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内部出版物
CNKI学位论文(18)
在“
Elsevier电子期刊
”中,
命中:
13
条,耗时:小于0.01 秒
在所有数据库中总计命中:
18
条
1.
Synthesis, cytostatic activity and AD
M
E properties of C-5 substituted and N-acyclic pyri
m
idine derivatives
作者:
Tatjana Gazivoda
Kral
jevi?
a
;
M
ateja Klika
a
;
M
arijeta
Kral
j
b
;
Irena
M
artin-Kleiner
b
;
Stella Jur
m
anovi?
c
;
Astrid
M
ili?
c
;
Jasna Padovan
c
;
Silvana Rai?-
M
ali?
a
;
sraic@fkit.hr
关键词:
5-Alkyl pyri
m
idine derivatives
;
Cytostatic evaluations
;
Cell cycle analysis
;
AD
M
E properties
刊名:Bioorganic and
M
edicinal Che
m
istry Letters
出版年:2012
2.
Parallel
m
edicinal che
m
istry approaches to selective HDAC1/HDAC2 inhibitor (SHI-1:2) opti
m
ization
作者:
Solo
m
on D. Kattar
;
Laura
M
. Surdi
;
Anna Zabierek
;
Joey L.
M
ethot
;
Richard E.
M
iddleton
;
Bethany Hughes
;
Alex
;
er A. Szewczak
;
Willia
m
K. Dahlberg
;
Astrid
M
.
Kral
;
Nicole Ozerova
;
Judith C. Fle
m
ing
;
Hon
关键词:
Histone deacetylases
;
Parallel synthesis
刊名:Bioorganic and
M
edicinal Che
m
istry Letters
出版年:2009
3.
Exploring the phar
m
acokinetic properties of phosphorus-containing selective HDAC 1 and 2 inhibitors (SHI-1:2)
作者:
Richard W. Heidebrecht Jr.
;
M
elissa Chenard
;
Joshua Close
;
Willia
m
K. Dahlberg
;
Judith Fle
m
ing
;
Jonathan B. Gri
mm
;
Julie E. Ha
m
ill
;
Andreas Harsch
;
Brian B. Haines
;
Bethany Hughes
;
Astrid
M
.
Kral
;
Ric
关键词:
Phar
m
acokinetics
;
Selective histone deacetylase inhibitor
;
Zolinza
;
Xenograft
;
Phosphorus-containing therapeutic
刊名:Bioorganic and
M
edicinal Che
m
istry Letters
出版年:2009
4.
Rapid asse
m
bly of diverse and potent allosteric Akt inhibitors
作者:
Zhicai Wu
;
Ronald G. Robinson
;
Sheng Fu
;
Stanley F. Barnett
;
Deborah Defeo-Jones
;
Ray
m
ond E. Jones
;
Astrid
M
.
Kral
;
Hans E. Huber
;
Nancy E. Kohl
;
George D. Hart
m
an
;
M
ark T. Bilodeau
关键词:
Akt inhibitor
;
Allosteric
;
Rapid asse
m
bly
;
Cancer
;
Kinase
刊名:Bioorganic and
M
edicinal Che
m
istry Letters
出版年:2008
5.
Phenylglycine and phenylalanine derivatives as potent and selective HDAC1 inhibitors (SHI-1)
作者:
Kevin J. Wilson
;
David J. Witter
;
Jonathan B. Gri
mm
;
Phieng Siliphaivanh
;
Karin
M
. Otte
;
Astrid
M
.
Kral
;
Judith C. Fle
m
ing
;
Andreas Harsch
;
Julie E. Ha
m
ill
;
Jonathan C. Cruz
;
M
elissa Chenard
;
Alex
;
er
关键词:
HDAC1 inhibitor
;
Selective
;
Biaryl
;
Benza
m
ide
刊名:Bioorganic and
M
edicinal Che
m
istry Letters
出版年:2008
6.
Develop
m
ent of Pyridopyri
m
idines as Potent Akt1/2 Inhibitors
作者:
Zhicai Wu
;
John C. Hartnett
;
Lou Anne Neilson
;
Ronald G. Robinson
;
Sheng Fu
;
Stanley F. Barnett
;
Deborah Defeo-Jones
;
Ray
m
ond E. Jones
;
Astrid
M
.
Kral
;
Hans E. Huber
;
George D. Hart
m
an
;
M
ark T. Bilod
关键词:
Akt
;
Kinase
;
Cancer
;
Pyridopyri
m
idine
刊名:Bioorganic and
M
edicinal Che
m
istry Letters
出版年:2008
7.
A
m
ino acid derivatives as histone deacetylase inhibitors
作者:
Jed L. Hubbs
;
Hua Zhou
;
Astrid
M
.
Kral
;
Judith C. Fle
m
ing
;
Willia
m
K. Dahlberg
;
Bethany L. Hughes
;
Richard E.
M
iddleton
;
Alex
;
er A. Szewczak
;
J. Paul Secrist
;
Tho
m
as A. Miller
关键词:
Histone deacetylase
;
Cancer
;
Ugi reaction
;
Lysine
;
A
m
ino acid
;
Benzothiophene
刊名:Bioorganic and
M
edicinal Che
m
istry Letters
出版年:2008
8.
Opti
m
ization of biaryl Selective HDAC1&2 Inhibitors (SHI-1:2)
作者:
David J. Witter
;
Paul Harrington
;
Kevin J. Wilson
;
M
elissa Chenard
;
Judith C. Fle
m
ing
;
Brian Haines
;
Astrid
M
.
Kral
;
J. Paul Secrist
;
Tho
m
as A. Miller
关键词:
Histone deacetylase
;
HDAC
;
A
m
inobenza
m
ides
;
Biaryl
刊名:Bioorganic and
M
edicinal Che
m
istry Letters
出版年:2008
9.
Opti
m
ization of 2,3,5-trisubstituted pyridine derivatives as potent allosteric Akt1 and Akt2 inhibitors
作者:
John C. Hartnett
;
Stanley F. Barnett
;
M
ark T. Bilodeau
;
Deborah Defeo-Jones
;
George D. Hart
m
an
;
Hans E. Huber
;
Ray
m
ond E. Jones
;
Astrid
M
.
Kral
;
Ronald G. Robinson
;
Zhicai Wu
关键词:
Inhibitors
;
Akt1
;
Akt2
;
Enzy
m
atic
;
Cellular
刊名:Bioorganic and
M
edicinal Che
m
istry Letters
出版年:2008
10.
Functional analysis of a Drosophila
m
elanogaster olfactory receptor expressed in Sf9 cells
作者:
Aidan Kiely
;
Astrid
Authier
;
Andrew V.
Kral
icek
;
Coral G. Warr
;
Richard D. Newco
m
b
关键词:
Olfactory receptor
;
Calciu
m
i
m
aging
;
Olfaction
;
Sf9
;
Odorant
;
Or22a
刊名:Journal of Neuroscience
M
ethods
出版年:2007
1
2
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作者(13)
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2009年(2)
2008年(6)
2007年(3)
2000年及以前(1)
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