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在“Elsevier电子期刊”中，命中：82条，耗时：0.0139913 秒

在所有数据库中总计命中：698条

1.Discovery of 2-(1H-indol-5-ylamino)-6-(2,4-difluorophenylsulfonyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one (7ao) as a potent selective inhibitor of Polo like kinase 2 (PLK2)

作者：M.V. Ramana Reddy^a ; ^{r.reddy@mssm.edu" class="auth_mail" title="E-mail the corresponding author} ; Balireddy Akula^b ; ^&dagger ; ; Shashidhar Jatiani^a ; ^&dagger ; ; Rodrigo Vasquez-Del Carpio^a ; ^&dagger ; ; Vinay K. Billa^a ; ^&dagger ; ; Muralidhar R. Mallireddigari^b ; ¹ ; Stephen C. Cosenza^a ; D.R.C. Venkata Subbaiah^a ; E. Vijaya Bharathi^a ; Venkat R. Pallela^b ; Poornima Ramkumar^a ; Rinku Jain^c ; Aneel K. Aggarwal^c ; E. Premkumar Reddy^a ; ^{ep.reddy@mssm.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：PLK ; Kinase inhibitor ; Apoptosis ; Cytotoxicity

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

2.Identification of acylthiourea derivatives as potent Plk1 PBD inhibitors

作者：Taikangxiang Yun^a ; Tan Qin^b ; Ying Liu^a ; ^b ; ^{liuying@pku.edu.cn" class="auth_mail" title="E-mail the corresponding author} ; Luhua Lai^a ; ^b ; ^c ; ^{lhlai@pku.edu.cn" class="auth_mail" title="E-mail the corresponding author}

关键词：Polo-like kinase 1 ; Polo-box domain ; Small molecular inhibitor ; Halogenosulfamoylphenyl acylthiourea ; Binding affinity ; In vitro assay

刊名：European Journal of Medicinal Chemistry

出版年：2016

3.In vitro anticancer properties and biological evaluation of novel natural alkaloid jerantinine B

作者：Mohannad E. Qazzaz^a ; Vijay J. Raja^a ; Kuan-Hon Lim^b ; Toh-Seok Kam^c ; Jong Bong Lee^a ; Pavel Gershkovich^a ; Tracey D. Bradshaw^a ; ^{tracey.bradshaw@nottingham.ac.uk" class="auth_mail" title="E-mail the corresponding author} ; ^{paxmq@nottingham.ac.uk" class="auth_mail" title="E-mail the corresponding author}

关键词：EB 1 ; end-binding protein 1 ; JB ; jerantinine B ; JBA ; jerantinine B acetate ; MTA ; microtubule targeting agent ; NP ; natural product ; ROS ; reactive oxygen species ; PLK1 ; Polo-like kinase 1

刊名：Cancer Letters

出版年：2016

4.355 - Therapeutic potential of novel PLK1 inhibitor CYC140 in esophageal cancer and acute leukemia

作者：S. Moureau ; E. Pohler ; K. Kroboth ; C. Saladino ; C. MacKay ; J. Hollick ; D. Zheleva ; S. Frame ; D. Blake

刊名：European Journal of Cancer

出版年：2016

5.Propionibacterium acnes inhibits FOXM1 and induces cell cycle alterations in human primary prostate cells

作者：Behnam Sayanjali^a ; Gitte J.M. Christensen^b ; Munir A. Al-Zeer^a ; Hans-Joachim Mollenkopf^a ; Thomas F. Meyer^a ; ^{meyer@mpiib-berlin.mpg.de" class="auth_mail" title="E-mail the corresponding author} ; Holger Brü ; ggemann^b

关键词：IL ; interleukin ; EPCAM ; epithelial cell adhesion molecule ; PrEC ; primary prostate epithelial cells ; CFU ; colony forming unit ; IPA ; Ingenuity Pathway Analysis ; DAVID ; Database for Annotation Visualization and Integrated Discovery ; MOI ; multiplicity of infection ; p.i. ; post infection ; PLK1 ; Polo-like kinase 1 ; CCNB1 ; Cyclin B1 ; CENPF ; Centromere protein F ; APC ; anaphase-promoting complex/cyclosome

刊名：International Journal of Medical Microbiology

出版年：2016

6.Neurobehavioral effects of liraglutide and sitagliptin in experimental models

作者：Mayur Kamble^a ; Rachna Gupta^b ; Harmeet S. Rehan^a ; Lalit K. Gupta^a ; ^{lkg71@rediffmail.com" class="auth_mail" title="E-mail the corresponding author}

关键词：Anxiety ; Cognition ; Depression ; GLP-1 ; Liraglutide ; Sitagliptin

刊名：European Journal of Pharmacology

出版年：2016

7.Promoting tumor penetration of nanoparticles for cancer stem cell therapy by TGF-β signaling pathway inhibition

作者：Zu-Qi Zuo^a ; ¹ ; Kai-Ge Chen^a ; ¹ ; Xiao-Yuan Yu^a ; Gui Zhao^a ; Song Shen^a ; Zhi-Ting Cao^b ; Ying-Li Luo^a ; Yu-Cai Wang^a ; Jun Wang^a ; ^b ; ^c ; ^d ; ^{jwang699@ustc.edu.cn" class="auth_mail" title="E-mail the corresponding author}

关键词：Tumor penetration ; Cancer stem cell ; Nanoparticle drug delivery system ; siRNA ; TGF-β signaling pathway inhibition

刊名：Biomaterials

出版年：2016

8.BI2536 - A PLK inhibitor augments paclitaxel efficacy in suppressing tamoxifen induced senescence and resistance in breast cancer cells

作者：B.N. Prashanth Kumar ; Shashi Rajput ; Rashmi Bharti ; Sheetal Parida ; Mahitosh Mandal ; ^{mahitosh@smst.iitkgp.ernet.in" class="auth_mail" title="E-mail the corresponding author}

关键词：Paclitaxel ; BI2536 ; p38 signaling ; Tamoxifen resistant breast cancer ; VEGFR2 ; Senescence

刊名：Biomedicine & Pharmacotherapy

出版年：2015

9.Discovery of wrightiadione as a novel template for the TrkA kinase inhibitors

作者：Yujeong Jeong^a ; ^b ; Sang Min Lim^a ; Sungwoo Hong^a ; ^b ; ^{hongorg@kaist.ac.kr" class="auth_mail" title="E-mail the corresponding author}

关键词：Kinase ; Trk inhibitor ; Wrightiadione ; Modeling ; Anticancer

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2015

10.PLK1-inhibition can cause radiosensitization or radioresistance dependent on the treatment schedule

作者：Christin Lund-Andersen ; Sebastian Patzke ; Viola Nä ; hse-Kumpf ; Randi G. Syljuå ; sen ; ^{randi.syljuasen@rr-research.no" class="auth_mail}

关键词：PLK1-inhibitors ; G2 checkpoint ; Mitosis ; DNA damage ; Ionizing radiation ; Cancer ; Combined treatment

刊名：Radiotherapy and Oncology

出版年：February, 2014

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