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内部出版物
在“
Elsevier电子期刊
”中,
命中:
101
条,耗时:0.0649691 秒
1.
Chemical exploration of 4-(4-fluorobenzyl)piperidine fragment for the development of new tyrosinase inhibitors
作者:
Stefania Ferro
a
;
sferro@unime.it
;
Laura De Luca
a
;
Maria Paola Germanò
;
a
;
Maria Rosa Buemi
a
;
Laura Ielo
a
;
Giovanna Certo
a
;
b
;
Margarita Kanteev
c
;
Ayelet Fishman
c
;
Antonio Rapisarda
a
;
Rosaria Gitto
a
关键词:
Synthesis
;
Tyrosinase inhibitors
;
SARs
;
Kinetic mechanism
;
Docking studies
;
Crystallography
刊名:European Journal of Medicinal Chemistry
出版年:2017
2.
Bioactive constituents from the leaves of Quercus phillyraeoides A. Gray for α-glucosidase inhibitor activity with concurrent antioxidant activity
作者:
Anastasia Wheni Indrianingsih
a
;
b
;
Sanro Tachibana
c
;
tatibana@agr.ehime-u.ac.jp" class="auth_mail" title="E-mail the corresponding author
关键词:
Quercus phillyraeoides A. Gray
;
α-Glucosidase inhibitor
;
Antioxidative activity
;
Lineweaver
&
ndash
;
Burk plot
刊名:Food Science and Human Wellness
出版年:2016
3.
Inhibitory effect on key enzymes relevant to acute type-2 diabetes and antioxidative activity of ethanolic extract of Artocarpus heterophyllus stem bark
作者:
Basiru Olaitan Ajiboye
;
bash1428@yahoo.co.uk" class="auth_mail" title="E-mail the corresponding author
;
Oluwafemi Adeleke Ojo
;
Oluwatosin Adeyonu
;
Oluwatosin Imiere
;
Isreal Olayide
;
Adewale Fadaka
;
Babatunji Emmanuel Oyinloye
关键词:
Artocarpus heterophyllus
;
GC&
ndash
;
MS
;
α-Amylase
;
α-Glucosidase
刊名:Journal of Acute Disease
出版年:2016
4.
Synthesis of 3-acyloxyxanthone derivatives as α-glucosidase inhibitors: A further insight into the 3-substituents‿effect
作者:
Gai-Li Li
a
;
Chao-Yun Cai
a
;
&dagger
;
;
Jia-Yun He
a
;
Li Rao
a
;
Lin Ma
a
;
Yan Liu
b
;
yanliu@gdut.edu.cn" class="auth_mail" title="E-mail the corresponding author
;
Bo Wang
a
;
ceswb@mail.sysu.edu.cn" class="auth_mail" title="E-mail the corresponding author
关键词:
Xanthone derivatives
;
α-Glucosidase
;
Inhibitory activity
;
Inhibition kinetics
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
5.
Design, synthesis and evaluation of novel 7-aminoalkyl-substituted flavonoid derivatives with improved cholinesterase inhibitory activities
作者:
Wen Luo
a
;
&dagger
;
;
luowen83@henu.edu.cn" class="auth_mail" title="E-mail the corresponding author
;
Ying Chen
a
;
&dagger
;
;
Ting Wang
a
;
Chen Hong
a
;
Li-Ping Chang
a
;
Cong-Cong Chang
a
;
Ya-Cheng Yang
a
;
Song-Qiang Xie
b
;
Chao-Jie Wang
a
;
wcjsxq@163.com" class="auth_mail" title="E-mail the corresponding author
关键词:
Flavonoid derivatives
;
Cholinesterase
;
Anti-Alzheimer agent
;
Molecular modeling
;
Cytotoxicity
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
6.
Tyrosinase inhibitory constituents from a polyphenol enriched fraction of rose oil distillation wastewater
作者:
Jessica Solimine
a
;
Eliane Garo
b
;
Jonas Wedler
a
;
Krasimir Rusanov
c
;
Orlando Fertig
b
;
Matthias Hamburger
b
;
Ivan Atanassov
c
;
Veronika Butterweck
a
;
veronika.butterweck@fhnw.ch" class="auth_mail" title="E-mail the corresponding author
关键词:
Rosa damascena
;
Rosaceae
;
Rose oil distillation
;
Tyrosinase inhibition
;
Hyperpigmentation
;
Ellagic acid
刊名:Fitoterapia
出版年:2016
7.
2-Benzoyl-6-benzylidenecyclohexanone analogs as potent dual inhibitors of acetylcholinesterase and butyrylcholinesterase
作者:
Sze Wei Leong
a
;
Faridah Abas
a
;
b
;
faridah_abas@upm.edu.my" class="auth_mail" title="E-mail the corresponding author
;
Kok Wai Lam
c
;
Khozirah Shaari
a
;
d
;
Nordin H. Lajis
a
;
nordinlajis@gmail.com" class="auth_mail" title="E-mail the corresponding author
关键词:
Acetylcholinesterase
;
Butyrylcholinesterase
;
2-Benzoyl-6-benzylidenecyclohexanone
;
Kinetic studies
;
Molecular docking
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
8.
Natural cholinesterase inhibitors from Myristica cinnamomea King
作者:
Siti Mariam Abdul Wahab
a
;
Yasodha Sivasothy
a
;
Sook Yee Liew
a
;
b
;
Marc Litaudon
c
;
Jamaludin Mohamad
d
;
Khalijah Awang
a
;
b
;
khalijah@um.edu.my" class="auth_mail" title="E-mail the corresponding author
关键词:
Myristica cinnamomea King
;
Myristicaceae
;
Acylphenols
;
Dimeric acylphenols
;
Malabaricone E
;
Acetylcholinesterase enzyme
;
Butyrylcholinesterase enzyme
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
9.
ArgTX-636, a polyamine isolated from spider venom: A novel class of melanogenesis inhibitors
作者:
Marion Verdoni
a
;
b
;
Hermine Roudaut
b
;
c
;
Harold De Pomyers
d
;
Didier Gigmes
a
;
Denis Bertin
a
;
José
;
Luis
c
;
Abd Haq Bengeloune
b
;
Kamel Mabrouk
a
;
kamel.mabrouk@univ-amu.fr" class="auth_mail" title="E-mail the corresponding author
关键词:
Melanogenesis
;
Tyrosinase
;
Tyrosinase related protein 1 (TRP-1)
;
Hyperpigmentation
;
DOPA oxydase activity
;
DHICA oxydase activity
;
Spider venoms
;
Argiotoxine
;
ArgTX-636
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
10.
Cholinesterase inhibitory activity of isoquinoline alkaloids from three Cryptocarya species (Lauraceae)
作者:
Wan Nurul Nazneem Wan Othman
a
;
Sook Yee Liew
a
;
b
;
Kooi Yeong Khaw
c
;
&dagger
;
;
Vikneswaran Murugaiyah
c
;
Marc Litaudon
d
;
Khalijah Awang
a
;
b
;
khalijah@um.edu.my" class="auth_mail" title="E-mail the corresponding author
关键词:
AChE
;
acetylcholinesterase
;
BChE
;
butyrylcholinesterase
;
ACh
;
acetylcholine
;
AD
;
Alzheimer&rsquo
;
s disease
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
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