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内部出版物
在“
Elsevier电子期刊
”中,
命中:
6
条,耗时:小于0.01 秒
1.
4,4-Dimethyl-1,2,3,4-tetrahydroquinoline-based PPARα/γ agonists. Part. II: Synthesis and pharmacological evaluation of oxime and acidic head group structural variations
作者:
Cé
;
cile Parmenon
;
Jé
;
rô
;
me Guillard
;
Daniel-Henri Caignard
;
Nathalie Hennuyer
;
Bart Staels
;
Valé
;
rie Audinot-Bouchez
;
Jean-Albert Boutin
;
Catherine Dacquet
;
Alain
Ktorza
;
Marie-Claude
关键词:
PPARs
;
Terahydroquinoline
;
Oxime
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
2.
4,4-Dimethyl-1,2,3,4-tetrahydroquinoline-based PPARα/γ agonists. Part I: Synthesis and pharmacological evaluation
作者:
Cé
;
cile Parmenon
;
Jé
;
rô
;
me Guillard
;
Daniel-Henri Caignard
;
Nathalie Hennuyer
;
Bart Staels
;
Valé
;
rie Audinot-Bouchez
;
Jean-Albert Boutin
;
Catherine Dacquet
;
Alain
Ktorza
;
Marie-Claude
关键词:4 ;
4-Dimethyl-1
23 ;
4-tetrahydroquinoline
;
PPAR
;
//www.sciencedirect.com/scidirimg/entities/204e.gif"" alt=""greek small letter alpha"" title=""greek small letter alpha"" border=""0"">/γ
;
agonists
;
Diabetes type-2
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2008
3.
Design and synthesis of novel imidazoline derivatives with potent antihyperglycemic activity in a rat model of type 2 diabetes
作者:
Louis Crane
;
Maria Anastassiadou
;
Salomé
;
El Hage
;
Jean Luc Stigliani
;
Geneviè
;
ve Baziard-Mouysset
;
Marc Payard
;
Jean Michel Leger
;
Jean-Guy Bizot-Espiard
;
Alain
Ktorza
;
Daniel-Henri Caignard
刊名:Bioorganic and Medicinal Chemistry
出版年:2006
4.
Structural requirements of the N-terminal region of GLP-1-[7-37]-NH
2
for receptor interaction and cAMP production
作者:
Cyril Sarrauste de Menthiè
;
re
;
Alain
Chavanieu
;
Gé
;
rard Grassy
;
Sté
;
phane Dalle
;
Guillermo Salazar
;
Alain
Kervran
;
Bruno Pfeiffer
;
Pierre Renard
;
Philippe Delagrange
;
Dominique Manechez
;
David Bakes
;
Alain
Ktorza
;
Bernard Calas
关键词:
Glucagon-Like Peptide-1
;
Structure-activity relationships
;
Plasma stability
;
Glucose tolerance test
;
Conformations
;
Circular dichroism
刊名:European Journal of Medicinal Chemistry
出版年:2004
5.
A better understanding of the pathophysiology of obesity and type 2 diabetes: a clue for new therapeutic approaches
作者:
Antoine Bril
;
Alain
Ktorza
刊名:Current Opinion in Pharmacology
出版年:2006
6.
A specific β
3
-adrenoceptor agonist induces increased pancreatic islet blood flow and insulin secretion in rats
作者:
Atef
;
Nadia
;
Lafontan
;
Max
;
Doublé
;
Alexandre
;
Hé
;
lary
;
Christophe
;
Ktorza
;
Alain
;
et. al.
关键词:
Glucose
;
Insulin
;
Pancreatic islet
;
blood flow
;
Blood pressure
;
β
;
-Adrenoceptor
刊名:European Journal of Pharmacology
出版年:1996
1
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