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CNKI学位论文(45)
知网期刊论文(2)
在“
Elsevier电子期刊
”中,
命中:
54
条,耗时:小于0.01 秒
在所有数据库中总计命中:
47
条
1.
7-Substituted umbelliferone derivatives as androgen receptor antagonists for the potential treatment of prostate and breast cancer
作者:
Sahar Kandil
;
Kandils1@cardiff.ac.uk" class="auth_mail" title="E-mail the corresponding author
;
Andrew D. Westwell
;
Christopher
McGuigan
关键词:
Androgen receptor (AR)
;
Prostate cancer (PC)
;
Breast cancer (BC)
;
Steroids
;
Triple negative breast cancer (TNBC)
;
Coumarin
;
Umbelliferone
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
2.
Design and synthesis of novel bicalutamide and enzalutamide derivatives as antiproliferative agents for the treatment of prostate cancer
作者:
Marcella Bassetto
1
;
Salvatore Ferla
;
1
;
Ferlas1@cardiff.ac.uk" class="auth_mail" title="E-mail the corresponding author
;
Fabrizio Pertusati
1
;
Sahar Kandil
;
Andrew D. Westwell
;
Andrea Brancale
;
Christopher
McGuigan
关键词:
Bicalutamide
;
Enzalutamide
;
Prostate cancer
;
Perfluoroalkyl
;
Androgen receptor
;
Antiproliferative activity
刊名:European Journal of Medicinal Chemistry
出版年:2016
3.
Rational design and synthesis of novel anti-prostate cancer agents bearing a 3,5-bis-trifluoromethylphenyl moiety
作者:
Salvatore Ferla
&dagger
;
;
Marcella Bassetto
;
&dagger
;
;
bassettom@cardiff.ac.uk" class="auth_mail" title="E-mail the corresponding author
;
Fabrizio Pertusati
&dagger
;
;
Sahar Kandil
;
Andrew D. Westwell
;
Andrea Brancale
;
Christopher
McGuigan
关键词:
Homology modelling
;
Rational drug design
;
Prostate cancer
;
Androgen-receptor
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
4.
A curriculum on care for people with disabilities: Effects on medical student self-reported attitudes and comfort level
作者:
Andrew B. Symons
;
Christopher
P. Morley
;
Denise
McGuigan
;
Elie A. Akl
关键词:
Disability
;
Medical education
;
Medical students
;
Evaluation
;
Curriculum
刊名:Disability and Health Journal
出版年:January, 2014
5.
Design, synthesis and biological evaluation of phosphorodiamidate prodrugs of antiviral and anticancer nucleosides
作者:
Christopher
McGuigan
;
Claire Bourdin
;
Marco Derudas
;
Nad猫ge Hamon
;
Karen Hinsinger
;
Sahar K
;
il
;
Karolina Madela
;
Silvia Meneghesso
;
Fabrizio Pertusati
;
Michaela Serpi
;
Magdalena Slusarczyk
;
Stanley Chamberlain
;
Alex
;
er Kolykhalov
;
John Vernachio
;
Christophe Vanpouille
;
Andrea Introini
;
Leonid Margolis
;
Jan Balzarini
关键词:
Nucleoside analogs
;
Antiviral
;
Anticancer
;
Phosphorodiamidates
;
Prodrugs
刊名:European Journal of Medicinal Chemistry
出版年:December, 2013
6.
Design, synthesis,?and biological evaluation of C1-phosphonamidate analogues of 2-deoxy-d-ribose-1-phosphate
作者:
Maurizio Quintiliani
;
Jan Balzarini
;
Christopher
McGuigan
关键词:
Deoxyribose
;
Phosphorylation
;
Phosphonates
;
Phosphonamidates
刊名:Tetrahedron
出版年:2013
7.
Serendipity and VZV drug discovery
作者:
Marco Derudas
;
derudasm@cardiff.ac.uk
;
Christopher
McGuigan
刊名:Drug Discovery Today: Technologies
出版年:2012
8.
DMPK and Metabolism Studies of Nucleoside Phosphoramidates Including INX-08189, A Novel Double Pro-drug and Clinical Candidate for Hepatitis C Virus Therapy
作者:
Jeff T. Hutchins
1
;
;
Christopher
McGuigan
2
;
Stanley D. Chamberlain
1
;
Karolina W. Madela
2
;
Mohamed Aljarah
2
;
John Vernachio
1
;
Joseph M. Patti
1
;
Geoffrey Henson
1
刊名:Antiviral Research
出版年:2011
9.
Application of the phosphoramidate ProTide approach to the antiviral drug ribavirin
作者:
Marco Derudas
;
Andrea Brancale
;
Lieve Naesens
;
Johan Neyts
;
Jan Balzarini
;
Christopher
McGuigan
关键词:
Ribavirin
;
ProTide
;
Carboxypeptidase Y
;
Human hint enzyme
刊名:Bioorganic and Medicinal Chemistry
出版年:2010
10.
Phosphoramidates of 2′-β-
d-arabinouridine (AraU) as phosphate prodrugs; design, synthesis, in vitro activity and metabolism
作者:
Youcef Mehellou
;
Rocco Valente
;
Huw Mottram
;
Elisabeth Walsby
;
Kenneth I. Mills
;
Jan Balzarini
;
Christopher
McGuigan
关键词:
Antiviral
;
Nucleosides
;
Nucleotides
;
Prodrugs
;
Protides
;
Anticancer
刊名:Bioorganic and Medicinal Chemistry
出版年:2010
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