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Elsevier电子期刊(16)
在“
Elsevier电子期刊
”中,
命中:
16
条,耗时:小于0.01 秒
在所有数据库中总计命中:
16
条
1.
New P2X3 receptor antagonists. Part 2: Identification and SAR of quinazolinones
作者:
Gá
;
bor Szá
;
ntó
;
Attila Makó
;
Istvá
;
n Vá
;
gó
;
Tamá
;
s Hergert
;
Imre Bata
;
Bence Farkas
;
Sá
;
ndor
Kolok
;
Mó
;
nika Vastag
关键词:
Purinergic receptor
;
ATP
;
Ion channel
;
P2X3 antagonist
;
Chronic cough
;
Structure&ndash
;
activity relationship
;
4-Oxo-6-aryl-phenethyl-quinazolines
;
Nanomolar activity
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
2.
New P2X3 receptor antagonists. Part 1: Discovery and optimization of tricyclic compounds
作者:
Gá
;
bor Szá
;
ntó
;
Attila Makó
;
Imre Bata
;
Bence Farkas
;
Sá
;
ndor
Kolok
;
Mó
;
nika Vastag
;
Attila Cselenyá
k
关键词:
Purinergic receptor
;
ATP
;
Ion channel
;
P2X3 antagonist
;
HTS campaign
;
Airway hyperractivity
;
New binding site
;
Chirality
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
3.
Poster #S17 ARE DOPAMINE PARTIAL AGONIST ANTIPSYCHOTICS SIMILAR? PRECLINICAL COMPARISON OF ARIPIPRAZOLE, BIFEPRUNOX AND CARIPRAZINE
作者:
Bé
;
la Kiss
;
Istvá
;
n Gyertyá
n ;
Zsolt Né
;
methy
;
Katalin Sá
;
ghy
;
Judit Laszy
;
Ká
;
roly Fazekas
;
Sá
;
ndor
Kolok
;
Zoltá
;
n Kapui
刊名:Schizophrenia Research
出版年:April, 2014
4.
Quinolinyl- and phenantridinyl-acetamides as bradykinin B1 receptor antagonists
作者:
Já
;
nos É
;
les
;
j.eles@richter.hu
;
Gyula Beke
;
Istvá
;
n Vá
;
gó
;
É
;
va Bozó
;
Jó
;
zsef Huszá
r ;
Á
;
kos Tarcsay
;
Sá
;
ndor
Kolok
;
É
;
va Schmidt
;
Mó
;
nika Vastag
;
Katalin Hornok
;
Sá
;
ndor
Farkas
;
Gyö
;
rgy Domá
;
ny
;
Gyö
;
rgy M. Keser?
关键词:
Bradykinin
;
B1 Antagonists
;
Quinoline
;
Phenantridine
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2012
5.
Carbamoyloximes as novel non-competitive mGlu5 receptor antagonists
作者:
Já
;
nos Galambos
;
Gá
;
bor Wá
;
gner
;
Katalin Nó
;
grá
;
di
;
Attila Bielik
;
Lá
;
szló
;
Molná
r ;
Amrita Bobok
;
Attila Horvá
;
th
;
Bé
;
la Kiss
;
Sá
;
ndor
Kolok
;
Jó
;
zsef N
关键词:
luR5 non-competitive antagonist carbamoyloxime
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
6.
Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluR5 NAMs
作者:
Gá
;
bor Wá
;
gner
;
Csaba Wé
;
ber
;
Olga Nyé
;
ki
;
Katalin Nó
;
grá
;
di
;
Attila Bielik
;
Lá
;
szló
;
Molná
r ;
Amrita Bobok
;
Attila Horvá
;
th
;
Bé
;
la Kiss
;
Sá
;
ndor
Kolok
关键词:
mGluR5
;
Negative allosteric modulator
;
Parallel synthesis
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
7.
Comparative pharmacology of adrenergic α
2C
receptors coupled to Ca
2+
signaling through different Gα proteins
作者:
Dalma Kurko
;
Zsó
;
fia Bekes
;
Anikó
;
Gere
;
Andrea Baki
;
Andrá
;
s Boros
;
Sá
;
ndor
Kolok
;
Gyula Bugovics
;
Jó
;
zsef Nagy
;
Zsolt Szombathelyi
;
Gyö
;
rgyi Igná
;
cz-Szendrei
关键词:
α
;
2C
-AR
;
Chimeric Gα
;
qi5
protein
;
Promiscuosus Gα
;
16
protein
;
Fluorometric Ca
2+
assay
;
High-throughput screening
刊名:Neurochemistry International
出版年:2009
8.
Kynurenic acid amides as novel NR2B selective NMDA receptor antagonists
作者:
Istvá
;
n Borza
;
Sá
;
ndor
Kolok
;
Korné
;
l Galgó
;
czy
;
Anikó
;
Gere
;
Csilla Horvá
;
th
;
Sá
;
ndor
Farkas
;
Istvá
;
n Greiner
;
Gyö
;
rgy Domá
;
ny
关键词:
NR2B antagonist
;
Kynurenic acid amide
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2007
9.
Functional characterization of sodium channel blockers by membrane potential measurements in cerebellar neurons: Prediction of compound preference for the open/inactivated state
作者:
Sá
;
ndor
Kolok
;
Jó
;
zsef Nagy
;
Zsolt Szombathelyi and Istvá
;
n Tarnawa
关键词:
Cerebellar neurons
;
Sodium channel blockers
;
Membrane potential fluorometry
;
Veratridine
;
GBR 12909
刊名:Neurochemistry International
出版年:2006
10.
Benzimidazole-2-carboxamides as novel NR2B selective NMDA receptor antagonists
作者:
Istvá
;
n Borza
;
Sá
;
ndor
Kolok
;
Anikó
;
Gere
;
Jó
;
zsef Nagy
;
Lá
;
szló
;
Fodor
;
Korné
;
l Galgó
;
czy
;
Jó
;
zsef Fetter
;
Ferenc Bertha
;
Bé
;
la Á
;
gai
;
Csilla Horvá
;
th
关键词:
NMDA
;
NR2B
;
Benzimidazole
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2006
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