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SpringerLink电子期刊(1)
Elsevier电子期刊(8)
ACS电子期刊(4)
在“
Elsevier电子期刊
”中,
命中:
8
条,耗时:小于0.01 秒
在所有数据库中总计命中:
13
条
1.
N-(2-alkylaminoethyl)-4-(1,2,4-oxadiazol-5-yl)piperazine-1-carboxamides as highly potent smoothened antagonists
作者:
Ester Muraglia
a
;
Jesus M. Ontoria
a
;
Danila Branca
a
;
Gabriella Dessole
a
;
Alberto Bresciani
a
;
Massimiliano Fonsi
a
;
Claudio Giuliano
a
;
Laura
Llauger
Bufi
a
;
Edith Monteagudo
a
;
Maria Cecilia Palumbi
a
;
Caterina Torrisi
a
;
Michael Rowley
a
;
Christian Steinkü
;
hler
a
;
Philip Jones
;
a
;
philip_jones@dfci.harvard.edu"" rel=""nofollow
关键词:
Hedgehog pathway
;
Smoothened antagonist
;
Hedgehog inhibitor
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2011
2.
Identification of a series of 4-[3-(quinolin-2-yl)-1,2,4-oxadiazol-5-yl]piperazinyl ureas as potent smoothened antagonist hedgehog pathway inhibitors
作者:
Jesus M. Ontoria
a
;
Laura
Llauger
Bufi
a
;
Caterina Torrisi
a
;
Alberto Bresciani
a
;
Claudia Giomini
a
;
Michael Rowley
a
;
Sergio Serafini
a
;
Hu Bin
b
;
Wu Hao
b
;
Christian Steinkü
;
hler
a
;
Philip Jones
a
;
philip_jones@dfci.harvard.edu"" rel=""nofollow
关键词:
Hedgehog pathway
;
Smoothened antagonist
;
Hedgehog inhibitor
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2011
3.
Identification and SAR of novel pyrrolo[1,2-a]pyrazin-1(2H)-one derivatives as inhibitors of poly(ADP-ribose) polymerase-1 (PARP-1)
作者:
Giovanna Pescatore
;
Danila Branca
;
Fabrizio Fiore
;
Olaf Kinzel
;
Laura
Llauger
Bufi
;
Ester Muraglia
;
Federica Orvieto
;
Michael Rowley
;
Carlo Toniatti
;
Caterina Torrisi
;
Philip Jones
关键词:
Pyrrolo[1
;
2-
a
]pyrazin-1(2
H
)-one
;
Poly(ADP-ribose) polymerase
;
PARP-1
;
Oncology
;
Selectivity
;
BRCA1
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
4.
Development of substituted 6-[4-fluoro-3-(piperazin-1-ylcarbonyl)benzyl]-4,5-dimethylpyridazin-3(2H)-ones as potent poly(ADP–ribose) polymerase-1 (PARP-1) inhibitors active in BRCA deficient cells
作者:
Federica Ferrigno
;
Danila Branca
;
Olaf Kinzel
;
Samuele Lillini
;
Laura
Llauger
Bufi
;
Edith Monteagudo
;
Ester Muraglia
;
Michael Rowley
;
Carsten Schultz-Fademrecht
;
Carlo Toniatti
;
Caterina Torrisi
;
Phil
关键词:
Anticancer agents
;
PARP-1 inhibitor
;
BRCA1 deficient cancer cells
;
6-[4-Fluoro-3-(piperazin-1-ylcarbonyl)benzyl]-4
;
5-dimethylpyridazin-3(2
H
)-ones
;
Coupling reactions
;
SAR exploration
;
Pharmacokinetic properties
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
5.
A novel base-mediated intramolecular hydroamination to build fused heteroaryl pyrazinones
作者:
Laura
Llauger
;
Costanza Bergami
;
Olaf D. Kinzel
;
Samuele Lillini
;
Giovanna Pescatore
;
Caterina Torrisi
;
Philip Jones
关键词:
Intramolecular hydroamination
;
Pyrrolopyrazinones
;
Fused-heteroaryl pyrazinones
;
DBU-mediated cyclisation
;
Isomerisation
刊名:Tetrahedron Letters
出版年:2009
6.
Synthesis of 8-arylsulfoxyl/sulfonyl adenines
作者:
Llauger
;
Laura
;
He
;
Huazhong
;
Chiosis
;
Gabriela
关键词:
Oxidation
;
Alumina supported OXONE
??
;
8-Arylsufoxyl adenines
;
8-Arylsufonyl adenines
刊名:Tetrahedron Letters
出版年:2004
7.
Synthesis of novel fluorescent probes for the molecular chaperone Hsp90
作者:
Llauger
-Bufi
;
Laura
;
Felts
;
Sara J.
;
Huezo
;
Henri
;
Rosen
;
Neal
;
Chiosis
;
Gabriela
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2003
8.
A Short Procedure for the Preparation of Highly Functionalized Di- and Tetrahydropyridines
作者:
Bennasar
;
M.-Lluï
;
sa
;
Zulaica
;
Ester
;
Juan
;
Cecí
;
lia
;
Llauger
;
Laura
;
Bosch
;
Joan
关键词:
Acylation
;
enolates
;
pyridinium salts
;
pyridines
刊名:Tetrahedron Letters
出版年:1999
1
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2000年及以前(1)
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