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在“Elsevier电子期刊”中，命中：167条，耗时：0.1189448 秒

在所有数据库中总计命中：1,681条

1.Synthesis and antiviral evaluation of novel N-6 substituted adenosine analogues

作者：Youwu Hao^a ; Gaohui Zhou^a ; Wei Wu^a ; Yang Zhang^a ; Liming Tao^a ; Jianhua Yao^b ; Wenping Xu^a ; ^{xuwp@ecust.edu.cn}

关键词：Adenosine analogues ; Antiviral activities ; Coxsackie virus B3 ; Herpes simplex virus type 1 ; Higher selectivity index

刊名：Tetrahedron Letters

出版年：2017

2.Design, synthesis and analgesic/anti-inflammatory evaluation of novel diarylthiazole and diarylimidazole derivatives towards selective COX-1 inhibitors with better gastric profile

作者：Ahmed H. Abdelazeem^a ; ^b ; ^{ahmed.abdelazeem@pharm.bsu.edu.eg} ; ^{ahmed.pharm@yahoo.com} ; Mohammed T. El-Saadi^a ; Asmaa G. Safi El-Din^a ; Hany A. Omar^c ; ^d ; Samir M. El-Moghazy^e ; ^{samirelmoghazy@gmail.com}

关键词：Selective COX-1 ; Mofezolac ; Diarylthiazole ; Diarylimidazole ; Analgesic ; Anti-inflammatory ; Ulcerogenicity

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

3.Synthesis, anti-inflammatory, cyclooxygenases inhibitions assays and histopathological study of poly-substituted 1,3,5-triazines: Confirmation of regiospecific pyrazole cyclization by HMBC

作者：Heba A.H. Elshemy^a ; Eman K.A. Abdelall^a ; ^{eman.ahmed@pharm.bsu.edu.eg} ; ^{emanabdelall70@yahoo.com} ; Amany A. Azouz^b ; Abeer Moawad^c ; Waleed A.M. Ali^d ; Nesreen M. Safwat^e

关键词：S-Triazines ; COX-2 inhibitors ; Anti-inflammatory activity ; Enaminone ; HMBC ; Histopathology

刊名：European Journal of Medicinal Chemistry

出版年：2017

4.Functional synchrony and stimulus selectivity of visual cortical units: Comparison between cats and mice

作者：Lyes Bachatene^&dagger ; ; Vishal Bharmauria^&dagger ; ; Sarah Cattan ; Nayan Chanauria ; Faustin Armel Etindele-Sosso ; Sté ; phane Molotchnikoff ; ^{stephane.molotchnikoff@umontreal.ca" class="auth_mail" title="E-mail the corresponding author}

关键词：CS ; connectivity strength ; FR ; firing rate ; OSI ; orientation selectivity index

刊名：Neuroscience

出版年：2016

5.Genotoxicity and cytotoxicity of oxindole alkaloids from Uncaria tomentosa (cat's claw): Chemotype relevance

作者：Samuel Kaiser^a ; ^{samokaiser@yahoo.com.br" class="auth_mail" title="E-mail the corresponding author} ; Â ; nderson Ramos Carvalho^a ; Vanessa Pittol^a ; Fabrí ; cia Dietrich^b ; Fabiana Manica^b ; Michel Mansur Machado^c ; Luis Flá ; vio Souza de Oliveira^c ; Ana Maria Oliveira Battastini^b ; George Gonzá ; lez Ortega^a

关键词：POA ; pentacyclic oxindole alkaloids ; TOA ; tetracyclic oxindole alkaloids ; OAPFs ; oxindole alkaloid purified fractions ; T24 ; human bladder cancer cell line ; U-251-MG ; human glioblastoma cell line ; SI ; selectivity index ; SPEC ; speciophylline ; UNCF ; uncarine F ; PTER ; pteropodine ; ISPTER ; isopteropodine ; MIT ; mitraphylline ; ISMITR ; isomitraphylline ; RHY ; rhynchophylline ; ISRHY ; isorhynchophylline ; S ; stem bark samples ; L ; leaf samples ; CE ; crude extract

刊名：Journal of Ethnopharmacology

出版年：2016

6.Removal of pesticides from white and red wines by microfiltration

作者：Danae S. Doulia^a ; ^{ntoulia@mail.ntua.gr" class="auth_mail" title="E-mail the corresponding author} ; Efstathios K. Anagnos^a ; Konstantinos S. Liapis^b ; Demetrios A. Klimentzos^a

关键词：AEI ; antagonistic (or synergistic) effect index ; CA ; cellulose acetate ; Cm ; capacity of each membrane ; CN ; cellulose nitrate ; Kow ; octanol-water partition coefficient ; MPR ; mean pesticide removal ; MRL ; maximum residue limit ; MRSP ; mean removal of significantly removed pesticides ; N ; total number of pesticides ; NY ; nylon ; PA ; polyamide ; PESU ; polyethersulfone ; PR ; pesticide removal ; RC ; regenerated cellulose ; Sm ; selectivity of each membrane ; TAEI ; total antagonistic effect index ; TSEI ; total syn

刊名：Journal of Hazardous Materials

出版年：2016

7.Inhibition of hepatitis B virus replication by targeting ribonucleotide reductase M2 protein

作者：Xia Liu^a ; ^e ; ¹ ; Zhijian Xu^b ; ¹ ; Chuanwei Hou^b ; ¹ ; Meng Wang^b ; Xinhuan Chen^a ; ^c ; Qinghui Lin^a ; Rui Song^a ; Meng Lou^a ; Lijun Zhu^a ; Yunqing Qiu^d ; Zhi Chen^d ; Chunhao Yang^b ; ^{chyang@simm.ac.cn" class="auth_mail" title="E-mail the corresponding author} ; Weiliang Zhu^b ; ^{wlzhu@mail.shcnc.ac.cn" class="auth_mail" title="E-mail the corresponding author} ; Jimin Shao^a ; ^{shaojimin@zju.edu.cn" class="auth_mail" title="E-mail the corresponding author}

关键词：3TC ; lamivudine ; cccDNA ; covalently-closed-circular DNA ; CI ; combination index ; CMC ; Comprehensive Medicinal Chemistry ; Gem ; gemcitabine ; HBV ; hepatitis B virus ; HCC ; hepatocellular carcinoma ; HU ; hydroxyurea ; NDPs ; ribonucleoside diphosphates ; dNDPs ; deoxyribonucleoside diphosphates ; RR ; ribonucleotide reductase ; RRM1 ; RR large subunit M1 ; RRM2 ; RR small subunit M2 ; RRM2B ; RR small subunit M2B ; SI ; selectivity index ; YZ51 ; 4-cyclopropyl-2-fluoro-N-(4-hydroxyphenyl) benzamide

刊名：Biochemical Pharmacology

出版年：2016

8.Synthesis and biological evaluation of quinoxaline di-N-oxide derivatives with in vitro trypanocidal activity

作者：Silvia Pé ; rez-Silanes^a ; ^b ; Enrique Torres^a ; Leire Arbillaga^c ; Javier Varela^d ; Hugo Cerecetto^d ; Mercedes Gonzá ; lez^d ; Amaya Azqueta^c ; ^e ; Elsa Moreno-Viguri^a ; ^b ; ^{emviguri@unav.es" class="auth_mail" title="E-mail the corresponding author}

关键词：BFX ; benzofuroxan ; CD ; chagas disease ; Nfx ; Nifurtimox ; Bnz ; Benznidazol ; NCE ; new chemical entity ; N.T. ; not tested ; NTD ; Neglected Tropical Diseases ; PGI ; percentage of growth inhibition ; SI ; selectivity index ; TPP ; Target Product Profile

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

9.Effects of nitro-heterocyclic derivatives against Leishmania (Leishmania) infantum promastigotes and intracellular amastigotes

作者：Simone Carolina Soares Petri e Silva^a ; Fanny Palace-Berl^b ; Leoberto Costa Tavares^b ; Sandra Regina Castro Soares^a ; José ; Angelo Lauletta Lindoso^a ; ^c ; ^d ; ^{jlindoso@usp.br" class="auth_mail" title="E-mail the corresponding author}

关键词：Leishmania (L.) infantum ; Nitroheterocyclic compounds ; THP-1 cells ; Nitric oxide ; Apoptosis

刊名：Experimental Parasitology

出版年：2016

10.In vitro and in vivo preclinical profile of abediterol (LAS100977), an inhaled long-acting β₂-adrenoceptor agonist, compared with indacaterol, olodaterol and vilanterol

作者：Mò ; nica Aparici ; ^{monica.aparici@almirall.com" class="auth_mail" title="E-mail the corresponding author} ; Amadeu Gavaldà ; Israel Ramos ; Carla Carcasona ; Raquel Otal ; Joan Antoni Ferná ; ndez-Blanco ; Jose Luí ; s Montero ; Vicente Marco García ; Rosa Ló ; pez ; Jorge De Alba ; Christopher Doe ; Carlos Puig ; Dolors Vilella ; Montserrat Miralpeix

关键词：ANOVA ; analysis of variance ; CGP12177 ; 4-(3-tert-butylamino-2-hydroxypropoxy)-benzimidazol-2-one hydrochloride ; COPD ; chronic obstructive pulmonary disease ; EFS ; electrical field stimulation ; EC50 ; concentration that induces 50% of the maximum effect ; Emax ; maximum effect ; FDA ; US Food and Drug Administration ; FEV1 ; forced expiratory volume in 1 s ; IC50 ; half maximal inhibitory concentration ; LABA ; long-acting β-adrenoceptor agonist

刊名：European Journal of Pharmacology

出版年：2016

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