. Part 6: Indole-5-cycloalkyl methylamines as selective serotonin reuptake inhibitors
作者:
Jonathan L. Ditta
;
jonathan.ditta@bms.com
;
Derek J. Denhart
;
Je
ff
rey A. Deskus
;
James R. Epperson
;
Zhaoxing Meng
;
Qi Gao
;
Gail K. Mattson
;
Mellissa A. LaPaglia
;
Matthew T. Taber
;
Thaddeus
F
.
Molski
;
Nicholas J. Lodge
;
Ronald J. Mattson
;
John E. Macor
关键词:
Indoles
;
Homotryptamines
;
SSRI
;
Serotonin
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2013
3.
NK1 receptor antagonism lowers occupancy requirement
f
or antidepressant-like e
ff
ects o
f
SSRIs in the Gerbil
f
orced swim test
作者:
Snjezana Lelas
;
Yu-Wen Li
;
Tanya L. Wallace-Boone
;
Matthew T. Taber
;
Amy E. Newton
;
Rick L. Pieschl
;
Carl D. Davis
;
Thaddeus
F
.
Molski
;
Kimberly S. Newberry
;
Michael
F
. Parker
;
Kevin W. Gillman
;
Joanne J. Bronson
;
John E. Macor
;
Nicholas J. Lodge
关键词:
Serotonin transporter
;
Neurokinin-1 receptor
;
Occupancy
;
Gerbil
;
Depression
;
BMS-795176
刊名:Neuropharmacology
出版年:2013
4.
[
18
F
](R)-5-chloro-1-(1-cyclopropyl-2-methoxyethyl)-3-(4-(2-
f
luoroethoxy)-2,5-dimethyl phenylamino)pyrazin-2(1H)-one: Introduction o
f
N
3
-phenylpyrazinones as potential CRF-R1 PET imaging agents
作者:
Je
ff
rey A. Deskus
;
Douglas D. Dischino
;
Ronald J. Mattson
;
Jonathan L. Ditta
;
Michael
F
. Parker
;
Derek J. Denhart
;
Dmitry Zuev
;
Hong Huang
;
Richard A. Hartz
;
Vijay T. Ahuja
;
Henry Wong
;
Gail K. Mattson
;
Thaddeus
F
.
Molski
;
James E. Grace Jr.
;
Larisa Zueva
;
Julia M. Nielsen
;
Heidi Dulac
;
Yu-Wen Li
;
Mary Guaraldi
;
Michael Azure
;
et al.
关键词:
Corticotropin-releasing
f
actor
;
Positron Emission Tomography
;
Antidepressants
;
Anxiolytics
;
Radioligand
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2012
5.
Synthesis and structure-activity relationships o
f
pyrido[3,2-b]pyrazin-3(4H)-ones and pteridin-7(8H)-ones as corticotropin-releasing
f
actor-1 receptor antagonists
作者:
Carolyn D. Dzierba
;
Thais M. Sielecki
;
Argyrios G. Arvanitis
;
Amy Galka
;
Tricia L. Johnson
;
Amy G. Takvorian
;
Maria Ra
f
alski
;
Padmaja Kasireddy-Polam
;
Shikha Vig
;
Bireshwar Dasgupta
;
Ge Zhang
;
Thaddeus
F
.
Molski
;
Harvey Wong
;
Robert C. Zaczek
;
Nicholas J. Lodge
;
Andrew P. Combs
;
Paul J. Gilligan
;
George L. Trainor
;
Joanne J. Bronson
;
John E. Macor
;
et al.
关键词:
GXWKAWZLOBUGGM-UH
F
FFAOYSA-N
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2012
6.
Synthesis and structure–activity relationships o
f
N
3
-pyridylpyrazinones as corticotropin-releasing
f
actor-1 (CRF
1
) receptor antagonists
作者:
Richard A. Hartz
;
Vijay T. Ahuja
;
William D. Schmitz
;
Thaddeus
F
.
Molski
;
Gail K. Mattson
;
Nicholas J. Lodge
;
Joanne J. Bronson
;
John E. Macor
关键词:
Corticotropin-releasing
f
actor
;
CR
F
;
Pyrazinone
;
G-protein coupled receptors
;
Pyridyl
;
Pyrimidyl
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
7.
5-Arylamino-1,2,4-triazin-6(1H)-one CR
F
1
receptor antagonists
作者:
William D. Schmitz
;
Allison B. Brenner
;
Joanne J. Bronson
;
Jonathan L. Ditta
;
Corrine R. Gri
ff
in
;
Yu-Wen Li
;
Nicholas J. Lodge
;
Thaddeus
F
.
Molski
;
Richard E. Olson
;
Xiaoliang Zhuo
;
John E. Macor
关键词:
Corticotropin releasing
f
actor
;
Triazinone
;
Depression
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
8.
Synthesis and hSERT activity o
f
homotryptamine analogs. Part 6: [3+2] dipolar cycloaddition o
f
3-vinylindoles
作者:
Lawrence R. Marcin
;
Ronald J. Mattson
;
Qi Gao
;
Dedong Wu
;
Thaddeus
F
.
Molski
;
Gail K. Mattson
;
Nicholas J. Lodge
关键词:
Homotryptamine
;
Serotonin
;
SERT
;
DAT
;
NET
;
SSRI
;
Dipolar cycloaddition
;
3-Vinylindole
;
Nitrone
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
9.
Con
f
ormationally restricted homotryptamines. Part 5: 3-(trans-2-aminomethylcyclopentyl)indoles as potent selective serotonin reuptake inhibitors
作者:
Derek J. Denhart
;
Je
ff
rey A. Deskus
;
Jonathan L. Ditta
;
Qi Gao
;
H. Dalton King
;
Edward S. Kozlowski
;
Zhaoxing Meng
;
Melissa A. LaPaglia
;
Gail K. Mattson
;
Thaddeus
F
.
Molski
;
Matthew T. Taber
;
Nicholas
关键词:
Indoles
;
Homotryptamines
;
SSRI
;
Serotonin
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
10.
Ex vivo assessment o
f
binding site occupancy o
f
monoamine reuptake inhibitors: Methodology and biological signi
f
icance
作者:
Kelly Lengyel
;
Rick Pieschl
;
Todd Strong
;
Thaddeus
Molski
;
Gail Mattson
;
Nicholas J. Lodge
;
Yu-Wen Li
关键词:
Monoamine transporter
;
Reuptake inhibitor
;
Dopamine
;
Norepinephrine
;
Serotonin
;
Occupancy
;
Ex vivo
;
Radioligand binding
刊名:Neuropharmacology
出版年:2008
1
2
按检索点细分(12)
作者(12)
按出版年细分(12)
2016年(1)
2013年(2)
2012年(2)
2010年(3)
2009年(1)
2008年(1)
2007年(1)
2005年(1)
NGLC 2004-2010.National Geological Library of China All Rights Reserved.
Add:29 Xueyuan Rd,Haidian District,Beijing,PRC. Mail Add: 8324 mailbox 100083
For exchange or info please contact us via
email
.