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CNKI学位论文(184)
CNKI期刊论文0611(1)
知网期刊论文(150)
在“
Elsevier电子期刊
”中,
命中:
11
条,耗时:小于0.01 秒
在所有数据库中总计命中:
339
条
1.
The application of phosphoramidate ProTide technology to the potent anti-HCV compound 4′-azidocytidine (
R1479
)
作者:
Christopher McGuigan
;
Mary Rose Kelleher
;
Plinio Perrone
;
Sinead Mulready
;
Giovanna Luoni
;
Felice Daverio
;
Sonal Rajyaguru
;
Sophie Le Pogam
;
Isabel Najera
;
Joseph A. Martin
;
Klaus Klumpp
;
David B. Smi
关键词:
HCV
;
Antiviral
;
R1479
;
ProTide
;
4′
;
-Azidocytidine
;
Prodrug
;
Nucleotide
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
2.
Design, synthesis, and antiviral properties of 4′-substituted ribonucleosides as inhibitors of hepatitis C virus replication: The discovery of
R1479
作者:
David B. Smith
;
Joseph A. Martin
;
Klaus Klumpp
;
Stewart J. Baker
;
Peter A. Blomgren
;
Rene Devos
;
Caroline Granycome
;
Julie Hang
;
Christopher J. Hobbs
;
Wen-Rong Jiang
;
et al.
关键词:
Hepatitis C
;
HCV
;
R1479
;
Antiviral
;
Nucleoside
;
Ribonucleoside
;
Replicon
;
NS5B
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2007
3.
In vitro selected Con1 subgenomic replicons resistant to 2′-C-Methyl-Cytidine or to
R1479
show lack of cross resistance
作者:
Sophie Le Pogam
;
Wen-Rong Jiang
;
Vincent Leveque
;
Sonal Rajyaguru
;
Han Ma
;
Hyunsoon Kang
;
Sharon Jiang
;
Margaret Singer
;
Samir Ali
;
Klaus Klumpp
et al.
刊名:Virology
出版年:2006
4.
851 ANTIVIRAL POTENCY OF
R1479
, ACTIVE COMPOUND DERIVED IN VIVO FROM PRODRUG R1626, DEMONSTRATED ACROSS HCV GENOTYPES 1-6 IN NS5B RECOMBINANT ENZYMES AND HCV REPLICONS
作者:
V. Leveque
;
S. Le Pogam
;
H. Kang
;
G. Ao-Ieong
;
A. Kosaka
;
A. Seshaadri
;
J. Symons
;
N. Cammack
;
K. Klumpp
;
I. Najera
刊名:Journal of Hepatology
出版年:2008
5.
[603]
R1479
, A NOVEL NUCLEOSIDE ANALOG AND POTENT INHIBITOR OF HCV REPLICATION, DOES NOT AFFECT RIBAVIRIN-INDUCED HEMOLYSIS AND ERYTHROCYTE FRAGILITY IN VITRO
作者:
W.R. Jiang
;
J. Symons
;
N. Cammack
;
K. Klumpp
刊名:Journal of Hepatology
出版年:2007
6.
[439] ADDITIVE TO SYNERGISTIC ANTIVIRAL EFFECTS OF AN NS3/4A PROTEASE INHIBITOR (ITMN-191) AND AN NS5B RNA-DEPENDENT RNA POLYMERASE INHIBITOR (
R1479
) IN AN HCV REPLICON SYSTEM
作者:
S.D. Seiwert
;
H. Tan
;
L.M. Blatt
刊名:Journal of Hepatology
出版年:2007
7.
[790] IN VITRO RESISTANCE SELECTION TO THE HCV NUCLEOSIDE POLYMERASE INHIBITOR
R1479
AND TO THE PROTEASE INHIBITOR VX-950
作者:
M. McCown
;
S. Rajyaguru
;
J. Symons
;
N. Cammack
;
I. Naiera
刊名:Journal of Hepatology
出版年:2007
8.
[622]
R1479
, A NOVEL HEPATITIS C POLYMERASE INHIBITOR: LACK OF PRE-EXISTING RESISTANCE MUTATION SUPPORTS THE OBSERVED IN VIVO HIGH BARRIER TO RESISTANCE
作者:
S. Le Pogam
;
A. Kosaka
;
S. Hu
;
H. Kang
;
A. Seshaadri
;
J. Symons
;
K. Klumpp
;
N. Cammack
;
I. Najera
刊名:Journal of Hepatology
出版年:2007
9.
Design and Characterization of R1626, A Prodrug of the HCV Replication Inhibitor
R1479
(4′-Azidocytidine) With Enhanced Oral Bioavailability
作者:
Klaus Klumpp
;
David Smith
;
Michael Br
l ;
Tom Alfredson
;
Keshab Sarma
;
Mark Smith
;
Isabel Najera
;
Wen-Rong Jiang
;
Sophie Le Pogam
;
Vincent Leveque
;
et al.
刊名:Antiviral Research
出版年:2007
10.
Biodistribution of [
18
f] S
R14
4385 and [
18
f] SR
1479
63: selective radioligands for positron emission tomographic studies of brain cannabinoid receptors
作者:
Mathews
;
William B.
;
Scheffel
;
Ursula
;
Finley
;
Paige
;
Ravert
;
Hayden T.
;
Frank
;
Richard A.
;
et. al.
关键词:
Cannabinoid antagonist
;
Fluorine-18
;
Mice
;
PET
刊名:Nuclear Medicine and Biology
出版年:2000
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