设为首页
收藏本站
网站地图
|
English
|
公务邮箱
About the library
Background
History
Leadership
Organization
Readers' Guide
Opening Hours
Collections
Help Via Email
Publications
Electronic Information Resources
常用资源
电子图书
期刊论文
学位会议
外文资源
特色专题
内部出版物
CNKI学位论文(25)
知网期刊论文(3)
在“
Elsevier电子期刊
”中,
命中:
31
条,耗时:小于0.01 秒
在所有数据库中总计命中:
28
条
1.
A western blot assay to
m
easure cyclin dependent kinase activity in cells or in vitro without the use of radioisotopes
作者:
Cody W. Lewis
;
Ryan G. Taylor
;
Philip
M
. Kubara
;
Kris
M
arshall
;
Laurent
M
eijer
;
Roy
M
.
Golsteyn
关键词:
Cdk1
;
cyclin dependent kinase 1
;
Cdk2
;
cyclin dependent kinase 2
;
CPT
;
ca
m
ptothecin
;
D
M
SO
;
di
m
ethyl sulfoxide
;
DTT
;
dithiothreitol
;
EGTA
;
ethyleneglycol-bis (beta-a
m
inoethylether)- N
;
N&pri
m
e
;
-tetraacetic acid
;
HEPES
;
4-(2-hydroxyethyl)-1-piperazineethanes
刊名:FEBS Letters
出版年:2013
2.
An unusual DNA binding co
m
pound, S23906, induces
m
itotic catastrophe in cultured hu
m
an cells
作者:
Nathalie Cahuzac
;
Auré
;
lie Studé
;
ny
;
Kris
M
arshall
;
Isabella Versteege
;
Kate Wetenhall
;
Bruno Pfeiffer
;
Sté
;
phane Lé
;
once
;
John A. Hick
m
an
;
Alain Pierré
;
Roy
M
.
Golsteyn
关键词:
Cytotoxic drug
;
Cyclin-dependent kinases
;
Cdk1
;
DNA da
m
age response
;
Checkpoint kinase 1
;
Histone γ
;
-H2AX
;
Checkpoint adaptation
刊名:Cancer Letters
出版年:2010
3.
Synthesis and CHK1 inhibitory potency of Hy
m
enialdisine analogues
作者:
Jean-Gilles Par
m
entier
;
Bernard Portevin
;
Roy
M
.
Golsteyn
;
Alain Pierré
;
John Hick
m
an
;
Philippe Gloanec
;
Guillau
m
e De Nanteuil
关键词:
Hy
m
enialdisine
;
CHK1 inhibitor
刊名:Bioorganic and
M
edicinal Che
m
istry Letters
出版年:2009
4.
A three-step synthesis fro
m
rebecca
m
ycin of an efficient checkpoint kinase 1 inhibitor
作者:
Fabrice Anizon
;
Roy
M
.
Golsteyn
;
Sté
;
phane Lé
;
once
;
Bruno Pfeiffer
;
M
ichelle Prudho
mm
e
关键词:
Rebecca
m
ycin
;
Staurosporine
;
Antitu
m
or agents
;
Indolocarbazoles
;
Chk1 inhibitors
刊名:European Journal of
M
edicinal Che
m
istry
出版年:2009
5.
Novel 5-azaindolocarbazoles as cytotoxic agents and Chk1 inhibitors
作者:
M
yria
m
Lefoix
;
Gé
;
rard Coudert
;
Sylvain Routier
;
Bruno Pfeiffer
;
Daniel-Henri Caignard
;
John Hick
m
an
;
Alain Pierré
;
Roy
M
.
Golsteyn
;
Sté
;
phane Lé
;
once
;
Cé
;
line Bossard
;
Jean-Yves
关键词:
5-Azaindole
;
5-Azaindolocarbazole
;
Chk1 inhibitors
;
Cytoxicity
刊名:Bioorganic and
M
edicinal Che
m
istry
出版年:2008
6.
Synthesis, checkpoint kinase 1 inhibitory properties and in vitro antiproliferative activities of new pyrrolocarbazoles
作者:
Elisabeth Conchon
;
Fabrice Anizon
;
Bettina Aboab
;
Roy
M
.
Golsteyn
;
Sté
;
phane Lé
;
once
;
Bruno Pfeiffer
;
M
ichelle Prudho
mm
e
关键词:
Granulati
m
ide
;
Pyrrolo[3
;
4-
c
]carbazoles
;
Antitu
m
or agents
;
Chk1 inhibitors
刊名:Bioorganic and
M
edicinal Che
m
istry
出版年:2008
7.
Synthesis, in vitro antiproliferative activities, and Chk1 inhibitory properties of pyrrolo[3,4-a]carbazole-1,3-diones, pyrrolo[3,4-c]carbazole-1,3-diones, and 2-a
m
inopyridazino[3,4-a]pyrrolo[3,4-c]carbazole-1,3,4,7-tetraone
作者:
Elisabeth Conchon
;
Fabrice Anizon
;
Bettina Aboab
;
Roy
M
.
Golsteyn
;
Sté
;
phane Lé
;
once
;
Bruno Pfeiffer
;
M
ichelle Prudho
mm
e
关键词:
Pyrrolo[3
;
4-
a
]carbazole-1
;
3-diones
;
2-A
m
ino-pyridazino[3
;
4-
a
]pyrrolo[3
;
4-
c
]carbazole-1
34 ;
7-tetraone
;
Antitu
m
or agents
;
Chk1 inhibitors
刊名:European Journal of
M
edicinal Che
m
istry
出版年:2008
8.
Bis-i
m
ide granulati
m
ide analogues as potent Checkpoint 1 kinase inhibitors
作者:
Hé
;
lè
;
ne Hé
;
non
;
Sa
m
ir Messaoudi
;
Fabrice Anizon
;
Bettina Aboab
;
Nathalie Kucharczyk
;
Sté
;
phane Lé
;
once
;
Roy
M
.
Golsteyn
;
Bruno Pfeiffer
;
M
ichelle Prudho
mm
e
关键词:
Granulati
m
ide
;
Isogranulati
m
ide
;
Antitu
m
or agent
;
Chk1 inhibitor
刊名:European Journal of Phar
m
acology
出版年:2007
9.
Synthesis and biological activities of isogranulati
m
ide analogues
作者:
Bernadette Hugon
;
Fabrice Anizon
;
Christian Bailly
;
Roy
M
.
Golsteyn
;
Alain Pierré
;
Sté
;
phane Lé
;
once
;
John Hick
m
an
;
Bruno Pfeiffer
;
M
ichelle Prudho
mm
e
关键词:
Isogranulati
m
ide
;
Chk1 inhibitors
;
Pyrrolo[3
;
4-
c
]carbazole
;
Antitu
m
or drugs
刊名:Bioorganic and
M
edicinal Che
m
istry
出版年:2007
10.
Phosphorylation of CDC25C at S263 controls its intracellular localisation
作者:
Charlotte Es
m
enjaud-Mailhat
;
Valé
;
rie Lobjois
;
Carine Fro
m
ent
;
Roy
M
.
Golsteyn
;
Bernard
M
onsarrat
;
Bernard Duco
mm
un
关键词:
CDC25C
;
Phosphorylation
;
M
itosis
;
Cell cycle
刊名:FEBS Letters
出版年:2007
1
2
3
4
按检索点细分(31)
作者(31)
按出版年细分(31)
2013年(1)
2010年(1)
2009年(2)
2008年(3)
2007年(3)
2006年(4)
2005年(2)
2004年(3)
2003年(2)
2001年(4)
2000年(3)
2000年及以前(3)
NGLC 2004-2010.National Geological Library of China All Rights Reserved.
Add:29 Xueyuan Rd,Haidian District,Beijing,PRC. Mail Add: 8324 mailbox 100083
For exchange or info please contact us via
email
.