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在“Elsevier电子期刊”中，命中：540条，耗时：0.1069847 秒

在所有数据库中总计命中：938条

1.Emamectin is a non-selective allosteric activator of nicotinic acetylcholine receptors and GABA_A/C receptors

作者：Xiaojun Xu^a ; ^b ; Caraline Sepich^c ; Ronald J. Lukas^b ; Guonian Zhu^a ; Yongchang Chang^b ; ^{Yongchang.chang@dignityhealth.org" class="auth_mail" title="E-mail the corresponding author}

关键词：Emamectin ; Ivermectin ; Nicotinic receptor ; GABAA/C receptor ; Allosteric activation

刊名：Biochemical and Biophysical Research Communications

出版年：2016

2.Synthesis, radiolabeling and evaluation of novel amine guanidine derivatives as potential positron emission tomography tracers for the ion channel of the N-methyl-d-aspartate receptor

作者：Pieter J. Klein ; ^{pj.klein@vumc.nl" class="auth_mail" title="E-mail the corresponding author} ; Marion Chomet ; Athanasios Metaxas ; Johannes A.M. Christiaans¹ ; Esther Kooijman ; Robert C. Schuit ; Adriaan A. Lammertsma ; Bart N.M. van Berckel ; Albert D. Windhorst

关键词：PET ; NMDA ; Radiolabeling ; SAR ; Non-competitive antagonists

刊名：European Journal of Medicinal Chemistry

出版年：2016

3.Discovery of novel 2′,4′-dimethyl-[4,5′-bithiazol]-2-yl amino derivatives as orally bioavailable TRPV4 antagonists for the treatment of pain: Part 1

作者：Naoki Tsuno^a ; ^{naoki.tsuno@shionogi.co.jp" class="auth_mail" title="E-mail the corresponding author} ; Akira Yukimasa^a ; Osamu Yoshida^a ; Yusuke Ichihashi^a ; Takatsugu Inoue^a ; Tatsuhiko Ueno^a ; Hiroki Yamaguchi^a ; Hidetoshi Matsuda^b ; Satoko Funaki^c ; Natsue Yamanada^a ; Miki Tanimura^a ; Daiki Nagamatsu^c ; Yoko Nishimura^c ; Tetsuji Ito^c ; Masahiko Soga^a ; Narumi Horita^b ; Miyuki Yamamoto^a ; Mikie Hinata^a ; Masayuki Imai^d ; Yasuhide Morioka^a ; Toshiyuki Kanemasa^a ; Gaku Sakaguchi^d ; Yasuyoshi Iso^a

关键词：Transient Receptor Potential Vanilloid 4 ; TRPV4 antagonist ; Ion channel ; Vanilloid receptor ; Thiazole ; Bi-cyclic ; Pain

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

4.Phencyclidine-induced disruption of oscillatory activity in prefrontal cortex: Effects of antipsychotic drugs and receptor ligands

作者：L. Lladó ; -Pelfort^a ; ^b ; ^c ; ¹ ; E. Troyano-Rodriguez^a ; ^b ; ^c ; ¹ ; H.E. van den Munkhof^a ; ^c ; A. Cervera-Ferri^d ; N. Jurado^a ; ^b ; ^c ; M. Nú ; ñ ; ez-Calvet^a ; ^c ; F. Artigas^a ; ^b ; ^c ; P. Celada^a ; ^b ; ^c ; ^{pau.celada@iibb.csic.es" class="auth_mail" title="E-mail the corresponding author}

关键词：Antipsychotic drugs ; NMDA receptor antagonists ; Oscillations ; Phencyclidine ; Prefrontal cortex ; Schizophrenia

刊名：European Neuropsychopharmacology

出版年：2016

5.Current basis for discovery and development of aryl hydrocarbon receptor antagonists for experimental and therapeutic use in atherosclerosis

作者：Larissa Pernomian ; ^{l.pernomian@usp.br" class="auth_mail" title="E-mail the corresponding author} ; Carlos H.T.P. da Silva

关键词：Atherosclerosis ; Cigarette smoke ; Aryl hydrocarbon receptor antagonists ; Molecular modeling ; Drug design

刊名：European Journal of Pharmacology

出版年：2015

6.Structural studies, homology modeling and molecular docking of novel non-competitive antagonists of GluK1/GluK2 receptors

作者：Agnieszka A. Kaczor ; Zbigniew Karczmarzyk ; Andrzej Fruzi艅ski ; Kalevi Pihlaja ; Jari Sinkkonen ; Kirsti Wiin盲maki ; Christiane Kronbach ; Klaus Unverferth ; Antti Poso ; Dariusz Matosiuk

关键词：Homology modeling ; Indole derivatives ; Kainate receptors ; Molecular docking ; X-ray structure determination

刊名：Bioorganic and Medicinal Chemistry

出版年：15 January, 2014

7.The effect of non-competitive NMDA receptor antagonist MK-801 on neuronal activity in rodent prefrontal cortex: an animal model for cognitive symptoms of schizophrenia

作者：Kevin Blot ; Jing Bai ; Satoru Otani

关键词：MK-801 ; NMDA receptor hypofunction ; Long-term potentiation ; LTP ; Hippocampo-prefrontal cortex pathway ; In vivo electrophysiology ; Schizophrenia

刊名：Journal of Physiology-Paris

出版年：December, 2013

8.Recent developments in 5-HT₃ receptor pharmacology

作者：Andrew J. Thompson ^{ajt44@cam.ac.uk}

关键词：5-HT3 ; antagonist ; agonist ; competitive ; non-competitive ; binding site

刊名：Trends in Pharmacological Sciences

出版年：2013

9.Non-competitive and selective dipeptidyl peptidase IV inhibitors with phenethylphenylphthalimide skeleton derived from thalidomide-related α-glucosidase inhibitors and liver X receptor antagonists

作者：Kazunori Motoshima^a ; Kazuyuki Sugita^a ; Yuichi Hashimoto ; ^a ; ^{hashimot@iam.u-tokyo.ac.jp"" rel=""nofollow} ; Minoru Ishikawa^a

关键词：Dipeptidyl peptidase IV ; Enzyme inhibitor ; Phthalimide ; Non-competitive inhibition ; Subtype selectivity

刊名：Bioorganic and Medicinal Chemistry Letters

出版年：2011

10.Putative TRP channel antagonists, SKF 96365, flufenamic acid and 2-APB, are non-competitive antagonists at recombinant human ¦Á1¦Â2¦Ã2 GABA_A receptors

作者：M.G. Rae^a ; ^m.rae@ucc.ie ; J. Hilton^b ; J. Sharkey^c

关键词：SKF 96365 ; 1-(2-(4-methoxyphenyl)-2-(3-(4-methoxyphenyl)propoxy)ethyl-1H-imidazole hydrochloride ; FF (flufenamic acid) ; N-(3-(trifluoromethyl)-phenyl)anthranilic acid ; 2-APB ; 2-aminoethoxydiphenyl borate ; GABA ; ¦Ã-amino butyric acid ; TRP ; transient recept

刊名：Neurochemistry International

出版年：2012

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