设为首页
收藏本站
网站地图
|
English
|
公务邮箱
About the library
Background
History
Leadership
Organization
Readers' Guide
Opening Hours
Collections
Help Via Email
Publications
Electronic Information Resources
常用资源
电子图书
期刊论文
学位会议
外文资源
特色专题
内部出版物
Wiley电子期刊(1)
SpringerLink电子期刊(1)
Elsevier电子期刊(13)
ACS电子期刊(1)
在“
Elsevier电子期刊
”中,
命中:
13
条,耗时:小于0.01 秒
在所有数据库中总计命中:
16
条
1.
Multitarget opioid ligands in pain relief: New players in an old game
作者:
Rita Turnaturi
a
;
rita.turnaturi@tiscali.it" class="auth_mail" title="E-mail the corresponding author
;
Giuseppina Aricò
;
a
;
Giuseppe Ronsisvalle
a
;
Carmela Parenti
b
;
1
;
Lorella
Pasquinucci
a
;
1
关键词:
Pain
;
MOR
;
DOR
;
KOR
;
Bifunctional ligands
;
Bivalent ligands
刊名:European Journal of Medicinal Chemistry
出版年:2016
2.
An LP1 analogue, selective MOR agonist with a peculiar pharmacological profile, used to scrutiny the ligand binding domain
作者:
Simone Ronsisvalle
a
;
s.ronsisvalle@unict.it" class="auth_mail" title="E-mail the corresponding author
;
Giuseppina Aricò
;
a
;
Federica Panarello
a
;
Angelo Spadaro
a
;
Lorella
Pasquinucci
a
;
Maria S. Pappalardo
a
;
Carmela Parenti
b
;
Nicole Ronsisvalle
c
关键词:
MOR agonists
;
6
;
7-Benzomorphan scaffold
;
Modeling studies
;
Radioligand competition-binding assay
;
Tail-flick test
;
GPI and MVD assays
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
3.
New bifunctional antioxidant/σ
1
agonist ligands: Preliminary chemico-physical and biological evaluation
作者:
Emanuela Arena
a
;
Ivana Cacciatore
b
;
Laura S. Cerasa
b
;
Hasan Turkez
b
;
c
;
Valeria Pittalà
;
a
;
Lorella
Pasquinucci
a
;
Agostino Marrazzo
a
;
Carmela Parenti
d
;
Antonio Di Stefano
b
;
Orazio Prezzavento
a
;
prezzave@unict.it" class="auth_mail" title="E-mail the corresponding author
关键词:
σ1 receptors
;
Oxidative stress
;
Neuroprotection
;
Chemical and enzymatic stabilities
;
Antioxidants
;
Lipoic acid
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
4.
Evaluation of N-substituent structural variations in opioid receptor profile of LP1
作者:
Lorella
Pasquinucci
a
;
Rita Turnaturi
a
;
rita.turnaturi@tiscali.it" class="auth_mail" title="E-mail the corresponding author
;
Giuseppina Aricò
;
a
;
Carmela Parenti
b
;
Paschalina Pallaki
c
;
Zafiroula Georgoussi
c
;
Simone Ronsisvalle
a
关键词:
Mu opioid receptor
;
6
;
7-Benzomorhan scaffold
;
Radioligand competition-binding assay
;
GPI and MVD assays
;
Tail-flick test
;
Modeling studies
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
5.
Differential scanning calorimetry approach to investigate the transfer of the multitarget opioid analgesic LP1 to biomembrane model
作者:
Maria Lorena Accolla
a
;
Rita Turnaturi
b
;
Maria Grazia Sarpietro
b
;
mg.sarpietro@unict.it" class="auth_mail
;
Simone Ronsisvalle
b
;
Francesco Castelli
b
;
Lorella
Pasquinucci
b
关键词:
DSC
;
Liposome
;
Biomembrane
;
LP1
;
Multitarget
;
Opioid
刊名:European Journal of Medicinal Chemistry
出版年:22 April, 2014
6.
The multitarget opioid ligand LP1's effects in persistent pain and in primary cell neuronal cultures
作者:
Carmela Parenti
a
;
Rita Turnaturi
b
;
Giuseppina Aricò
;
b
;
garico@unict.it
;
Alexandra Gramowski-Voß
;
c
;
Olaf H.-U. Schroeder
d
;
Agostino Marrazzo
b
;
Orazio Prezzavento
b
;
Simone Ronsisvalle
b
;
Giovanna M. Scoto
a
;
Giuseppe Ronsisvalle
b
;
Lorella
Pasquinucci
b
关键词:
Neuropathic pain
;
Inflammatory pain
;
Opioid receptors
;
LP1
;
Micro-electrode array (MEA)
;
Electrophysiological behaviour
刊名:Neuropharmacology
出版年:2013
7.
The benzomorphan-based LP1 ligand is a suitable MOR/DOR agonist for chronic pain treatment
作者:
Lorella
Pasquinucci
a
;
lpasquin@unict.it
;
Carmela Parenti
b
;
Rita Turnaturi
a
;
Giuseppina Aricò
;
a
;
Agostino Marrazzo
a
;
Orazio Prezzavento
a
;
Simone Ronsisvalle
a
;
Zafiroula Georgoussi
c
;
Danai-Dionysia Fourla
c
;
Giovanna M. Scoto
b
;
Giuseppe Ronsisvalle
a
关键词:
Bifunctional drugs
;
Antinociceptive tolerance
;
[35S]GTP¦ÃS binding studies
;
Tail-flick test
刊名:Life Sciences
出版年:2012
8.
Antinociceptive profile of LP1, a non-peptide multitarget opioid ligand
作者:
Carmela Parenti
;
Rita Turnaturi
;
Giuseppina Aric¨°
;
Agostino Marrazzo
;
Orazio Prezzavento
;
Simone Ronsisvalle
;
Giovanna M. Scoto
;
Giuseppe Ronsisvalle
;
Lorella
Pasquinucci
关键词:
Supraspinal analgesia
;
6
;
7-benzomorphan ligand
;
Naloxone methiodide
;
Selective opioid antagonists
;
Rat
刊名:Life Sciences
出版年:2012
9.
Antiproliferative activity of phenylbutyrate ester of haloperidol metabolite II [(±)-MRJF4] in prostate cancer cells
作者:
Agostino Marrazzo
;
Jole Fiorito
;
Laura Zappalà
;
Orazio Prezzavento
;
Simone Ronsisvalle
;
Lorella
Pasquinucci
;
Giovanna M. Scoto
;
Renato Bernardini
;
Giuseppe Ronsisvalle
关键词:
Histone deacetylase
;
Inhibitors
;
LNCaP
;
PC3
;
Sigma receptors
刊名:European Journal of Medicinal Chemistry
出版年:2011
10.
Evaluation of N-substitution in 6,7-benzomorphan compounds
作者:
Lorella
Pasquinucci
;
Orazio Prezzavento
;
Agostino Marrazzo
;
Emanuele Amata
;
Simone Ronsisvalle
;
Zafiroula Georgoussi
;
Danai-Dionysia Fourla
;
Giovanna M. Scoto
;
Carmela Parenti
;
Giuseppina Aricò
关键词:6 ;
7-Benzomorphan derivatives
;
μ
;
/δ
;
opioid agonist
;
cAMP accumulation assay
;
Tail-flick test
刊名:Bioorganic and Medicinal Chemistry
出版年:2010
1
2
按检索点细分(13)
作者(13)
按出版年细分(13)
2027年及以后(1)
2016年(4)
2013年(1)
2012年(2)
2011年(1)
2010年(1)
2001年(2)
2000年(1)
NGLC 2004-2010.National Geological Library of China All Rights Reserved.
Add:29 Xueyuan Rd,Haidian District,Beijing,PRC. Mail Add: 8324 mailbox 100083
For exchange or info please contact us via
email
.