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CNKI学位论文(1)
在“
Elsevier电子期刊
”中,
命中:
14
条,耗时:小于0.01 秒
在所有数据库中总计命中:
1
条
1.
Synthesis and biological evaluation of novel delta (未) opioid receptor ligands with diazatricyclodecane skeletons
作者:
Giovanni Loriga
;
Paolo Lazzari
;
Stefania Ruiu
;
Giorgio Marchese
;
Ilaria Manca
;
Gian Luca Casu
;
Christian Dess矛
;
G茅rard Aim猫 Pinna
;
Battistina Asproni
;
Gabriele
Murineddu
关键词:
未-Agonist SNC-80
;
未-Opioid receptor ligands
;
9
;
10-Diazatricyclo[4.2.1.12
;
5]decane
;
2
;
7-Diazatricyclo[4.4.0.03
;
8]decane
;
Binding assays
;
Antinociceptive activity
刊名:European Journal of Medicinal Chemistry
出版年:November, 2013
2.
NESS06SM reduces body weight with an improved profile relative to SR141716A
作者:
Andrea Mastinu
;
Marilena Pira
;
G¨¦rard Aim¨¨ Pinna
;
Carla Pisu
;
Maria Antonietta Casu
;
Roberta Reali
;
Stefania Marcello
;
Gabriele
Murineddu
;
Paolo Lazzari
关键词:
NESS06SM
;
SR141716A
;
Obesity
;
DIO mice
;
Mood disorders
刊名:Pharmacological Research
出版年:2013
3.
Synthesis of 3,6-diazabicyclo[3.1.1]heptanes as novel ligands for neuronal nicotinic acetylcholine receptors
作者:
Gabriele
Murineddu
;
Caterina Murruzzu
;
Maria M. Curzu
;
Giorgio Chelucci
;
Cecilia Gotti
;
Annalisa Gaimarri
;
Laura Legnani
;
Lucio Toma
;
Gerard A. Pinna
关键词:3 ;
6-Diazabicyclo[3.1.1]heptanes
;
Neuronal nicotinic acetylcholine receptors
;
Binding affinity
;
Modeling
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2008
4.
3-{2-[Bis-(4-fluorophenyl)methoxy]ethyl}-6-substituted-3,6-diazabicyclo[3.1.1]heptanes as novel potent dopamine uptake inhibitors
作者:
Giovanni Loriga
;
Stefania Ruiu
;
Ilaria Manca
;
Gabriele
Murineddu
;
Christian Dessi
;
Luca Pani
;
Gé
;
rard A. Pinna
关键词:
Cocaine abuse treatment
;
Synthesis of 3
;
6-diazabicyclo[3.1.1]heptanes
;
DAT inhibitors
刊名:Bioorganic and Medicinal Chemistry
出版年:2007
5.
Synthesis of 3,6-diazabicyclo[3.1.1]heptanes as novel ligands for the opioid receptors
作者:
Giovanni Loriga
;
Ilaria Manca
;
Gabriele
Murineddu
;
Giorgio Chelucci
;
Stefania Villa
;
Stefania Gessi
;
Lucio Toma
;
Giorgio Cignarella and Gerard A. Pinna
关键词:
Synthesis of 3
;
6-diazabicyclo[
;
3.1.1]
;
heptanes
;
Opioid receptors affinities and selectivities
;
Molecular modelling
刊名:Bioorganic and Medicinal Chemistry
出版年:2006
6.
Tricyclic pyrazoles. Part 2: Synthesis and biological evaluation of novel 4,5-dihydro-1H-benzo[g]indazole-based ligands for cannabinoid receptors
作者:
Murineddu
;
Gabriele
;
Ruiu
;
Stefania
;
Mussinu
;
Jean-Mario
;
Loriga
;
Giovanni
;
Grella
;
Giuseppe E.
;
et. al.
关键词:
Cannabinoids
;
4
;
5-Dihydro-1
H
-benzo[
;
g
]
;
indazoles
;
1-(2′
;
4′
;
-Dichlorophenyl)-7-iodo-
N
-piperidin-1-yl-4
;
5-dihydro-1
H
-benzo[
;
g
]
;
indazole-3-carboxamide
;
Selective CB
1
receptor ligands
刊名:Bioorganic & Medicinal Chemistry
出版年:2005
7.
Chromophore-modified bis-benzo[
g
]indole carboxamides: synthesis and antiproliferative activity of bis-benzo[
g
]indazole-3-carboxamides and related dimers
作者:
Pinna
;
Gé
;
rard A.
;
Pirisi
;
Maria A.
;
Mussinu
;
Jean-Mario
;
Murineddu
;
Gabriele
;
Loriga
;
Giovanni
;
et. al.
关键词:
Tricyclic pyrazole
;
Cytotoxic activity
;
Viscosity
刊名:Il Farmaco
出版年:2003
8.
Chiral pyridine N-oxides: useful ligands for asymmetric catalysis
作者:
Chelucci
;
Giorgio
;
Murineddu
;
Gabriele
;
Pinna
;
Gerard A.
刊名:Tetrahedron: Asymmetry
出版年:2004
9.
Chiral pyridine N-oxides: useful ligands for asymmetric catalysis
作者:
Chelucci
;
Giorgio
;
Murineddu
;
Gabriele
;
Pinna
;
Gerard A.
刊名:Tetrahedron: Asymmetry
出版年:2004
10.
Synthesis and application in asymmetric copper(I)-catalyzed allylic oxidation of a new chiral 1,10-phenanthroline derived from pinene
作者:
Chelucci
;
Giorgio
;
Loriga
;
Giovanni
;
Murineddu
;
Gabriele
;
Pinna
;
Gerard A.
关键词:1 ;
10-phenanthrolines
;
copper complex
;
allylic oxidation
;
enantioselectivity
刊名:Tetrahedron Letters
出版年:2002
1
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