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CNKI期刊论文0611(1)
知网期刊论文(1149)
在“
Elsevier电子期刊
”中,
命中:
2,508
条,耗时:0.0289862 秒
在所有数据库中总计命中:
4,710
条
1.
Imidazo[1,2-a]pyrazin-8-amine core for the design of new
adenosine
receptor
antagonist
s: Structural exploration to target the A
3
and A
2A
subtypes
作者:
Daniela Poli
a
;
Matteo Falsini
a
;
Flavia Varano
a
;
Marco Betti
a
;
Katia Varani
b
;
Fabrizio Vincenzi
b
;
Anna Maria Pugliese
c
;
Felicita Pedata
c
;
Diego Dal Ben
d
;
Ajiroghene Thomas
d
;
Ilaria Palchetti
e
;
f
;
Francesca Bettazzi
e
;
Daniela Catarzi
a
;
daniela.catarzi@unifi.it
;
Vittoria Colotta
a
关键词:
G protein-coupled receptors
;
Adenosine
receptor
antagonist
s
;
Imidazopyrazines
;
Bicyclic heteroaromatic systems
;
Ligand-receptor modeling studies
刊名:European Journal of Medicinal Chemistry
出版年:2017
2.
Synthesis and evaluation of N-substituted 2-amino-4,5-diarylpyrimidines as selective
adenosine
A
1
receptor
antagonist
s
作者:
Georgios Alachouzos
;
Eelke B. Lenselink
;
Thea Mulder-Krieger
;
Henk de Vries
;
Adriaan P. IJzerman
;
Julien Louvel
;
j.a.louvel@lacdr.leidenuniv.nl
关键词:
Structure-affinity relationships
;
Adenosine
A1 receptor
;
Adenosine
A2A receptor
;
Selectivity
;
Antagonist
s
刊名:European Journal of Medicinal Chemistry
出版年:2017
3.
Selected C8 two-chain linkers enhance the
adenosine
A
1
/A
2A
receptor affinity and selectivity of caffeine
作者:
M.M. van der Walt
a
;
dalenevanderwalt@gmail.com
;
13035134@nwu.ac.za
;
G. Terre'Blanche
a
;
b
关键词:
Caffeine
;
Adenosine
A2A receptor
antagonist
;
Adenosine
A1 receptor
antagonist
;
1
3 ;
7-trimethylxanthine
;
Parkinson's disease
刊名:European Journal of Medicinal Chemistry
出版年:2017
4.
A
2B
adenosine
receptor
antagonist
s: Design, synthesis and biological evaluation of novel xanthine derivatives
作者:
Sujay Basu
a
;
b
;
c
;
sujay.basu@advinus.com
;
Dinesh A. Barawkar
a
;
b
;
c
;
Vidya Ramdas
a
;
b
;
c
;
Yogesh Waman
a
;
b
;
c
;
Meena Patel
a
;
b
;
c
;
Anil Panmand
a
;
b
;
c
;
Santosh Kumar
a
;
b
;
c
;
Sachin Thorat
a
;
b
;
c
;
Rajesh Bonagiri
a
;
b
;
c
;
Dilip Jadhav
a
;
b
;
c
;
Partha Mukhopadhyay
a
;
b
;
c
;
Vandna Prasad
a
;
b
;
c
;
B. Srinivasa Reddy
a
;
b
;
c
;
Arnab Goswami
a
;
b
;
c
;
Sandhya Chaturvedi
a
;
b
;
c
;
Suraj Menon
a
;
b
;
c
;
Azfar Quraishi
a
;
b
;
c
;
Indraneel Ghosh
a
;
b
;
c
;
Sushant Dusange
a
;
b
;
c
;
Shalini Paliwal
a
;
b
;
c
;
Abhay Kulkarni
a
;
b
;
c
;
Vikas Karande
a
;
b
;
c
;
Rhishikesh Thakre
a
;
b
;
c
;
Gaurav Bedse
a
;
b
;
c
;
Sreekanth Rouduri
a
;
b
;
c
;
Jayasagar Gundu
a
;
b
;
c
;
Venkata P. Palle
a
;
b
;
c
;
Anita Chugh
a
;
b
;
c
;
Kasim A. Mookhtiar
a
;
b
;
c
;
kasim.mookhtiar@advinus.com
关键词:
Adenosine
receptors
;
Xanthine
;
2-Oxopyrrolidine
;
Mouse liver microsomes
;
Pharmacokinetics
刊名:European Journal of Medicinal Chemistry
出版年:2017
5.
Adenosine
A
2A
and A
2B
Receptors Differentially Modulate Keratinocyte Proliferation: Possible Deregulation in Psoriatic Epidermis
作者:
Rosa M. André
;
s
1
;
2
;
Marí
;
a Carmen Terencio
1
;
2
;
Jorge Arasa
1
;
2
;
Miguel Payá
;
1
;
2
;
Francisca Valcuende-Cavero
3
;
4
;
Pedro Navaló
;
n
5
;
Marí
;
a Carmen Montesinos
1
;
2
;
m.carmen.montesinos@uv.es
关键词:
AR
;
adenosine
receptors
;
BAY
;
BAY60&ndash
;
6583
;
CGS
;
CGS-21680
;
iCa2+
;
intracellular calcium
;
MRS
;
MRS-1706
;
MTT
;
3-(4
;
5-dimethylthiazol-2-yl)-2
;
5-diphenyltetrazolium bromide
;
NECA
;
5'-N-ethylcarboxamido
adenosine
;
NHEK
;
normal human epidermal keratinocyte
;
SCH
;
SCH-442416
;
TNF
;
tumor necrosis factor
;
TPA
;
12-O-tetradecanoylphorbol-13-acetate
刊名:Journal of Investigative Dermatology
出版年:2017
6.
Purinergic signaling in kidney disease
作者:
Robert I. Menzies
1
;
Frederick W. Tam
2
;
Robert J. Unwin
3
;
4
;
robert.unwin@ucl.ac.uk
;
Matthew A. Bailey
1
关键词:
adenosine
;
ATP
;
inflammation
;
kidney
;
P2X
;
P2Y
;
renal tubule
;
vasculature
刊名:Kidney International
出版年:2017
7.
Impact on monoclonal antibody production in murine hybridoma cell cultures of
adenosine
receptor
antagonist
s and phosphodiesterase inhibitors
作者:
Geoffrey F. Kelso
;
Shahid A. Kazi
;
Simon J. Harris
;
Reinhard I. Boysen
;
Jamil Chowdhury
;
Milton T.W. Hearn
;
milton.hearn@monash.edu" class="auth_mail" title="E-mail the corresponding author
关键词:
Monoclonal antibody
;
Hybridoma
;
Adenosine
antagonist
;
Phosphodiesterase inhibitor
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
8.
Discovery of aminoquinazoline derivatives as human A
2A
adenosine
receptor
antagonist
s
作者:
Gang Zhou
a
;
;
Robert Aslanian
b
;
Gioconda Gallo
a
;
Tanweer Khan
b
;
Rongze Kuang
a
;
Biju Purakkattle
b
;
Manuel De Ruiz
c
;
Andrew Stamford
a
;
Pauline Ting
a
;
Heping Wu
a
;
Hongwu Wang
b
;
Dong Xiao
b
;
Tao Yu
a
;
Yonglian Zhang
a
;
Deborra Mullins
b
;
Robert Hodgson
b
关键词:
Adenosine
A2A receptor
antagonist
;
Aminoquinazoline
;
Parkinson&rsquo
;
s disease
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
9.
Activation of transient receptor potential vanilloid 1 accelerates re-endothelialization and inhibits neointimal formation after vascular injury
作者:
Linan Su
;
MD
;
MSc
;
Yunrong Zhang
;
MD
;
Kecheng He
;
MD
;
MSc
;
Shujie Wei
;
MD
;
Haifeng Pei
;
MD
;
PhD
;
Qiang Wang
;
MD
;
PhD
;
Dachun Yang
;
MD
;
PhD
;
yangdc71@126.com
;
Yongjian Yang
;
MD
;
PhD
刊名:Journal of Vascular Surgery
出版年:2017
10.
5,7-Disubstituted-[1,2,4]triazolo[1,5-a][1,3,5]triazines as pharmacological tools to explore the
antagonist
selectivity profiles toward
adenosine
receptors
作者:
Stephanie Federico
a
;
Antonella Ciancetta
b
;
Nicola Porta
b
;
Sara Redenti
a
;
Giorgia Pastorin
c
;
Barbara Cacciari
d
;
Karl Norbert Klotz
e
;
Stefano Moro
b
;
stefano.moro@unipd.it" class="auth_mail" title="E-mail the corresponding author
;
Giampiero Spalluto
a
;
spalluto@units.it" class="auth_mail" title="E-mail the corresponding author
关键词:
G protein-coupled receptor
;
Antagonist
s
;
Molecular modeling
;
Structure activity relationship
;
Triazolo-triazine
;
Adenosine
receptors
刊名:European Journal of Medicinal Chemistry
出版年:2016
1
2
3
4
5
6
7
8
9
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