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内部出版物
在“
Elsevier电子期刊
”中,
命中:
1,910
条,耗时:小于0.01 秒
1.
C0818, a novel curcumin derivative, interacts with
Hsp90
and inhibits Hsp90 ATPase activity
作者:
Yingjuan Fan
a
;
b
;
Yang Liu
a
;
b
;
Lianru Zhang
c
;
Fang Cai
a
;
b
;
Liping Zhu
a
;
b
;
Jianhua Xu
a
;
b
;
xjh@mail.fjmu.edu.cn
关键词:
Curcumin derivative
;
Hsp90
;
ATPase activity
;
Fluorescence spectrometry
;
Interaction
刊名:Acta Pharmaceutica Sinica B
出版年:2017
2.
Virtual screening and biophysical studies lead to
HSP90
inhibitors
作者:
Renjie Huang
;
Daniel M. Ayine-Tora
;
M. Nasri Muhammad Rosdi
;
Yu Li
;
Jó
;
hannes Reynisson
;
j.reynisson@auckland.ac.nz
;
Ivanhoe K.H. Leung
;
i.leung@auckland.ac.nz
关键词:
17-AAG
;
17-allylamino-17-demethoxygeldanamycin
;
17-DMAG
;
17-(dimethylaminoethylamino)-17-demethoxygeldanamycin (17-DMAG)
;
ADP
;
adenosine diphosphate
;
AMPPCP
;
5&prime
;
-adenylylmethylenediphosphonate
;
ASP
;
Astex statistical potential
;
ATP
;
adenosine triphosphate
;
CS
;
ChemScore
;
GS
;
GoldScore
;
HB
;
hydrogen bonding
;
HSP90
;
heat shock protein 90
;
HSQC
;
heteronuclear single quantum correlation
;
KD
;
binding affinity
;
ND
;
N-domain
;
NMR
;
nuclear magnetic resonance
;
NOE
;
nuclear Overhauser effect
;
Tm
;
pro
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
3.
Optimization and bioevaluation of Cdc37-derived peptides: An insight into
Hsp90
-Cdc37 protein-protein interaction modulators
作者:
Lei Wang
a
;
b
;
Li Li
a
;
b
;
Wei-Tao Fu
c
;
Zheng-Yu Jiang
a
;
b
;
Qi-Dong You
a
;
b
;
youqidong@gmail.com
;
Xiao-Li Xu
a
;
b
;
xiaoli_xu@126.com
关键词:
Protein-protein interaction
;
Hsp90
-Cdc37 PPI
;
Hot-spots
;
Peptides
;
MD simulation
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
4.
Synthesis and in vitro antiproliferative activity of C5-benzyl substituted 2-amino-pyrrolo[2,3-d]pyrimidines as potent
Hsp90
inhibitors
作者:
Ju-Hyeon Lee
a
;
c
;
1
;
Sang Chul Shin
b
;
d
;
1
;
Seon Hee Seo
a
;
Young Ho Seo
e
;
Nakcheol Jeong
c
;
Chan-Wha Kim
d
;
Eunice EunKyeong Kim
b
;
eunice@kist.re.kr
;
Gyochang Keum
a
;
gkeum@kist.re.kr
关键词:
Hsp90
;
Structure-based design
;
Cancer
;
Antiproliferative
;
Pyrrolo[2
;
3-d]pyrimidines
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
5.
Design, synthesis and biological evaluation of alkylamino biphenylamides as
Hsp90
C-terminal inhibitors
作者:
Gaurav Garg
;
Huiping Zhao
;
Brian S.J. Blagg
;
bblagg@ku.edu
关键词:
Heat shock protein 90
;
Hsp90
C-terminal inhibitors
;
Alkylamino biphenylamides
;
Structure-activity relationship
;
Breast cancer
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
6.
Design, synthesis and biological evaluation of 7-(aryl)-2,3-dihydro-[1,4]dioxino[2,3-g]quinoline derivatives as potential
Hsp90
inhibitors and anticancer agents
作者:
Sina Omid Malayeri
a
;
b
;
Khalil Abnous
c
;
Atefeh Arab
d
;
Maryam Akaberi
e
;
Soghra Mehri
c
;
Afshin Zarghi
f
;
Razieh Ghodsi
a
;
b
;
ghodsir@mums.ac.ir
关键词:
Quinolines
;
Heat Shock Protein 90
;
Anti-cancer activity
;
Her2
;
Molecular docking
;
Hsp90
inhibitor
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
7.
Design, synthesis and pharmacological evaluation of 4,5-diarylisoxazols bearing amino acid residues within the 3-amido motif as potent heat shock protein 90 (
Hsp90
) inhibitors
作者:
Chi Zhang
a
;
c
;
1
;
Xin Wang
b
;
d
;
1
;
Hongchun Liu
b
;
Minmin Zhang
b
;
Meiyu Geng
b
;
Liping Sun
a
;
chslp@cpu.edu.cn
;
Aijun Shen
b
;
shenaj@simm.ac.cn
;
Ao Zhang
c
;
aozhang@simm.ac.cn
关键词:
Diarylisoxazole
;
Resorcinol
;
Amino acid
;
Hsp90
inhibitor
;
Antiproliferative effect
刊名:European Journal of Medicinal Chemistry
出版年:2017
8.
Spontaneous assembly of
HSP90
inhibitors at water/octanol interface: A molecular dynamics simulation study
作者:
Amin Reza Zolghadr
;
arzolghadr@shirazu.ac.ir
;
Samaneh Boroomand
关键词:
HSP90
inhibitors
;
Water/octanol interface
;
Molecular dynamics simulation
刊名:Chemical Physics Letters
出版年:2017
9.
Topically Applied
Hsp90
Blocker 17AAG Inhibits Autoantibody-Mediated Blister-Inducing Cutaneous Inflammation
作者:
Stefan Tukaj
1
;
2
;
5
;
Katja Bieber
3
;
5
;
Konrad Kleszczyński
1
;
Mareike Witte
1
;
Rebecca Cames
1
;
Kathrin Kalies
4
;
Detlef Zillikens
1
;
3
;
Ralf J. Ludwig
1
;
3
;
Tobias W. Fischer
1
;
Michael Kasperkiewicz
1
;
Michael.Kasperkiewicz@uksh.de
关键词:
17AAG
;
17-allylamino-demethoxygeldanamycin
;
COL7
;
type VII collagen
;
EBA
;
epidermolysis bullosa acquisita
;
MMP
;
matrix metalloproteinase
;
PBS
;
phosphate buffered saline
;
qRT-PCR
;
quantitative real-time reverse transcriptase-PCR
;
RT
;
room temperature
刊名:Journal of Investigative Dermatology
出版年:2017
10.
HSP70 and
HSP90
are involved in shrimp Penaeus vannamei tolerance to AHPND-causing strain of Vibrio parahaemolyticus after non-lethal heat shock
作者:
Wisarut Junprung
a
;
Premruethai Supungul
b
;
Anchalee Tassanakajon
a
;
anchalee.k@chula.ac.th
关键词:
Heat shock protein
;
Penaeus vannamei
;
Vibrio parahaemolyticus
;
Acute hepatopancreatic necrosis disease
;
Chronic heat stress
刊名:Fish & Shellfish Immunology
出版年:2017
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