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在“Elsevier电子期刊”中，命中：44条，耗时：0.0159899 秒

1.Solid-phase synthesis of 6,7-cycloalkane-fused 1,4-diazepane-2,5-diones via a cyclization/release strategy

作者：Jurgen Caroen^a ; An Clemmen^a ; Judit Ká ; má ; n^a ; ^b ; Fré ; derique Backaert^a ; Jan L. Goeman^a ; Ferenc Fü ; lö ; p^b ; Johan Van der Eycken^a ; ^{Johan.VanderEycken@UGent.be" class="auth_mail" title="E-mail the corresponding author}

关键词：Solid-phase synthesis ; 1 ; 4-Diazepane-2 ; 5-diones ; Homodiketopiperazines ; Cyclization/release strategy ; Conformational analysis of cyclic dipeptides

刊名：Tetrahedron

出版年：2016

2.Synthesis, selected coordination chemistry and extraction behavior of a (phosphinoylmethyl)pyridyl N-oxide-functionalized ligand based upon a 1,4-diazepane platform

作者：Sabrina Ouizem^a ; ¹ ; Daniel Rosario Amorin^a ; ² ; Diane A. Dickie^a ; Roger E. Cramer^b ; Charles F. Campana^c ; Benjamin P. Hay^d ; Julien Podair^e ; Laetitia H. Delmau^e ; Robert T. Paine^a ; ^{rtpaine@unm.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：Diazepane ; Pyridyl ; Phosphine oxide ; Coordination chemistry ; X-ray crystal structures

刊名：Polyhedron

出版年：2015

3.Discovery of diazepane amide DORAs and 2-SORAs enabled by exploration of isosteric quinazoline replacements

作者：Anthony J. Roecker^a ; ^{anthony_roecker@merck.com" class="auth_mail" title="E-mail the corresponding author} ; Swati P. Mercer^a ; Jeffrey M. Bergman^a ; Kevin F. Gilbert^a ; Scott D. Kuduk^a ; C. Meacham Harrell^b ; Susan L. Garson^b ; Steven V. Fox^b ; Anthony L. Gotter^b ; Pamela L. Tannenbaum^b ; Thomayant Prueksaritanont^c ; Tamara D. Cabalu^c ; Donghui Cui^c ; Wei Lemaire^d ; Christopher J. Winrow^b ; John J. Renger^b ; Paul J. Coleman^a

关键词：Orexin ; Antagonists ; Sleep ; Isostere ; Quinazoline

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2015

4.New ⁶⁸Ga-PhenA bisphosphonates as potential bone imaging agents

作者：Zehui Wu^a ; ¹ ; Zhihao Zha^a ; ¹ ; Seok Rye Choi^a ; Karl Plö ; ssl^a ; Lin Zhu^a ; Hank F. Kung^a ; ^b ; ^{kunghf@gmail.com" class="auth_mail" title="E-mail the corresponding author}

关键词：PET ; positron emission tomography ; SPECT ; single photon emission computed tomography ; MRI ; magnetic resonance imaging ; NET ; neuroendocrine tumor ; DTPA ; diethylenetriaminepentaacetic acid [1] ; DOTA ; 147 ; 10-tetraazacyclododecane-147 ; 10-tetraacetic acid [2] ; NOTA ; 14 ; 7-triazacyclononane-N ; N&prime ; N&Prime ; -triacetic acid [3 ; 4] ; NODAGA ; 1-(1 ; 3-carboxypropyl)-4 ; 7-carboxymethyl-14 ; 7-triazacyclononane [1 ; 5&ndash ; 9] ; TRAP ; 14 ; 7-triazacyclononane-N ; N&prime ; N&Prime ; -tris(methylenephosphonic) aci

刊名：Nuclear Medicine and Biology

出版年：2016

5.Exploration of the molecular architecture of the orthosteric binding site in the 伪4尾2 nicotinic acetylcholine receptor with analogs of 3-(dimethylamino)butyl dimethylcarbamate (DMABC) and 1-(pyridin-3-yl)-1,4-diazepane

作者：Tinna B. Bach^a ; Anders A. Jensen^a ; Jette G. Petersen^a ; Troels E. Sø ; rensen^a ; ^b ; Serena Della Volpe^a ; Jun Liu^b ; Antoni R. Blaazer^c ; Jacqueline E. van Muijlwijk-Koezen^c ; Thomas Balle^b ; ^{thomas.balle@sydney.edu.au" class="auth_mail" title="E-mail the corresponding author} ; Bente Frø ; lund^a ; ^{bfr@sund.ku.dk" class="auth_mail" title="E-mail the corresponding author}

关键词：nACh receptor agonists ; Structure&ndash ; activity studies ; Ls-AChBP ; Ac-AChBP ; Lobeline ; DMABC analogs

刊名：European Journal of Medicinal Chemistry

出版年：2015

6.Antibacterial oxazolidinone analogues having a N-hydroxyacetyl-substituted seven-membered [1,2,5]triazepane or [1,2,5]oxadiazepane C-ring unit

作者：Hideyuki Suzuki^a ; ^{hsuzuki@itsuu.or.jp} ; Iwao Utsunomiya^a ; Koichi Shudo^a ; Norio Fukuhara^b ; Tsutomu Iwaki^b ; Tatsuro Yasukata^c

关键词：Antibacterial ; Oxazolidinone ; [12 ; 5]Triazepane ; [12 ; 5]Oxadiazepane

刊名：European Journal of Medicinal Chemistry

出版年：2013

7.Synthesis and in聽vitro/in聽vivo antibacterial activity of oxazolidinones having thiocarbamate at C-5 on the A-ring and an amide- or urea-substituted [1,2,5]triazepane or [1,2,5]oxadiazepane as the C-ring

作者：Hideyuki Suzuki ; Iwao Utsunomiya ; Koichi Shudo ; Norio Fukuhara ; Tsutomu Iwaki ; Tatsuro Yasukata

关键词：Antibacterial ; Oxazolidinone ; Methicillin-resistant Staphylococcus aureus ; [12 ; 5]Triazepane ; [12 ; 5]Oxadiazepane

刊名：European Journal of Medicinal Chemistry

出版年：November, 2013

8.Discovery of novel series of 6-benzyl substituted 4-aminocarbonyl-1,4-diazepane-2,5-diones as human chymase inhibitors using structure-based drug design

作者：Taisaku Tanaka ; ^{tanaka.taisaku.fu@asubio.co.jp} ; Hajime Sugawara ; Hiroshi Maruoka ; Seiichi Imajo ; Tsuyoshi Muto ; ^{muto.tsuyoshi.ba@asubio.co.jp}

关键词：Chymase inbibitor ; Atopic dermatitis ; Amino acid derivatives ; Heteroaromatic derivatives

刊名：Bioorganic and Medicinal Chemistry

出版年：2013

9.Aryl 1,4-diazepane compounds as potent and selective CB2 agonists: Optimization of drug-like properties and target independent parameters

作者：René ; e Zindell^a ; ^{renee.zindell@boehringer-ingelheim.com"" rel=""nofollow} ; Edward R. Walker^d ; John Scott^d ; Patricia Amouzegh^d ; Lifen Wu^a ; Monika Ermann^d ; David Thomson^a ; Micheal B. Fisher^c ; Cody Lee Fullenwider^c ; Heather Grbic^c ; Paul Kaplita^c ; Brian Linehan^c ; Mita Patel^c ; Monica Patel^c ; Sabine Lö ; bbe^e ; Svenja Block^e ; Claudia Albrecht^e ; Mark J. Gemkow^e ; Daw-Tsun Shih^b ; Doris Riether^a

关键词：Cannabinoid receptor ; CB2 ; 1 ; 4-Diazepane ; Drug-like parameters ; Permeability

刊名：Bioorganic and Medicinal Chemistry Letters

出版年：2011

10.Discovery of dual orexin receptor antagonists with rat sleep efficacy enabled by expansion of the acetonitrile-assisted/diphosgene-mediated 2,4-dichloropyrimidine synthesis

作者：Anthony J. Roecker^a ; ^{anthony_roecker@merck.com" class="auth_mail} ; Swati P. Mercer^a ; C. Meacham Harrell^b ; Susan L. Garson^b ; Steven V. Fox^b ; Anthony L. Gotter^b ; Thomayant Prueksaritanont^c ; Tamara D. Cabalu^c ; Donghui Cui^c ; Wei Lemaire^d ; Christopher J. Winrow^b ; John J. Renger^b ; Paul J. Coleman^a

关键词：Orexin ; Antagonist ; Sleep ; Bioactivation ; Pyrimidine

刊名：Bioorganic and Medicinal Chemistry Letters

出版年：1 May, 2014

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