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CNKI会议论文(6)
CNKI学位论文(16155)
CNKI期刊论文0611(11)
知网期刊论文(7795)
在“
Elsevier电子期刊
”中,
命中:
2,914
条,耗时:0.0339832 秒
在所有数据库中总计命中:
23,967
条
1.
Synthesis,
COX
-1/
2
inhibition
activities and molecular docking study of isothiazolopyridine derivatives
作者:
Piotr Świątek
a
;
piotr.swiatek@umed.wroc.pl
;
Malgorzata Strzelecka
a
;
Rafal Urniaz
b
;
Katarzyna Gębczak
c
;
Tomasz Gębarowski
c
;
Kazimierz Gąsiorowski
c
;
Wieslaw Malinka
a
关键词:
Isothiazolopyridine
;
Cyclooxygenase
inhibition
;
Molecular docking
刊名:Bioorganic & Medicinal Chemistry
出版年:
2
017
2.
Design, synthesis and analgesic/anti-inflammatory evaluation of novel diarylthiazole and diarylimidazole derivatives towards selective
COX
-1 inhibitors with better gastric profile
作者:
Ahmed H. Abdelazeem
a
;
b
;
ahmed.abdelazeem@pharm.bsu.edu.eg
;
ahmed.pharm@yahoo.com
;
Mohammed T. El-Saadi
a
;
Asmaa G. Safi El-Din
a
;
Hany A. Omar
c
;
d
;
Samir M. El-Moghazy
e
;
samirelmoghazy@gmail.com
关键词:
Selective
COX
-1
;
Mofezolac
;
Diarylthiazole
;
Diarylimidazole
;
Analgesic
;
Anti-inflammatory
;
Ulcerogenicity
刊名:Bioorganic & Medicinal Chemistry
出版年:
2
017
3.
A traditional Chinese formula composed of Chuanxiong Rhizoma and Gastrodiae Rhizoma (Da Chuanxiong Formula) suppresses inflammatory response in LPS -induced RAW
2
64.7 cells through
inhibition
of NF-κB pathway
作者:
Zhi-Ke Liu
a
;
b
;
liuzhikebee@163.com
;
Chun-Fai Ng
a
;
b
;
ncf0000@hotmail.com
;
Hoi-Ting Shiu
a
;
b
;
hoitingshiu@gmail.com
;
Hing-Lok Wong
a
;
b
;
vhlwong@yahoo.com
;
Chun-Wai Wong
a
;
b
;
cwwong_eric@cuhk.edu.hk
;
Kai-Kai Li
a
;
b
;
likaicuhk@gmail.com
;
Jin-Fang Zhang
d
;
zhangjf06@cuhk.edu.hk
;
Ping-Kuen Lam
e
;
lampingkuen@yahoo.com.hk
;
Wai-Sang Poon
e
;
wpoon@surgery.cuhk.edu.hk
;
Clara Bik-San Lau
a
;
b
;
c
;
claralau@cuhk.edu.hk
;
Ping-Chung Leung
a
;
b
;
c
;
pingcleung@cuhk.edu.hk
;
Chun-Hay Ko
a
;
b
;
c
;
gohey@yahoo.com
;
gohey@cuhk.edu.hk
关键词:
CR
;
Chuanxiong Rhizoma
;
GR
;
Gastrodiae Rhizoma
;
DCXF
;
Da Chuanxiong Formula
;
LPS
;
Lipopolysaccharide
;
NO
;
Nitric oxide
;
COX
-
2
;
Cyclooxygenase-
2
;
iNOS
;
inducible nitric oxide synthase
;
PGE
2
;
prostaglandin E
2
刊名:Journal of Ethnopharmacology
出版年:
2
017
4.
Anti-inflammatory, analgesic and
COX
-
2
inhibitory activity of novel thiadiazoles in irradiated rats
作者:
Fatma A. Ragab
a
;
Helmi I. Heiba
b
;
Marwa G. El-Gazzar
b
;
marwa.galal@eaea.org.eg
;
Sahar M. Abou-Seri
a
;
Walaa A. El-Sabbagh
b
;
Reham M. El-Hazek
b
关键词:
Thiadiazoles
;
COX
-
2
inhibitors
;
Anti-inflammatory
;
Analgesic
;
Toxicological studies
;
Irradiated rats
;
Docking
刊名:Journal of Photochemistry and Photobiology B: Biology
出版年:
2
017
5.
Saponin fraction isolated from Conyza blinii H.Lév. demonstrates strong anti-cancer activity that is due to its NF-κB
inhibition
作者:
Long Ma
a
;
b
;
woshimalong1983@163.com
;
malong@tust.edu.cn
;
Haiyan Liu
a
;
Ping Qin
a
;
Chenxi Hu
a
;
Shuli Man
a
;
Yuyin Li
a
;
Zhen Liu
a
;
Zhenxing Liu
a
;
Aipo Diao
a
;
b
;
diaoaipo@tust.edu.cn
关键词:
Saponin
;
Conyza blinii H.Lé
;
v.
;
Traditional Chinese medicine (TCM)
;
Anti-Cancer activity
;
Apoptosis
;
NF-κB
inhibition
刊名:Biochemical and Biophysical Research Communications
出版年:
2
017
6.
In silico receptor-based drug design of X,Y-benzenesulfonamide derivatives as selective
COX
-
2
inhibitors
作者:
David J. Pé
;
rez
a
;
Orlando Sarabia
a
;
Manuel Villanueva-Garcí
;
a
b
;
Kayim Pineda-Urbina
a
;
Á
;
ngel Ramos-Organillo
a
;
Jorge Gonzalez-Gonzalez
a
;
Zeferino Gó
;
mez-Sandoval
a
;
zgomez@ucol.com
;
Rodrigo Said Razo-Herná
;
ndez
a
;
c
;
rrazo@ucol.mx
关键词:
QSAR
;
Docking
;
Cyclooxygenase
;
Benzenesulfonamides
;
Drug design
;
Artificial neural networks
刊名:Comptes Rendus Chimie
出版年:
2
017
7.
First isolation of glutinol and a bioactive fraction with good anti-inflammatory activity from n-hexane fraction of Peltophorum africanum leaf
作者:
Salmon A. Adebayo
1
;
2
;
Leshweni J. Shai
2
;
shaiLJ@tut.ac.za
;
Jacobus N. Eloff
1
关键词:
Peltophorum africanum
;
COX
-1/COX-
2
;
iNOS
;
Nitric oxide
;
Anti-inflammatory
刊名:Asian Pacific Journal of Tropical Medicine
出版年:
2
017
8.
Novel
2
,4-dichlorophenoxy acetic acid substituted thiazolidin-4-ones as anti-inflammatory agents: Design, synthesis and biological screening
作者:
Yakub Ali
a
;
Mohammad Sarwar Alam
a
;
msalam@jamiahamdard.ac.in
;
msalam5555@gmail.com
;
Hinna Hamid
a
;
hhamid@jamiahamdard.ac.in
;
Asif Husain
b
;
Abhijeet Dhulap
c
;
Sameena Bano
a
;
Chetna Kharbanda
a
关键词:
2
-Imino-4-thiazolidinone
;
Anti-inflammatory
;
COX
-
2
;
TNF-α
;
Anti-nociceptive
;
Ulcerogenic
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:
2
017
9.
The anti-inflammatory effects of N-methyl-(
2
S,4R)-trans-4-hydroxy-l-proline from Syderoxylon obtusifolium are related to its
inhibition
of TNF-alpha and inflammatory enzymes
作者:
Pedro Everson Alexandre de Aquino
a
;
Talita Rocha Magalhã
;
es
a
;
Lucas Antô
;
nio Duarte Nicolau
a
;
Luzia Kalyne A. Moreira Leal
a
;
Nayara Coriolano de Aquino
b
;
Sabrina Matias dos Santos
b
;
Kelly Rose Tavares Neves
a
;
Edilberto Rocha Silveira
b
;
Glauce Socorro de Barros Viana
a
;
c
;
gbviana@live.com
关键词:
Sideroxylon obtusifolium
;
Inflammation
;
Cytokines
;
Oxidative stress
刊名:Phytomedicine
出版年:
2
017
10.
Polyfluorinated salicylic acid derivatives as analogs of known drugs: Synthesis, molecular docking and biological evaluation
作者:
E.V. Shchegol'kov
a
;
schegolkov@ios.uran.ru
;
I.V. Shchur
a
;
Ya.V. Burgart
a
;
V.I. Saloutin
a
;
A.N. Trefilova
b
;
G.A. Ljushina
b
;
S.Yu. Solodnikov
b
;
L.N. Markova
b
;
V.V. Maslova
b
;
O.P. Krasnykh
b
;
S.S. Borisevich
c
;
S.L. Khursan
c
关键词:
Polyfluoronated salicylates
;
Nucleophilic substitution
;
ortho-Methoxylation
;
Molecular docking
;
Anti-inflammatory and analgesic activities
;
COX
-1
inhibition
;
Toxicity
;
Permeability
刊名:Bioorganic & Medicinal Chemistry
出版年:
2
017
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