搜索页_+Aminopiperidine

设为首页

收藏本站

网站地图 | English | 公务邮箱

About the library

Background
History
Leadership
Organization

Readers' Guide

Opening Hours
Collections
Help Via Email

Publications

Electronic Information Resources

常用资源

在“Elsevier电子期刊”中，命中：75条，耗时：小于0.01 秒

1.Identification of novel aminopiperidine derivatives for antibacterial activity against Gram-positive bacteria

作者：Hee-Yeol Lee ; Kyung-Mi An ; Juyoung Jung ; Je-Min Koo ; Jeong-Geun Kim ; Jong-Min Yoon ; Myong-Jae Lee ; HyeonSoo Jang ; Hong-Sub Lee ; Soobong Park ; Jae-Hoon Kang ; ^{jhkang@ildong.com" class="auth_mail" title="E-mail the corresponding author}

关键词：Peptide deformylase ; Antibacterial ; Gram-positive ; Resistant ; Aminopiperidine

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

2.Replacement of cardiotoxic aminopiperidine linker with piperazine moiety reduces cardiotoxicity? Mycobacterium tuberculosis novel bacterial topoisomerase inhibitors

作者：Karyakulam Andrews Bobesh^a ; ^&dagger ; ; Janupally Renuka^a ; ^&dagger ; ; Rudraraju Reshma Srilakshmi^a ; Swapna Yellanki^b ; ^c ; Pushkar Kulkarni^b ; ^c ; Perumal Yogeeswari^a ; Dharmarajan Sriram^a ; ^{dsriram@hyderabad.bits-pilani.ac.in" class="auth_mail" title="E-mail the corresponding author}

关键词：DNA gyrase ; Topoisomerase ; Tuberculosis ; 1 ; 5-Naphthyridin-2(1H)-one ; zERG toxicity

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

3.Pyrazole antagonists of the CB1 receptor with reduced brain penetration

作者：Alan Fulp ; Yanan Zhang ; Katherine Bortoff ; Herbert Seltzman ; Rodney Snyder ; Robert Wiethe ; George Amato ; Rangan Maitra ; ^{rmaitra@rti.org" class="auth_mail" title="E-mail the corresponding author}

关键词：BBB ; blood&ndash ; brain barrier ; BOP ; benzotriazol-1-yl-oxytris(dimethylamino)phosphonium hexafluorophosphate ; CB ; cannabinoid receptors ; CB1 ; cannabinoid receptor 1 ; CB2 ; cannabinoid receptor 2 ; CHO-K1 ; Chinese hamster ovary cells ; CMA 80 ; 80% chloroform ; 18% methanol ; and 2% ammonium hydroxide ; CNS ; central nervous system ; Ke ; apparent affinity constant ; MDCK-mdr1 ; Madin&ndash ; Darby canine kidney cells transfected with the human MDR1 gene ; IP3 ; inositol phosphatase 3 ; MRM ; multiple reaction mon

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

4.Development of acridine derivatives as selective Mycobacterium tuberculosis DNA gyrase inhibitors

作者：Brahmam Medapi^a ; Nikhila Meda^a ; Pushkar Kulkarni^b ; Perumal Yogeeswari^a ; Dharmarajan Sriram^a ; ^{dsriram@hyderabad.bits-pilani.ac.in" class="auth_mail" title="E-mail the corresponding author}

关键词：Tuberculosis ; DNA gyrase ; Acridine derivatives

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

5.Kinetic modeling of the synthesis of N-aminopiperidine via the Raschig process: Reaction optimization and continuous process

作者：C. Darwich ; M. Elkhatib ; V. Pasquet ; H. Delalu

关键词：Kinetic modeling ; Synthesis optimization ; Raschig process ; N-aminopiperidine

刊名：Chemical Engineering Journal

出版年：15 March, 2014

6.Development of novel N-linked aminopiperidine-based mycobacterial DNA gyrase B inhibitors: Scaffold hopping from known antibacterial leads

作者：Variam Ullas Jeankumar^a ; Janupally Renuka^a ; Venkat Koushik Pulla^a ; Vijay Soni^a ; Jonnalagadda Padma Sridevi^a ; Priyanka Suryadevara^a ; Morla Shravan^a ; Raghavender Medishetti^b ; ^c ; Pushkar Kulkarni^b ; ^c ; Perumal Yogeeswari^a ; Dharmarajan Sriram^a ; ^{dsriram@hyderabad.bits-pilani.ac.in" class="auth_mail} ; ^{drdsriram@yahoo.com" class="auth_mail}

关键词：Tuberculosis ; DNA gyrase ; GyrB domain ; Aminopiperidine

刊名：International Journal of Antimicrobial Agents

出版年：March, 2014

7.Design and synthesis of an aminopiperidine series of 纬-secretase modulators

作者：Tomonori Kobayashi ; Seiji Iwama ; Akira Fusano ; Yoshihiro Kato ; Atsushi Ikeda ; Yasuhiro Teranishi ; Akemi Nishihara ; Masanori Tobe

关键词：Alzheimer&rsquo ; s disease ; 纬-Secretase modulator ; 纬-Secretase inhibitor ; Amyloid 尾 peptide ; Piperidine

刊名：Bioorganic and Medicinal Chemistry Letters

出版年：1 January, 2014

8.A concise enantioselective synthesis of l-(−)-733,061 and (2S,3S)-methyl 3-aminopiperidine-2-carboxylate using catalytic enantioselective aza-Henry reaction as key step

作者：Gullapalli Kumaraswamy ; ^a ; ^{gkswamy_iict@yahoo.co.in} ; Arigala Pitchaiah^a

关键词：Organocatalysis ; Piperidine motif ; l-(− ; )-733061 ; (2S ; 3S)-Methyl 3-aminopiperidine-2-carboxylate ; aza-Henry reaction ; Febrifugine ; Glycosidase inhibitors

刊名：Tetrahedron

出版年：2011

9.Thiazole-aminopiperidine hybrid analogues: Design and synthesis of novel Mycobacterium tuberculosis GyrB inhibitors

作者：Variam Ullas Jeankumar ; Janupally Renuka ; Peddi Santosh ; Vijay Soni ; Jonnalagadda Padma Sridevi ; Priyanka Suryadevara ; Perumal Yogeeswari ; Dharmarajan Sriram

关键词：Tuberculosis ; DNA gyrase ; GyrB subunit ; Thiazole ; Amino piperidine

刊名：European Journal of Medicinal Chemistry

出版年：December, 2013

10.Evaluation of a 4-aminopiperidine replacement in several series of CCR5 antagonists

作者：Ré ; my C. Lemoine ; Ann C. Petersen ; Lina Setti ; Lijing Chen ; Jutta Wanner ; Andreas Jekle ; Gabrielle Heilek ; André ; deRosier ; Changhua Ji ; David M. Rotstein

关键词：5-Amino-3-azabicyclo[3.3.0]octane ; 4-Aminopiperidine ; Replacement ; CCR5 antagonists ; Chemokine receptor

刊名：Bioorganic and Medicinal Chemistry Letters

出版年：2010

按检索点细分(75)

题名(38)

关键词(18)

文摘(56)

按出版年细分(75)

2027年及以后(2)

2016年(4)

2013年(3)

2012年(4)

2011年(4)

2010年(4)

2009年(3)

2008年(5)

2007年(7)

2006年(6)

2005年(7)

2004年(1)

2003年(6)

2001年(5)

2000年(1)

2000年及以前(13)