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CNKI学位论文(2)
在“
Elsevier电子期刊
”中,
命中:
19
条,耗时:0.0160205 秒
在所有数据库中总计命中:
2
条
1.
New melatonin (MT
1
/MT
2
) ligands: Design and synthesis of (8,9-dihydro-7H-furo[3,2-f]chromen-1-yl) derivatives
作者:
Elodie L
;
agaray
;
Mohamed Ettaoussi
;
V茅ronique Leclerc
;
Balla Traor茅
;
Val茅rie Perez
;
Olivier Nosjean
;
Jean A. Boutin
;
Daniel
-
Henri
Caignard
;
Philippe Delagrange
;
Pascal Berthelot
;
Sa茂d Yous
关键词:
[35S]-GTP纬S
;
guanosine-5&prime
;
[纬-35S]-triphosphate
;
CHO
;
Chinese Hamster Ovary
;
HEK
;
Human Embryonic Kidney
;
MLT
;
melatonin
刊名:Bioorganic and Medicinal Chemistry
出版年:1 February, 2014
2.
Design and synthesis of naphthalenic derivatives as new ligands at the melatonin binding site MT
3
作者:
Vé
;
ronique Leclerc
;
Mohamed Ettaoussi
;
Marouan Rami
;
Amaury Farce
;
Jean Albert Boutin
;
Philippe Delagrange
;
Daniel
-
Henri
Caignard
;
Pierre Renard
;
Pascal Berthelot
;
Saï
;
d Yous
关键词:
Melatonin
;
MCA-NAT
;
MT
3
binding site
;
Naphthalenic ligands
;
Binding
;
Quinone reductase 2
刊名:European Journal of Medicinal Chemistry
出版年:2011
3.
Preparation and pharmacological evaluation of a novel series of 2-(phenylthio)benzo[b]thiophenes as selective MT
2
receptor ligands
作者:
Christophe Mé
;
sangeau
;
Mikaë
;
l Fraise
;
Philippe Delagrange
;
Daniel
Henri
Caignard
;
Jean Albert Boutin
;
Pascal Berthelot
;
Saï
;
d Yous
关键词:
Melatonin
;
MT2
;
Antagonist
;
Selective ligands
刊名:European Journal of Medicinal Chemistry
出版年:2011
4.
4,4-Dimethyl-1,2,3,4-tetrahydroquinoline-based PPARα/γ agonists. Part. II: Synthesis and pharmacological evaluation of oxime and acidic head group structural variations
作者:
Cé
;
cile Parmenon
;
Jé
;
rô
;
me Guillard
;
Daniel
-
Henri
Caignard
;
Nathalie Hennuyer
;
Bart Staels
;
Valé
;
rie Audinot-Bouchez
;
Jean-Albert Boutin
;
Catherine Dacquet
;
Alain Ktorza
;
Marie-Claude
关键词:
PPARs
;
Terahydroquinoline
;
Oxime
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
5.
S26948, a new specific peroxisome proliferator activated receptor gamma modulator improved in vivo
作者:
Kyung-Ah Kim Sohn
;
Cé
;
line Cruciani-Guglielmacci
;
Nadim Kassis
;
Laurence Clé
;
ment
;
Fetta Ouali
;
Michè
;
le Caü
;
zac
;
Nicolas Lebè
;
gue
;
Pascal Berthelot
;
Daniel
-
Henri
Caignard
;
Jean-Pa
关键词:
SPPARMγ
;
agonist
;
Liver
;
Glucose hepatic production
;
Fatty acid
;
Glucose homeostasis
刊名:European Journal of Pharmacology
出版年:2009
6.
Novel 5-azaindolocarbazoles as cytotoxic agents and Chk1 inhibitors
作者:
Myriam Lefoix
;
Gé
;
rard Coudert
;
Sylvain Routier
;
Bruno Pfeiffer
;
Daniel
-
Henri
Caignard
;
John Hickman
;
Alain Pierré
;
Roy M. Golsteyn
;
Sté
;
phane Lé
;
once
;
Cé
;
line Bossard
;
Jean-Yves
关键词:
5-Azaindole
;
5-Azaindolocarbazole
;
Chk1 inhibitors
;
Cytoxicity
刊名:Bioorganic and Medicinal Chemistry
出版年:2008
7.
Synthesis and pharmacological evaluation of a second generation of pyridothiadiazine 1,1-dioxides acting as AMPA potentiators
作者:
Pierre Francotte
;
Pascal de Tullio
;
Tchao Podona
;
Ousmane Diouf
;
Pierre Fraikin
;
Pierre Lestage
;
Laurence Danober
;
Jean-Yves Thomas
;
Daniel
-
Henri
Caignard
;
Bernard Pirotte
关键词:
AMPA potentiator
;
Allosteric modulation
;
Cognitive enhancer
刊名:Bioorganic and Medicinal Chemistry
出版年:2008
8.
Synthesis of potential Rho-kinase inhibitors based on the chemistry of an original heterocycle: 4,4-Dimethyl-3,4-dihydro-1H-quinolin-2-one
作者:
Marie-Anne Letellier
;
Jé
;
rô
;
me Guillard
;
Daniel
-
Henri
Caignard
;
Gilles Ferry
;
Jean A. Boutin
;
Marie-Claude Viaud-Massuard
关键词:
Rho-kinase inhibitors
;
Hypertension
;
Heterocyclic chemistry
刊名:European Journal of Medicinal Chemistry
出版年:2008
9.
4,4-Dimethyl-1,2,3,4-tetrahydroquinoline-based PPARα/γ agonists. Part I: Synthesis and pharmacological evaluation
作者:
Cé
;
cile Parmenon
;
Jé
;
rô
;
me Guillard
;
Daniel
-
Henri
Caignard
;
Nathalie Hennuyer
;
Bart Staels
;
Valé
;
rie Audinot-Bouchez
;
Jean-Albert Boutin
;
Catherine Dacquet
;
Alain Ktorza
;
Marie-Claude
关键词:4 ;
4-Dimethyl-1
23 ;
4-tetrahydroquinoline
;
PPAR
;
//www.sciencedirect.com/scidirimg/entities/204e.gif"" alt=""greek small letter alpha"" title=""greek small letter alpha"" border=""0"">/γ
;
agonists
;
Diabetes type-2
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2008
10.
Synthesis of 3-phenylnaphthalenic derivatives as new selective MT
2
melatoninergic ligands
作者:
Sophie Poissonnier-Durieux
;
Mohamed Ettaoussi
;
Basile Pé
;
rè
s ;
Jean A. Boutin
;
Valé
;
rie Audinot
;
Caroline Bennejean
;
Philippe Delagrange
;
Daniel
Henri
Caignard
;
Pierre Renard
;
Pascal Berth
关键词:
Melatonin
;
MT
2
receptors
;
3-Phenylnaphthalene
;
Selective antagonists
刊名:Bioorganic and Medicinal Chemistry
出版年:2008
1
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