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在“Elsevier电子期刊”中，命中：658条，耗时：小于0.01 秒

1.Transformation of arylcarboxamides into 1,3-dioxo-1,3-dihydroisobenzofuran-4-carboxamides

作者：Benjamin Prek ; Jure Bezen&scaron ; ek ; Marta Počkaj ; Branko Stanovnik ; ^{branko.stanovnik@fkkt.uni-lj.si}

关键词：Enaminones ; Carboxamides ; Aroylacetamidines ; (E)-N-(1-(dimethylamino)ethylidene)-carboxamides ; 1 ; 3-Dioxo-1 ; 3-dihydroisobenzofuran-4-carboxamides

刊名：Tetrahedron

出版年：2017

2.Synthesis, biological evaluation, docking study and ulcerogenicity profiling of some novel quinoline-2-carboxamides as dual COXs/LOX inhibitors endowed with anti-inflammatory activity

作者：Mostafa H. Abdelrahman^a ; Bahaa G.M. Youssif^b ; ^c ; ^{bgyoussif@ju.edu.sa} ; Mohamed A. abdelgawad^c ; ^d ; Ahmed H. Abdelazeem^e ; ^f ; Hussein M. Ibrahim^g ; ^h ; Abd El Ghany A. Moustafa^h ; ⁱ ; Laurent Treamblu^j ; Syed Nasir Abbas Bukhari^c ; ^{snab_hussaini@yahoo.com}

关键词：Quinoline-2-carboxamides ; COXs ; LOX ; Docking ; Anti-inflammatory

刊名：European Journal of Medicinal Chemistry

出版年：2017

3.Crystal structures, binding interactions, and ADME evaluation of brain penetrant N-substituted indazole-5-carboxamides as subnanomolar, selective monoamine oxidase B and dual MAO-A/B inhibitors

作者：Nikolay T. Tzvetkov^a ; ^{ntzvetkov@ntzlab.com} ; Hans-Georg Stammler^b ; Beate Neumann^b ; Silvia Hristova^c ; Liudmil Antonov^c ; Marcus Gastreich^d

关键词：ADME ; MAO inhibitors ; Molecular modeling ; Indazole-5-carboxamides ; Parkinson's disease ; X-ray

刊名：European Journal of Medicinal Chemistry

出版年：2017

4.Structure-activity relationship study and discovery of indazole 3-carboxamides as calcium-release activated calcium channel blockers

作者：Sha Bai^a ; Masazumi Nagai^a ; Steffi K. Koerner^a ; Aristidis Veves^b ; Lijun Sun^a ; ^{lsun1@bidmc.harvard.edu}

关键词：Mast cell ; Inflammation ; Calcium channel blockers ; Indazole-3-carboxamides

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

5.Sonochemistry in organocatalytic enamine-azide [3+2] cycloadditions: A rapid alternative for the synthesis of 1,2,3-triazoyl carboxamides

关键词：Sonochemistry ; Cycloadditions ; Organocatalysis ; 12 ; 3-Triazoles ; Carboxamides

刊名：Ultrasonics Sonochemistry

出版年：2017

6.Structure-based optimization of 1H-imidazole-2-carboxamides as Axl kinase inhibitors utilizing a Mer mutant surrogate

作者：Walter Keung^a ; ^{walter.keung@takeda.com} ; Amogh Boloor^a ; Jason Brown^a ; Andre Kiryanov^a ; Anthony Gangloff^a ; J. David Lawson^b ; Robert Skene^b ; Isaac Hoffman^b ; Josephine Atienza^c ; Jason Kahana^c ; Ron De Jong^c ; Pamela Farrell^c ; Deepika Balakrishna^c ; Petro Halkowycz^c

关键词：Axl ; Mer ; Structure design ; Oncology design ; Modeling ; Crystallography ; SBDD

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

7.New pyridazinone-4-carboxamides as new cannabinoid receptor type-2 inverse agonists: Synthesis, pharmacological data and molecular docking

作者：Giulio Ragusa^a ; Marí ; a Gó ; mez-Cañ ; as^b ; ^c ; ^d ; Paula Morales^e ; Carmen Rodrí ; guez-Cueto^b ; ^c ; ^d ; Marí ; a R. Pazos^b ; ^c ; ^d ; Battistina Asproni^a ; Elena Cichero^f ; Paola Fossa^f ; Gerard A. Pinna^a ; Nadine Jagerovic^e ; Javier Ferná ; ndez-Ruiz^b ; ^c ; ^d ; Gabriele Murineddu^a ; ^{muri@uniss.it}

关键词：Scaffold hopping ; Synthesis ; Cannabinoid receptors ; CB2 antagonism ; ADME model ; Docking studies

刊名：European Journal of Medicinal Chemistry

出版年：2017

8.Linker-switch approach towards new ATP binding site inhibitors of DNA gyrase B

作者：Marko Jukič^a ; Janez Ila&scaron ; ^a ; Matjaž Brvar^b ; Danijel Kikelj^a ; Jožko Cesar^a ; Marko Anderluh^a ; ^{marko.anderluh@ffa.uni-lj.si}

关键词：Antibiotics ; Antibacterials ; Inhibitor ; DNA gyrase B ; ATP binding site ; Pyrrole-2-carboxamides ; Structure-based drug design ; Ligand-based drug design

刊名：European Journal of Medicinal Chemistry

出版年：2017

9.Design, synthesis and docking studies of novel 1,2-dihydro-4-hydroxy-2-oxoquinoline-3-carboxamide derivatives as a potential anti-proliferative agents

作者：Saleha Banu^a ; Rajitha Bollu^a ; Rajashaker Bantu^a ; Lingaiah Nagarapu^a ; ; Sowjanya Polepalli^b ; Nishant Jain^b ; Radhika Vangala^c ; Vijjulatha Manga^c

关键词：Roquinimex ; 1 ; 2-dihydro-4-hydroxy-2-oxoquinoline-3-carboxamides ; Piperazines ; Anti-proliferative ; Multiple sclerosis ; Cell lines and molecular modeling

刊名：European Journal of Medicinal Chemistry

出版年：2017

10.Synthesis and structure-activity studies of side chain analogues of the anti-tubercular agent, Q203

作者：Sunhee Kang^a ; ^d ; Young Mi Kim^a ; Ryang Yeo Kim^b ; Min Jung Seo^a ; Zaesung No^a ; Kiyean Nam^c ; Sanghee Kim^d ; ^{pennkim@snu.ac.kr} ; Jaeseung Kim^a ; ^{silanediol@gmail.com}

关键词：Tuberculosis ; Imidazo[1 ; 2-a]pyridine-3-carboxamide (IPA) ; Pharmacokinetics ; Structure-activity relationship (SAR) ; Q203

刊名：European Journal of Medicinal Chemistry

出版年：2017

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