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CNKI学位论文(1)
在“
Elsevier电子期刊
”中,
命中:
7
条,耗时:小于0.01 秒
在所有数据库中总计命中:
1
条
1.
Identification and synthesis of potent and selective pyridyl-isoxazole based agonists of sphingosine-1-phosphate 1 (S1P
1
)
作者:
Junqing Guo
;
junqing.guo@bms.com" class="auth_mail" title="E-mail the corresponding author
;
Scott H. Watterson
;
Steven H. Spergel
;
James Kempson
;
Charles M. Langevine
;
Ding Ren Shen
;
Melissa Yarde
;
Mary Ellen Cvijic
;
Dana Banas
;
Richard Liu
;
Suzanne J. Suchard
;
Kathleen
Gillooly
;
Tracy Taylor
;
Sandra Rex-Rabe
;
David J. Shuster
;
Kim W. McIntyre
;
Georgia Cornelius
;
Celia D&rsquo
;
Arienzo
;
Anthony Marino
;
Praveen Balimane
;
Luisa Salter-Cid
;
Murray McKinnon
;
Joel C. Barrish
;
Percy H. Carter
;
William J. Pitts
;
Jenny Xie
;
Alaric J. Dyckman
关键词:
Sphingosine-1-phosphate
;
Sphingosine-1-phosphate 1
;
S1P1
;
Isoxazole
;
FTY720
;
Fingolimod
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
2.
Imidazo[4,5-d]thiazolo[5,4-b]pyridine based inhibitors of IKK2: Synthesis, SAR, PK/PD and activity in a preclinical model of rheumatoid arthritis
作者:
Alaric J. Dyckman
;
Charles M. Langevine
;
Claude Quesnelle
;
James Kempson
;
Junqing Guo
;
Patrice Gill
;
Steven H. Spergel
;
Scott H. Watterson
;
Tianle Li
;
David S. Nirschl
;
Kathleen
M.
Gillooly
;
Mark A. P
关键词:
IKK
;
IKK2
;
IKKβ
;
NF-κ
B
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2011
3.
5-Amino-pyrazoles as potent and selective p38α inhibitors
作者:
Jagab
;
hu Das
;
Robert V. Moquin
;
Alaric J. Dyckman
;
Tianle Li
;
Sidney Pitt
;
Rosemary Zhang
;
Ding Ren Shen
;
Kim W. McIntyre
;
Kathleen
Gillooly
;
Arthur M. Doweyko
;
John A. Newitt
;
John S. Sack
;
Hongjian
关键词:
p38 Inhibitors
;
Amino-pyrazoles
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
4.
PS3-21 Preclinical validation of CCR5 pharmacodynamic biomarkers
作者:
Chen-Yi Hung
;
Kathleen
Gillooly
;
Jesse Miller
;
Ragini Vuppugalla
;
Jian Pang
;
Vojkan Susulic
;
Nicole Vincelli
;
Sophie Beyer
;
Jenny Xie
;
Kim McIntyre
;
W
;
a West
;
Percy Carter
;
Paul Davies
;
Luisa Salter-C
刊名:Cytokine
出版年:2010
5.
The discovery of (R)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbamoyl)phenyl) thiazole-5-carboxamide (BMS-640994)—A potent and efficacious p38α MAP kinase inhibitor
作者:
John Hynes Jr.
;
Hong Wu
;
Sidney Pitt
;
Ding Ren Shen
;
Rosemary Zhang
;
Gary L. Schieven
;
Kathleen
M.
Gillooly
;
David J. Shuster
;
Tracy L. Taylor
;
XiaoXia Yang
;
Kim W. McIntyre
;
Murray McKinnon
;
Hongjian
关键词:
p38
;
MAP kinase
;
Aminothiazole
;
TNF
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2008
6.
Synthesis and SAR of new pyrrolo[2,1-f][1,2,4]triazines as potent p38α MAP kinase inhibitors
作者:
Stephen T. Wrobleski
;
Shuqun Lin
;
John Hynes Jr.
;
Hong Wu
;
Sidney Pitt
;
Ding Ren Shen
;
Rosemary Zhang
;
Kathleen
M.
Gillooly
;
David J. Shuster
;
Kim W. McIntyre
;
Arthur M. Doweyko
;
Kevin F. Kish
;
Jeffre
关键词:
p38
;
Kinase
;
Inflammation
;
Pyrrolotriazines
;
TNF-
;
//www.sciencedirect.com/scidirimg/entities/204e.gif"" alt=""greek small letter alpha"" title=""greek small letter alpha"" border=""0"">
;
IL-1
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2008
7.
Pyrazolo-pyrimidines: A novel heterocyclic scaffold for potent and selective p38α inhibitors
作者:
Jagab
;
hu Das
;
Robert V. Moquin
;
Sidney Pitt
;
Rosemary Zhang
;
Ding Ren Shen
;
Kim W. McIntyre
;
Kathleen
Gillooly
;
Arthur M. Doweyko
;
John S. Sack
;
Hongjian Zhang
;
Susan E. Kiefer
;
Kevin Kish
;
Murray McK
关键词:
p38
;
//www.sciencedirect.com/scidirimg/entities/204e.gif"" alt=""greek small letter alpha"" title=""greek small letter alpha"" border=""0""> inhibitors
;
Pyrazolo-pyrimidines
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2008
1
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