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内部出版物
在“
Elsevier电子期刊
”中,
命中:
11
条,耗时:小于0.01 秒
1.
Arylamino methylene bisphosphonate derivatives as bone seeking matrix metalloproteinase inhibitors
作者:
Marilena Tauro
;
Antonio Laghezza
;
Fulvio
Loiodice
;
Mariangela Agamennone
;
Cristina Campestre
;
Paolo Tortorella
关键词:
Matrix metalloproteinase inhibitors
;
Zinc binding group
;
Bone targeting
;
Bisphosphonates
刊名:Bioorganic and Medicinal Chemistry
出版年:2013
2.
An efficient synthesis of the optically active isomers of 2H-1,4-benzoxazine derivatives, novel KATP channel modulators
作者:
Luca Piemontese
;
Antonio Laghezza
;
Giuseppe Fracchiolla
;
Giuseppe Carbonara
;
Paolo Tortorella
;
Fulvio
Loiodice
刊名:Tetrahedron: Asymmetry
出版年:2013
3.
Kidney CLC-K Chloride Channels Show Differential Pharmacological Profiles Depending on the Heterologous Expression System
作者:
Antonella Liantonio
1
;
Paola Imbrici
1
;
Gianluca Gramegna
1
;
Antonella Gradogna
2
;
Giovanni Zifarelli
2
;
Antonio Laghezza
1
;
Giuseppe Fracchiolla
1
;
Giuseppe Carbonara
1
;
Fulvio
Loiodice
1
;
Michael Pusch
2
;
Diana Conte Camerino
1
刊名:Biophysical Journal
出版年:2013
4.
Design, synthesis and biological evaluation of 5-hydroxy, 5-substituted-pyrimidine-2,4,6-triones as potent inhibitors of gelatinases MMP-2 and MMP-9
作者:
Orazio Nicolotti
;
orazio.nicolotti@uniba.it
;
Marco Catto
;
Ilenia Giangreco
;
Maria Barletta
;
Francesco Leonetti
;
Angela Stefanachi
;
Leonardo Pisani
;
Saverio Cellamare
;
Paolo Tortorella
;
Fulvio
Loiodice
;
Angelo Carotti
;
angelo.carotti@uniba.it
关键词:
MMP
;
Gelatinases
;
ZBG
;
QSAR
;
Molecular docking
刊名:European Journal of Medicinal Chemistry
出版年:2012
5.
Synthesis, biological evaluation, and molecular modeling investigation of chiral 2-(4-chloro-phenoxy)-3-phenyl-propanoic acid derivatives with PPARα and PPARγ agonist activity
作者:
Giuseppe Fracchiolla
;
Antonio Lavecchia
;
Antonio Laghezza
;
Luca Piemontese
;
Raffaella Trisolini
;
Giuseppe Carbonara
;
Paolo Tortorella
;
Ettore Novellino
;
Fulvio
Loiodice
关键词:
Chirality
;
Peroxisome proliferator-activated receptor
;
Docking
;
Molecular dynamics
;
MM–
;
PBSA
刊名:Bioorganic and Medicinal Chemistry
出版年:2008
6.
Exploring the molecular basis of the enantioselective binding of penicillin G acylase towards a series of 2-aryloxyalkanoic acids: A docking and molecular dynamics study
作者:
Antonio Lavecchia
;
S
;
ro Cosconati
;
Ettore Novellino
;
Enrica Calleri
;
Caterina Temporini
;
Gabriella Massolini
;
Giuseppe Carbonara
;
Giuseppe Fracchiolla
;
Fulvio
Loiodice
关键词:
Docking
;
Enantioselectivity
;
Molecular dynamics
;
Molecular modeling
;
Penicillin G acylase
刊名:Journal of Molecular Graphics and Modelling
出版年:2007
7.
Enantiomeric separation of 2-aryloxyalkyl- and 2-arylalkyl-2-aryloxyacetic acids on a Penicillin G Acylase-based chiral stationary phase: Influence of the chemical structure on retention and enantiose
作者:
Caterina Temporini
;
Enrica Calleri
;
Giuseppe Fracchiolla
;
Giuseppe Carbonara
;
Fulvio
Loiodice
;
Antonio Lavecchia
;
Paolo Tortorella
;
Gloria Brusotti
;
Gabriella Massolini
关键词:
Chiral HPLC
;
Monolithic PGA column
;
Enantiomeric discrimination
;
Molecular modelling
刊名:Journal of Pharmaceutical and Biomedical Analysis
出版年:2007
8.
Carboxylic acids and skeletal muscle chloride channel conductance: effects on the biological activity induced by the introduction of methyl groups on the aromatic ring of chiral α-(4-chloro-pheno
作者:
Ferorelli
;
Savina
;
Loiodice
;
Fulvio
;
Tortorella
;
Vincenzo
;
Conte-Camerino
;
Diana
;
De Luca
;
Anna Maria
关键词:
Enantioselective synthesis
;
Absolute configuration
;
Chiroptical properties
;
Chloride channel conductance
;
Myotonic-inducing effects
刊名:Il Farmaco
出版年:2001
9.
Carboxylic acids and skeletal muscle chloride channel conductance: effects on the biological activity induced by the introduction of an aryloxyalkyl group α to the carboxylic function of 4-chloro
作者:
Carbonara
;
Giuseppe
;
Fracchiolla
;
Giuseppe
;
Loiodice
;
Fulvio
;
Tortorella
;
Paolo
;
Conte-Camerino
;
Diana
;
et. al.
关键词:
Aryloxyalkanoic acids
;
Chloride channel conductance
;
Rat skeletal muscle
;
Myotonic-inducing effects
刊名:Il Farmaco
出版年:2001
10.
Lipase-mediated kinetic resolution of rigid clofibrate analogues with lipid-modifying activity
作者:
Ferorelli
;
Savina
;
Franchini
;
Carlo
;
Loiodice
;
Fulvio
;
Perrone
;
Maria Grazia
;
Scilimati
;
Antonio
;
et. al.
刊名:Tetrahedron: Asymmetry
出版年:2001
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