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ProQuest学位论文(1)
Elsevier电子期刊(8)
ACS电子期刊(1)
在“
Elsevier电子期刊
”中,
命中:
8
条,耗时:0.0319878 秒
在所有数据库中总计命中:
10
条
1.
Preclinical characterization of substituted 6,7-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-8(5H)-one P2X7 receptor antagonists
作者:
Michael
K.
Ameriks
;
Hong Ao
;
Nicholas I. Carruthers
;
Brian Lord
;
Suchitra Ravula
;
Jason C. Rech
;
Brad M. Savall
;
Jessica L. Wall
;
Qi Wang
;
Anindya Bhattacharya
;
Michael
A. Letavic
关键词:
P2X7
;
6
;
7-Dihydro-[1
2 ;
4]triazolo[4
;
3-a]pyrazin-8(5H)-one
;
Autoradiography
;
Depression
;
CNS
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
2.
Diazinones as P2 replacements for pyrazole-based cathepsin S inhibitors
作者:
Michael
K.
Ameriks
;
Scott D. Bembenek
;
Matthew T. Burdett
;
Ingrid C. Choong
;
James P. Edwards
;
Damara Gebauer
;
Yin Gu
;
Lars Karlsson
;
Hans E. Purkey
;
Bart L. Staker
;
Siquan Sun
;
Robin L. Thurmond
;
Jia
关键词:
Cathepsin
;
Protease
;
Tethering
;
X-ray crystallography
;
Fragment-based screening
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
3.
Discovery and SAR of novel pyrazole-based thioethers as cathepsin S inhibitors: Part 1
作者:
Alice Lee-Dutra
;
Danielle K. Wiener
;
Kristen L. Arienti
;
Jing Liu
;
Neelak
;
ha Mani
;
Michael
K.
Ameriks
;
Frank U. Axe
;
Damara Gebauer
;
Pragnya J. Desai
;
Steven Nguyen
;
Mike R
;
al
;
Robin L. Thurmond
;
Siqu
关键词:
Cathepsin
;
Protease
;
Thioether
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
4.
Pyrazole-based arylalkyne cathepsin S inhibitors. Part II: Optimization of cellular potency
作者:
Michael
K.
Ameriks
;
Hui Cai
;
James P. Edwards
;
Damara Gebauer
;
Elizabeth Gleason
;
Yin Gu
;
Lars Karlsson
;
Steven Nguyen
;
Siquan Sun
;
Robin L. Thurmond
;
Jian Zhu
关键词:
Cathepsin
;
Protease
;
Invariant chain
;
Lysosomotropism
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
5.
Discovery of the first known small-molecule inhibitors of heme-regulated eukaryotic initiation factor 2α (HRI) kinase
作者:
Mark D. Rosen
;
Craig R. Woods
;
Steven D. Goldberg
;
Michael
D. Hack
;
A. Dawn Bounds
;
Young Yang
;
Pamela C. Wagaman
;
Victor K. Phuong
;
Angela P.
Ameriks
;
Terrance D. Barrett
;
Kimon C. Kanelakis
;
Jui Cha
关键词:
Anemia
;
Kinase inhibitors
;
Hemoglobin
;
HRI kinase
;
Blood
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
6.
Pyrazole-based cathepsin S inhibitors with arylalkynes as P1 binding elements
作者:
Michael
K.
Ameriks
;
Frank U. Axe
;
Scott D. Bembenek
;
James P. Edwards
;
Yin Gu
;
Lars Karlsson
;
Mike R
;
al
;
Siquan Sun
;
Robin L. Thurmond
;
Jian Zhu
关键词:
Cathepsin
;
Protease
;
Alkyne
;
X-ray crystallography
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
7.
Corrigendum to “Discovery of the first known small-molecule inhibitors of heme-regulated eukaryotic initiation factor 2α (HRI) kinase” [Bioorg. Med. Chem. Lett. 19 (2009) 6548]
作者:
Mark D. Rosen
;
Craig R. Woods
;
Steven D. Goldberg
;
Michael
D. Hack
;
A. Dawn Bounds
;
Young Yang
;
Pamela C. Wagaman
;
Victor K. Phuong
;
Angela P.
Ameriks
;
Terrance D. Barrett
;
Kimon C. Kanelakis
;
Jui Cha
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
8.
A Novel Approach to Oligocyclopropane Structural Units
作者:
Taylor
;
Richard E.
;
Ameriks
;
Michael
K.
;
LaMarche
;
Matthew J.
刊名:Tetrahedron Letters
出版年:1997
1
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2000年及以前(1)
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