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Wiley电子期刊(1)	NATURE电子期刊(4)	ACS电子期刊(75)
SpringerLink电子期刊(64)	Elsevier电子期刊(287)

在“Elsevier电子期刊”中，命中：287条，耗时：小于0.01 秒

在所有数据库中总计命中：431条

1.Synthesis and biological evaluation of cis-restricted triazole/tetrazole mimics of combretastatin-benzothiazole hybrids as tubulin polymerization inhibitors and apoptosis inducers

作者：A.V. Subba Rao^a ; ^b ; Konderu Swapna^c ; Siddiq Pasha Shaik^a ; ^b ; V. Lakshma Nayak^a ; T. Srinivasa Reddy^c ; Satish Sunkari^a ; ^b ; Thokhir Basha Shaik^a ; Chandrakant Bagul^c ; Ahmed Kamal^a ; ^b ; ^c ;

关键词：Combretastatin A-4 ; Benzothiazole ; Triazoles and tetrazoles ; Antiproliferative activity ; Tubulin polymerization ; Colchicine competition assay ; Apoptosis

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

2.Bioreductively activatable prodrug conjugates of phenstatin designed to target tumor hypoxia

作者：Blake A. Winn^a ; Zhe Shi^a ; Graham J. Carlson^a ; Yifan Wang^a ; Benson L. Nguyen^a ; Evan M. Kelly^a ; R. David Ross IV^a ; Ernest Hamel^b ; David J. Chaplin^a ; ^c ; Mary L. Trawick^a ; ^{Mary_Lynn_Trawick@baylor.edu} ; Kevin G. Pinney^a ; ^{Kevin_Pinney@baylor.edu}

关键词：BAPC ; bioreductively activatable prodrug conjugate ; CA1 ; combretastatin A-1 ; CA4 ; combretastatin A-4 ; Et3N ; triethylamine ; HPLC ; high performance liquid chromatography ; HRMS ; high resolution mass spectrometry ; MeOH ; methanol ; NaBH4 ; sodium borohydride ; TLC ; thin layer chromatography ; THF ; tetrahydrofuran ; EtOAc ; ethyl acetate ; POR ; NADPH cytochrome P450 oxidoreductase ; DMP ; Dess-Martin periodinane ; DEAD ; diethylazodicarboxylate ; DIAD ; diisopropyl azodicarboxylate ; ADDP ; 1 ; 1&prime ; -(azodicarbonyl

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

3.Design, synthesis, and biological evaluation of novel alkylsulfanyl-1,2,4-triazoles as cis-restricted combretastatin A-4 analogues

作者：Yan-Hong Li¹ ; Bei Zhang¹ ; Hai-Kui Yang ; Qiu Li ; Peng-Cheng Diao ; Wen-Wei You ; ^{youww@smu.edu.cn} ; Pei-Liang Zhao ; ^{plzhao@smu.edu.cn}

关键词：Alkylsulfanyl-12 ; 4-triazoles ; Synthesis ; Antiproliferative activity

刊名：European Journal of Medicinal Chemistry

出版年：2017

4.Understanding the Binding of cis and trans Isomers of Combretastatin to Tubulin

作者：Isabel Rozas¹ ; ^{rozasi@tcd.ie}

刊名：Chem

出版年：2017

5.Discovery and preclinical evaluation of 7-benzyl-N-(substituted)-pyrrolo[3,2-d]pyrimidin-4-amines as single agents with microtubule targeting effects along with triple-acting angiokinase inhibition as antitumor agents

作者：Roheeth Kumar Pavana^a ; Shruti Choudhary^a ; Anja Bastian^b ; Michael A. Ihnat^c ; Ruoli Bai^d ; Ernest Hamel^d ; Aleem Gangjee^a ; ^{gangjee@duq.edu}

关键词：AA ; antiangiogenic agents ; MTA ; microtubule targeting agents ; VEGFR-2 ; vascular endothelial growth factor receptor-2 ; PDGFR-β ; platelet-derived growth factor receptor-β ; CAM ; chorioallantoic membrane ; CA ; combretastatin A-4 ; Pgp ; P-glycoprotein ; EGFR ; epidermal growth factor receptor ; TBS ; Tris-buffered saline ; HRP ; horseradish peroxidase ; PY ; phosphotyrosine

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

6.Piperlongumine (piplartine) and analogues: Antiproliferative microtubule-destabilising agents

作者：Mary J. Meegan^a ; Seema Nathwani^b ; Brendan Twamley^c ; Daniela M. Zisterer^b ; Niamh M. O'Boyle^a ; ^b ; ^{oboyleni@tcd.ie}

关键词：Antiproliferative ; Anticancer ; Combretastatin A-4 ; Microtubule-destabilising ; Piperlongumine ; Tubulin

刊名：European Journal of Medicinal Chemistry

出版年：2017

7.Structural Basis of cis- and trans-Combretastatin Binding to Tubulin

作者：Roberto Gaspari¹ ; ⁴ ; Andrea E. Prota² ; ⁴ ; Katja Bargsten² ; Andrea Cavalli¹ ; ³ ; ^{andrea.cavalli@iit.it} ; Michel O. Steinmetz² ; ⁵ ; ^{michel.steinmetz@psi.ch}

关键词：microtubule-targeting agents ; tubulin ; protein-ligand interaction ; cis-trans isomerism ; switchable molecules ; X-ray crystallography ; metadynamics

刊名：Chem

出版年：2017

8.Novel indole-based compounds that differentiate alkylindole-sensitive receptors from cannabinoid receptors and microtubules: Characterization of their activity on glioma cell migration

作者：Susan Fung^a ; ^b ; Cong Xu^a ; Ernest Hamel^c ; James B. Wager-Miller^d ; Grace Woodruff^a ; Aaron Miller^a ; Christina Sanford^a ; Ken Mackie^d ; Nephi Stella^a ; ^e ; ^{nstella@uw.edu}

关键词：2-AG ; arachidonoylglycerol ; AI ; alkylindole ; CB ; cannabinoid ; CB1 ; cannabinoid receptor 1 ; CB2 ; cannabinoid receptor 2 ; CSA4 ; combretastatin A4 ; DBT ; delayed Brain Tumor ; HA ; hemagglutinin ; LPA ; lysophosphatidic acid ; GBM ; glioblastoma multiforme ; SAR ; structure activity relationship ; THC ; tetrahydrocannabinol ; WIN-2 ; WIN55212-2

刊名：Pharmacological Research

出版年：2017

9.Combretastatins: In vitro structure-activity relationship, mode of action and current clinical status

作者：Karol Jaroch^a ; ^{karol.jaroch@cm.umk.pl" class="auth_mail" title="E-mail the corresponding author} ; Maciej Karolak^b ; Przemysław Gó ; rski^a ; Alina Jaroch^c ; ^d ; Adrian Krajewski^e ; Aleksandra Ilnicka^f ; Anna Sloderbach^a ; Tomasz Stefański^g ; ^h ; Stanisław Sobiak^b

关键词：Combretastatin ; CA4P ; Structure-activity relationship ; SAR ; Clinical trials

刊名：Pharmacological Reports

出版年：2016

10.pH-sensitive drug controlled release core/shell fibers fabricated by combination of electrospinning and photopolymerization

作者：Xiaolei Zhu ; Hongwei Zhang ; Jun Nie ; Guiping Ma ; ^{magp@mail.buct.edu.cn}

关键词：Electrospinning ; Photo-polymerization ; Core shell fibers

刊名：Journal of Industrial and Engineering Chemistry

出版年：2017

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