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内部出版物
在“
Elsevier电子期刊
”中,
命中:
9
条,耗时:小于0.01 秒
1.
Acute myeloid leukemia with t(16;16) (p13;q22) showing a new CBFB-MYH11 fusion transcript associated with an atypical leukemic blasts morphology
作者:
Francesco Albano
;
Luisa Anelli
;
Antonella Zagaria
;
Nicoletta Coccaro
;
Giuseppina Tota
;
Luciana Impera
;
Crescenzio Francesco Minervini
;
Angelo
Cellamare
;
Mario Delia
;
Angela Minervini
;
Paola Casieri
;
Giorgina Specchia
关键词:
t(16
;
16)
;
CBFB-MYH11 fusion gene
;
Fusion transcript variants
;
Bilobed leukemic blast
刊名:Human Pathology
出版年:March, 2014
2.
Design, synthesis and biological evaluation of coumarin alkylamines as potent and selective dual binding site inhibitors of acetylcholinesterase
作者:
Marco Catto
;
marco.catto@uniba.it
;
Leonardo Pisani
;
Francesco Leonetti
;
Orazio Nicolotti
;
Paolo Pesce
;
Angela Stefanachi
;
Saverio
Cellamare
;
Angelo
Carotti
;
angelo
.carotti@uniba.it
关键词:
Alzheimer&rsquo
;
s disease
;
Coumarin derivatives
;
Acetylcholinesterase
;
Dual binding site inhibitors
;
Selective cholinesterase inhibition
刊名:Bioorganic and Medicinal Chemistry
出版年:2013
3.
Design, synthesis and biological evaluation of 5-hydroxy, 5-substituted-pyrimidine-2,4,6-triones as potent inhibitors of gelatinases MMP-2 and MMP-9
作者:
Orazio Nicolotti
;
orazio.nicolotti@uniba.it
;
Marco Catto
;
Ilenia Giangreco
;
Maria Barletta
;
Francesco Leonetti
;
Angela Stefanachi
;
Leonardo Pisani
;
Saverio
Cellamare
;
Paolo Tortorella
;
Fulvio Loiodice
;
Angelo
Carotti
;
angelo
.carotti@uniba.it
关键词:
MMP
;
Gelatinases
;
ZBG
;
QSAR
;
Molecular docking
刊名:European Journal of Medicinal Chemistry
出版年:2012
4.
Toward a fragment-based approach to MMPs inhibitors: an expedite and efficient synthesis of N-hydroxylactams
作者:
Francesco Leonetti
;
Giovanni Muncipinto
;
Angela Stefanachi
;
Orazio Nicolotti
;
Saverio
Cellamare
;
Marco Catto
;
Leonardo Pisani
;
Giovanni Pellegrino
;
Angelo
Carotti
关键词:
Ring closing metathesis
;
N-Hydroxylactams
;
Metalloproteinase inhibitors
;
Zinc-enzymes
刊名:Tetrahedron Letters
出版年:2012
5.
Design, synthesis and biological evaluation of indane-2-arylhydrazinylmethylene-1,3-diones and indol-2-aryldiazenylmethylene-3-ones as β-amyloid aggregation inhibitors
作者:
Marco Catto
;
Rosaria Aliano
;
Angelo
Carotti
;
Saverio
Cellamare
;
Fausta Palluotto
;
Rosa Purgatorio
;
Angelo
De Stradis
;
Francesco Campagna
关键词:
β
;
-Amyloid peptide
;
Alzheimer's disease
;
Amyloid aggregation inhibitors
刊名:European Journal of Medicinal Chemistry
出版年:2010
6.
1,3-Dialkyl-8-(hetero)aryl-9-OH-9-deazaxanthines as potent A
2B
adenosine receptor antagonists: Design, synthesis, structure–affinity and structure–selectivity relationships
作者:
Angela Stefanachi
;
Orazio Nicolotti
;
Francesco Leonetti
;
Saverio
Cellamare
;
Francesco Campagna
;
Maria Isabel Loza
;
Jose Manuel Brea
;
Fern
;
o Mazza
;
Enrico Gavuzzo
;
Angelo
Carotti
关键词:1 ;
3-Dialkyl-8-(hetero)aryl-9-OH-9-deazaxanthines
;
Adenosine receptor antagonists
;
Structure–
;
affinity relationships
;
Structure–
;
selectivity relationships
;
X-ray crystallography
刊名:Bioorganic and Medicinal Chemistry
出版年:2008
7.
Design, synthesis, and biological evaluation of glycine-based molecular tongs as inhibitors of Aβ
1–40
aggregation in vitro
作者:
Saverio
Cellamare
;
Angela Stefanachi
;
Diana A. Stolfa
;
Teodora Basile
;
Marco Catto
;
Francesco Campagna
;
Eddy Sotelo
;
Pasquale Acquafredda
;
Angelo
Carotti
关键词:
Aβ
;
1–
;
40
;
β
;
-Amyloid aggregation
;
Glycine-based molecular tongs
;
Polyphenolic amides inhibitors
刊名:Bioorganic and Medicinal Chemistry
出版年:2008
8.
Insights into structure–activity relationships from lipophilicity profiles of pyridin-2(1H)-one analogs of the cardiotonic agent milrinone
作者:
Modesto de Candia
;
Paola Fossa
;
Saverio
Cellamare
;
Luisa Mosti
;
Angelo
Carotti and Cosimo Altomare
关键词:
Milrinone analogs
;
Positive inotropic effects
;
Lipophilicity
;
Tautomerism
刊名:European Journal of Pharmaceutical Sciences
出版年:2005
9.
Isoquinoline derivatives as endogenous neurotoxins in the aetiology of Parkinsons disease
作者:
McNaught
;
Kevin St. P.
;
Carrupt
;
Pierre-Alain
;
Altomare
;
Cosimo
;
Cellamare
;
Saverio
;
Carotti
;
Angelo
;
et. al.
关键词:
isoquinoline derivatives
;
1-methyl-4-phenyl-1
23 ;
6-tetrahydropyridine (MPTP)
;
1-methyl-4-phenylpyridinium (MPP
+
)
;
1
23 ;
4-tetrahydroisoquinoline
;
neurotoxin
;
Parkinson
;
s disease
刊名:Biochemical Pharmacology
出版年:1998
1
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