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在“
Elsevier电子期刊
”中,
命中:
7,141
条,耗时:0.044979 秒
在所有数据库中总计命中:
102,699
条
1.
Simultaneous Inhibition of
PI3K
δ and PI3Kα Induces ABC-DLBCL Regression by Blocking BCR-Dependent and -Independent Activation of NF-κB and AKT
作者:
Juliane Paul
1
;
5
;
Maurice Soujon
1
;
5
;
Antje M. Wengner
1
;
Sabine Zitzmann-Kolbe
1
;
Andrea Sturz
1
;
Katja Haike
1
;
Koh Hui Keng Magdalene
2
;
Sze Huey Tan
3
;
Martin Lange
1
;
Soo Yong Tan
2
;
6
;
Dominik Mumberg
1
;
Soon Thye Lim
4
;
Karl Ziegelbauer
1
;
Ningshu Liu
1
;
ningshu.liu@bayer.com
关键词:
PI3K
α
;
PI3K
δ
;
NF-κB
;
BCR
;
MYD88
;
CARD11
;
DLBCL
;
follicular lymphoma
;
ibrutinib-resistance
;
copanlisib
刊名:Cancer Cell
出版年:2017
2.
Identification of allosteric binding sites for
PI3K
α oncogenic mutant specific inhibitor design
作者:
Michelle S. Miller
a
;
Sweta Maheshwari
b
;
Fiona M. McRobb
c
;
Kenneth W. Kinzler
d
;
L. Mario Amzel
b
;
Bert Vogelstein
d
;
Sandra B. Gabelli
a
;
b
;
e
;
gabelli@jhmi.edu
关键词:
PI
K3CA
;
PI3K
;
PI
P2
;
PI
P3
;
Fragment-based drug discovery
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
3.
La inhibición de la
PI3K
γ protege contra la miocardiopatía diabética en ratones
作者:
Angelo Maffei
a
;
Giuseppe Cifelli
a
;
Raimondo Carnevale
a
;
Roberta Iacobucci
a
;
Fabio Pallante
a
;
Valentina Fardella
a
;
Stefania Fardella
a
;
Emilio Hirsch
b
;
Giuseppe Lembo
a
;
c
;
Daniela Carnevale
a
;
c
;
Daniela.carnevale@uniroma1.it
关键词:
Diabetes mellitus
;
Miocardiopatí
a ;
Fá
;
rmacos en investigació
n ;
Proteí
;
na
PI3K
γ
;
Rató
n
刊名:Revista Española de Cardiología
出版年:2017
4.
PI3K
γ Inhibition Protects Against Diabetic Cardiomyopathy in Mice
作者:
Angelo Maffei
a
;
Giuseppe Cifelli
a
;
Raimondo Carnevale
a
;
Roberta Iacobucci
a
;
Fabio Pallante
a
;
Valentina Fardella
a
;
Stefania Fardella
a
;
Emilio Hirsch
b
;
Giuseppe Lembo
a
;
c
;
Daniela Carnevale
a
;
c
;
Daniela.carnevale@uniroma1.it
关键词:
Diabetes mellitus
;
Cardiomyopathy
;
Investigational drugs
;
PI3K
γ protein
;
Mouse
刊名:Revista Española de Cardiología (English Edition)
出版年:2017
5.
Kinetic modelling of in vitro data of
PI3K
, mTOR1, PTEN enzymes and on-target inhibitors Rapamycin, BEZ235, and LY294002
作者:
Alexey Goltsov
a
;
a.goltsov@abertay.ac.uk
;
Ghassan Tashkandi
b
;
s1163633@exseed.ed.ac.uk
;
Simon P. Langdon
b
;
Simon.Langdon@ed.ac.uk
;
David J. Harrison
c
;
David.Harrison@st-andrews.ac.uk
;
James L. Bown
a
;
d
;
j.bown@abertay.ac.uk
关键词:
Kinetic modelling
;
PI3K
;
mTOR1
;
PTEN
;
Rapamycin
;
BEZ235
刊名:European Journal of Pharmaceutical Sciences
出版年:2017
6.
Discovery of triazole aminopyrazines as a highly potent and selective series of
PI3K
δ inhibitors
作者:
Ina Terstiege
a
;
Ina.Terstiege@astrazeneca.com
;
Matthew Perry
a
;
Jens Petersen
b
;
Christian Tyrchan
a
;
Tor Svensson
a
;
Helena Lindmark
b
;
Linda Ö
;
ster
b
关键词:
Phosphoinositide 3-kinase
;
PI3K
δ inhibitor
;
Aminopyrazine
;
Inflammation
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
7.
Target regulation of
PI3K
/Akt/mTOR pathway by cannabidiol in treatment of experimental multiple sclerosis
作者:
Sabrina Giacoppo
a
;
Federica Pollastro
b
;
Gianpaolo Grassi
c
;
Placido Bramanti
a
;
Emanuela Mazzon
a
;
emazzon.irccs@gmail.com
关键词:
Cannabidiol
;
Multiple sclerosis
;
PI3K
/Akt/mTOR pathway
;
BDNF
;
Inflammation
;
Neuronal survival
刊名:Fitotera
pi
a
出版年:2017
8.
Inhibiting
PI3K
-AKt signaling pathway is involved in antitumor effects of ginsenoside Rg3 in lung cancer cell
作者:
Qipeng Xie
a
;
1
;
Huaikai Wen
a
;
1
;
Qiong Zhang
b
;
Weihe Zhou
c
;
Xiaoming Lin
d
;
Deyao Xie
d
;
Yu Liu
d
;
48936053@qq.com
关键词:
Ginsenoside Rg3
;
Lung cancer
;
Apoptosis
;
PI3K
/Akt
刊名:Biomedicine & Pharmacotherapy
出版年:2017
9.
SAR study of 5-alkynyl substituted quinazolin-4(3H)-ones as phosphoinositide 3-kinase delta (
PI3K
δ) inhibitors
作者:
Manman Wei
a
;
c
;
1
;
Xi Zhang
b
;
1
;
Xiang Wang
b
;
Zilan Song
a
;
Jian Ding
b
;
Ling-Hua Meng
b
;
lhmeng@simm.ac.cn
;
Ao Zhang
a
;
c
;
aozhang@simm.ac.cn
关键词:
Chronic lymphocytic leukemia
;
PI3K
δ
;
Structure-activity relationship
;
5-Alkynyl
;
Quinazolinone
刊名:European Journal of Medicinal Chemistry
出版年:2017
10.
Discovery of 7-(3-(
pi
perazin-1-yl)phenyl)pyrrolo[2,1-f][1,2,4]triazin-4-amine derivatives as highly potent and selective PI
3K
δ inhibitors
作者:
Lan-Ying Qin
;
lan-ying.qin@bms.com
;
Zheming Ruan
;
Robert J. Cherney
;
T.G. Murali Dhar
;
James Neels
;
Carolyn A. Weigelt
;
John S. Sack
;
Anurag S. Srivastava
;
Lyndon A.M. Cornelius
;
Joseph A. Tino
;
Kevin Stefanski
;
Xiaomei Gu
;
Jenny Xie
;
Vojkan Susulic
;
Xiaoxia Yang
;
Melissa Yarde-Chinn
;
Stacey Skala
;
Ruth Bosnius
;
Christine Goldstein
;
Paul Davies
;
Stefan Ruepp
;
Luisa Salter-Cid
;
Rajeev S. Bhide
;
Michael A. Poss
关键词:
PI3K
δ
;
7-Phenylpyrrolo[2
;
1-f][1
2 ;
4]triazin-4-amine
;
Autoimmune diseases
;
Rheumatoid arthritis
;
Phosphoinositide 3-kinases
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
1
2
3
4
5
6
7
8
9
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作者(4)
关键词(1918)
文摘(5868)
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