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CNKI学位论文(1)
知网期刊论文(1)
在“
Elsevier电子期刊
”中,
命中:
9
条,耗时:0.018989 秒
在所有数据库中总计命中:
2
条
1.
Allosteric modulators of human A
2B
adenosine receptor
作者:
Maria Letizia Trincavelli
;
Chiara Giacomelli
;
Simona
Da
niele
;
Sabrina Taliani
;
Barbara Cosimelli
;
Sonia Laneri
;
El
da
Severi
;
Elisabetta Barresi
;
Isabella Pugliesi
;
Giovanni Greco
;
Ettore Novellino
;
Federico
Da
Settimo
;
Claudia Martini
关键词:
A
DA
;
adenosine deaminase
;
AR
;
adenosine receptor
;
cAMP
;
3&prime
;
5&prime
;
-cyclic adenosine monophosphate
;
BAY 60-6583
;
2-[6-amino-3
;
5-dicyano-4-[4-(cyclopropylmethoxy)phenyl]pyridin-2-ylsulfanyl]acetamide
;
CHO
;
Chinese hamster ovary
;
DMAP
;
4-dimethylaminopyridine
;
DMEM
;
Dulbecco's Modified Eagle Medium
;
GPCR
;
G protein-coupled receptor
;
[35S]GTP纬S
;
[35S]guanosine 5&prime
;
-O-[gamma-thio]triphosphate
;
[3H]MRS 1754
;
[3H]N-(4-cyanophenyl)-2-[4-(2
36 ;
7-tetrahydro-2
;
6-dioxo-1
;
3-dipropyl-1H-purin-8-y
刊名:Biochimica et Biophysica Acta (BBA)/General Subjects
出版年:March, 2014
2.
A novel 2,3-diphenyl-4H-pyrido[1,2-a]pyrimidin-4-one derivative inhibits endothelial cell dysfunction and smooth muscle cell proliferation/activation
作者:
Serena Del Turco
;
Stefania Sartini
;
Cass
;
ra Sentieri
;
Chiara Saponaro
;
Teresa Navarra
;
Bianca
Da
rio
;
Federico
Da
Settimo
;
Concettina La Motta
;
Giuseppina Basta
关键词:2 ;
3-Diphenyl-4H-pyrido[1
;
2-a]pyrimidin-4-ones
;
2-(3
;
4-Dimethoxyphenyl)-3-phenyl-4H-pyrido[1
;
2-a]pyrimidin-4-one
;
Human aortic smooth muscle cells
;
Human umbilical vein endothelial cells
;
Cell proliferation
;
Cell dysfunction
刊名:European Journal of Medicinal Chemistry
出版年:24 January, 2014
3.
Modulation of A
2B
adenosine receptor by 1-Benzyl-3-ketoindole derivatives
作者:
Sabrina Taliani
;
Maria Letizia Trincavelli
;
Barbara Cosimelli
;
Sonia Laneri
;
El
da
Severi
;
Elisabetta Barresi
;
Isabella Pugliesi
;
Simona
Da
niele
;
Chiara Giacomelli
;
Giovanni Greco
;
Ettore Novellino
;
Claudia Martini
;
Federico
Da
Settimo
关键词:
1-Benzyl-3-ketoindole derivatives
;
A2B adenosine receptor
;
Positive modulators
;
Negative modulators
;
GPCR modulators
;
Ligand&n
da
sh
;
receptor interaction
刊名:European Journal of Medicinal Chemistry
出版年:November, 2013
4.
Synthesis and biological evaluation in U87MG glioma cells of (ethynylthiophene)sulfonamido-based hydroxamates as matrix metalloproteinase inhibitors
作者:
Elisa Nuti
;
Francesca Casalini
;
Salvatore Santamaria
;
Pamela Gabelloni
;
Sara Bendinelli
;
Eleonora
Da
Pozzo
;
Barbara Costa
;
Luciana Marinelli
;
Valeria La Pietra
;
Ettore Novellino
;
M. Margari
da
Bernardo
;
Rafael Fridman
;
Federico
Da
Settimo
;
Claudia Martini
;
Arm
;
o Rossello
关键词:
Matrix metalloproteinase inhibitors
;
Hydroxamic acids
;
Anti-glioma agents
;
MMP-2
;
MMP-9
;
MMP-25
刊名:European Journal of Medicinal Chemistry
出版年:2011
5.
Identification of 5-arylidene-4-thiazolidinone derivatives endowed with dual activity as aldose reductase inhibitors and antioxi
da
nt agents for the treatment of diabetic complications
作者:
Rosaria Ottanà
;
Rosanna Maccari
;
Marco Giglio
;
Antonella Del Corso
;
Mario Cappiello
;
Umberto Mura
;
S
;
ro Cosconati
;
Luciana Marinelli
;
Ettore Novellino
;
Stefania Sartini
;
Concettina La Motta
;
Federico
Da
Settimo
关键词:
Diabetes mellitus
;
Aldose reductase
;
Antioxi
da
nt agent
;
5-arylidene-4-thiazolidinones
;
Molecular docking
刊名:European Journal of Medicinal Chemistry
出版年:2011
6.
Spirohy
da
ntoin derivatives of thiopyrano[2,3-b]pyridin-4(4H)-one as potent in vitro and in vivo aldose reductase inhibitors
作者:
Da
Settimo
;
Federico
;
Primofiore
;
Giampaolo
;
La Motta
;
Concettina
;
Salerno
;
Silvia
;
Novellino
;
Ettore
;
et. al.
关键词:
Aldose reductase
;
Inhibitors
;
Spirohy
da
ntoin derivatives
;
Cataract
刊名:Bioorganic and Medicinal Chemistry
出版年:2005
7.
Effects of newly-developed benzodiazepine ligands on noise-induced mitochondrial
da
mage in the rat
作者:
Marco Gesi
;
Antonio Pellegrini
;
Paola Lenzi
;
Federico
Da
Settimo
;
Claudia Martini
;
Francesca Salvetti
;
Sabrina Taliani
;
Francesco Fornai
关键词:
Noise stress
;
Heart
;
Mitochondria
;
Benzodiazepine ligands
;
Transmission electron microscopy
;
Rat
;
N-arylalkylindol-3-ylglyoxylylamide derivatives
刊名:Annals of Anatomy - Anatomischer Anzeiger
出版年:2000
8.
Synthesis, DNA binding and in vitro antiproliferative activity of purinoquinazoline, pyridopyrimidopurine and pyridopyrimidobenzimi
da
zole derivatives as potential antitumor agents
作者:
Da
Settimo
;
Antonio
;
Da
Settimo
;
Federico
;
Marini
;
Anna Maria
;
Primofiore
;
Giampaolo
;
Salerno
;
Silvia
;
et. al.
关键词:
purinoquinazolines
;
pyridopyrimidopurines
;
pyridopyrimidobenzimi
da
zoles
;
antiproliferative properties
;
DNA binding agents
刊名:European Journal of Medicinal Chemistry
出版年:1998
9.
Indole amide derivatives: synthesis, structure-activity relationships and molecular modelling studies of a new series of histamine H
1
-receptor antagonists
作者:
Battaglia
;
Sandra
;
Boldrini
;
Enrico
;
Da
Settimo
;
Federico
;
Dondio
;
Giulio
;
La Motta
;
Concettina
;
et. al.
关键词:
indole derivatives
;
non-classic H
1
-antagonists
;
astemizole
;
structure-activity relationships
刊名:European Journal of Medicinal Chemistry
出版年:1999
1
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2000年及以前(2)
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