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馆藏书目(7)
CNKI学位论文(16)
知网期刊论文(5)
在“
Elsevier电子期刊
”中,
命中:
16
条,耗时:小于0.01 秒
在所有数据库中总计命中:
28
条
1.
Differential induction of dyskinesia and neuroinflammation by pulsatile versus continuous l-DOPA delivery in the 6-OHDA model of Parkinson's disease
作者:
Giovanna Mulas
;
PhD
a
;
Elena Espa
;
PhD
a
;
Sandro Fenu
;
PhD
a
;
Saturnino Spiga
;
PhD
b
;
Giovanni Cossu
;
MD
c
;
Elisabetta Pillai
a
;
Ezio Carboni
;
PhD
a
;
Gabriella Simbula
;
PhD
a
;
Dragana Jadžić
a
;
Fabrizio
Angius
;
PhD
a
;
Stefano Spolitu
;
PhD
a
;
Barbara Batetta
;
PhD
a
;
Daniela Lecca
;
PhD
a
;
Andrea Giuffrida
;
PhD
d
;
Anna R.
Carta
;
PhD
a
;
a
carta
@unica.it" class="auth_mail" title="E-mail the corresponding author
关键词:
Dyskinesia
;
Inflammation
;
Microglia
;
Parkinson
;
Cytokine
;
TNF-alpha
;
l-DOPA
刊名:Experimental Neurology
出版年:2016
2.
Combining the tail and the ring approaches for obtaining potent and isoform-selective carbonic anhydrase inhibitors: Solution and X-ray crystallographic studies
作者:
Murat Bozdag
;
Marta Ferraroni
;
Elisa Nuti
;
Daniela Vullo
;
Arm
;
o Rossello
;
Fabrizio
Carta
;
Andrea Scozzafava
;
Claudiu T. Supuran
关键词:
Carbonic anhydrase
;
Inhibitor
;
Sulfonamide
;
Tosylureido
;
X-ray crystallography
刊名:Bioorganic and Medicinal Chemistry
出版年:1 January, 2014
3.
Mono-/dihydroxybenzoic acid esters and phenol pyridinium derivatives as inhibitors of the mammalian carbonic anhydrase isoforms I, II, VII, IX, XII and XIV
作者:
Fabrizio
Carta
;
fabrizio
.
carta
@unifi.it
;
Daniela Vullo
;
Alfonso Maresca
;
Andrea Scozzafava
;
Claudiu T. Supuran
;
claudiu.supuran@unifi.it
关键词:
Carbonic anhydrase
;
Phenol
;
Hydroxy-/dihydroxybenzoic acid
;
Dopamine
;
Aminophenol
刊名:Bioorganic and Medicinal Chemistry
出版年:2013
4.
7-Substituted-sulfocoumarins are isoform-selective, potent carbonic anhydrase II inhibitors
作者:
Muhammet Tanc
;
Fabrizio
Carta
;
Murat Bozdag
;
Andrea Scozzafava
;
Claudiu T. Supuran
关键词:
Carbonic anhydrase
;
Sulfocoumarin
;
Coumarin
;
Sulfonamide
;
Isoform-selective inhibitor
刊名:Bioorganic and Medicinal Chemistry
出版年:2013
5.
Carbonic anhydrase inhibitors: Synthesis and inhibition of the cytosolic mammalian carbonic anhydrase isoforms I, II and VII with benzene sulfonamides incorporating 4,5,6,7-tetrachlorophthalimide moiety
作者:
Kalyan K. Sethi
;
Saurabh M. Verma
;
Muhammet Tan?
;
Fabrizio
Carta
;
Claudiu T. Supuran
关键词:
Human carbonic anhydrase inhibitors
;
Benzenesulfonamide
;
4
56 ;
7-Tetrachloro-1
;
3-dioxoisoindolin-2-yl benzenesulfonamide
;
Structure&ndash
;
activity relationship
刊名:Bioorganic and Medicinal Chemistry
出版年:2013
6.
Carbonic anhydrase inhibitors: Synthesis and inhibition of the human carbonic anhydrase isoforms I, II, VII, IX and XII with benzene sulfonamides incorporating 4,5,6,7-tetrabromophthalimide moiety
作者:
Kalyan K. Sethi
;
Daniella Vullo
;
Saurabh M. Verma
;
Muhammet Tan?
;
Fabrizio
Carta
;
Claudiu T. Supuran
关键词:
CA
;
carbonic anhydrase
;
hCA
;
human carbonic anhydrase
;
CAI
;
carbonic anhydrase inhibitor
;
SAR
;
structure&ndash
;
activity relationship
;
Zn
;
zinc
;
AZM
;
acetazolamide
;
MZA
;
methazolamide
;
EZA
;
ethoxzolamide
;
DCP
;
dibromophenamide
;
DZA
;
dorzolamide
;
BRZ
;
brinz
刊名:Bioorganic and Medicinal Chemistry
出版年:2013
7.
New chemotypes acting as isozyme-selective carbonic anhydrase inhibitors with low affinity for the offtarget cytosolic isoform II
作者:
Fabrizio
Carta
;
Daniela Vullo
;
Alfonso Maresca
;
Andrea Scozzafava
;
Claudiu T. Supuran
;
claudiu.supuran@unifi.it
关键词:
Carbonic anhydrase
;
Offtarget isoform
;
2-Hydroxyquinoline
;
Coumarin oxime
;
Coumaphos
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2012
8.
Novel coumarins and 2-thioxo-coumarins as inhibitors of the tumor-associated carbonic anhydrases IX and XII
作者:
Fabrizio
Carta
;
Alfonso Maresca
;
Andrea Scozzafava
;
Claudiu T. Supuran
;
claudiu.supuran@unifi.it
关键词:
Carbonic anhydrase
;
Coumarin
;
Transmembrane isoform
;
Tumor-associated enzyme
;
Selective inhibition
刊名:Bioorganic and Medicinal Chemistry
出版年:2012
9.
5- and 6-Membered (thio)lactones are prodrug type carbonic anhydrase inhibitors
作者:
Fabrizio
Carta
;
Alfonso Maresca
;
Andrea Scozzafava
;
Claudiu T. Supuran
;
claudiu.supuran@unifi.it
关键词:
Carbonic anhydrase
;
Lactone
;
Thiolactone
;
Coumarin
;
Prodrug
;
Esterase activity
;
Isoform-selective inhibitor
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2012
10.
Ureido-substituted sulfamates show potent carbonic anhydrase IX inhibitory and antiproliferative activities against breast cancer cell lines
作者:
Jean-Yves Winum
;
Fabrizio
Carta
;
Carol Ward
;
Peter Mullen
;
David Harrison
;
Simon P. Langdon
;
Aless
;
ro Cecchi
;
Andrea Scozzafava
;
Ian Kunkler
;
Claudiu T. Supuran
关键词:
Carbonic anhydrase
;
Inhibitor
;
Isoform IX and XII
;
Antitumor agent
;
Sulfamate
;
Breast cancer
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2012
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