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内部出版物
知网期刊论文(1)
在“
Elsevier电子期刊
”中,
命中:
7
条,耗时:小于0.01 秒
在所有数据库中总计命中:
1
条
1.
Discovery of N-[5-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-b]pyridazin-6-yl}oxy)-2-methylphenyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide (TAK-593), a highly potent VEGFR2 kinase inhibitor
作者:
Naoki Miyamoto
;
Nozomu Sakai
;
Takaharu Hirayama
;
Kazuhiro Miwa
;
Yuya Oguro
;
Hideyuki Oki
;
Kengo Okada
;
Terufumi
Takagi
;
Hidehisa Iwata
;
Yoshiko Awazu
;
Seiji Yamasaki
;
Toshiyuki Takeuchi
;
Hiroshi Miki
;
Akira Hori
;
Shinichi Imamura
;
shin-ichi.imamura@takeda.com
关键词:
DZFZXPPHBWCXPQ-UHFFFAOYSA-N
刊名:Bioorganic and Medicinal Chemistry
出版年:2013
2.
Design, synthesis, and evaluation of imidazo[1,2-b]pyridazine derivatives having a benzamide unit as novel VEGFR2 kinase inhibitors
作者:
Naoki Miyamoto
;
Yuya Oguro
;
Terufumi
Takagi
;
Hidehisa Iwata
;
Hiroshi Miki
;
Akira Hori
;
Shinichi Imamura
;
shin-ichi.imamura@takeda.com
关键词:
BRFOGQVFBWDQGX-UHFFFAOYSA-N
刊名:Bioorganic and Medicinal Chemistry
出版年:2012
3.
Design and synthesis of novel DFG-out RAF/vascular endothelial growth factor receptor 2 (VEGFR2) inhibitors: 3. Evaluation of 5-amino-linked thiazolo[5,4-d]pyrimidine and thiazolo[5,4-b]pyridine derivatives
作者:
Masaaki Hirose
;
Masanori Okaniwa
;
Tohru Miyazaki
;
Takashi Imada
;
Tomohiro Ohashi
;
Yuta Tanaka
;
Takeo Arita
;
Masato Yabuki
;
Tomohiro Kawamoto
;
Shunichirou Tsutsumi
;
Akihiko Sumita
;
Terufumi
Takagi
;
Bi-Ching Sang
;
Jason Yano
;
Kathleen Aertgeerts
;
Sei Yoshida
;
Tomoyasu Ishikawa
关键词:
BSBQPLUISHJULY-UHFFFAOYSA-N
刊名:Bioorganic and Medicinal Chemistry
出版年:2012
4.
Design and synthesis of novel DFG-out RAF/vascular endothelial growth factor receptor 2 (VEGFR2) inhibitors: 2. Synthesis and characterization of a novel imide-type prodrug for improving oral absorption
作者:
Masanori Okaniwa
;
Takashi Imada
;
Tomohiro Ohashi
;
Tohru Miyazaki
;
Takeo Arita
;
Masato Yabuki
;
Akihiko Sumita
;
Shunichirou Tsutsumi
;
Keiko Higashikawa
;
Terufumi
Takagi
;
Tomohiro Kawamoto
;
Yoshitaka Inui
;
Sei Yoshida
;
Tomoyasu Ishikawa
关键词:
MDPMAXSABUPRJI-UHFFFAOYSA-N
;
BFDNRMPCCWFLHE-UHFFFAOYSA-N
;
JUQXULZEMQJOCI-UHFFFAOYSA-N
刊名:Bioorganic and Medicinal Chemistry
出版年:2012
5.
N-Phenyl-N′-[4-(5H-pyrrolo[3,2-d]pyrimidin-4-yloxy)phenyl]ureas as novel inhibitors of VEGFR and FGFR kinases
作者:
Yuya Oguro
;
Naoki Miyamoto
;
Terufumi
Takagi
;
Kengo Okada
;
Yoshiko Awazu
;
Hiroshi Miki
;
Akira Hori
;
Keiji Kamiyama
;
Shinichi Imamura
关键词:
VEGFR
;
FGFR
;
Pyrrolo[3
;
2-
d
]pyrimidine
;
Urea
刊名:Bioorganic and Medicinal Chemistry
出版年:2010
6.
Design, synthesis, and evaluation of 5-methyl-4-phenoxy-5H-pyrrolo[3,2-d]pyrimidine derivatives: Novel VEGFR2 kinase inhibitors binding to inactive kinase conformation
作者:
Yuya Oguro
;
Naoki Miyamoto
;
Kengo Okada
;
Terufumi
Takagi
;
Hidehisa Iwata
;
Yoshiko Awazu
;
Hiroshi Miki
;
Akira Hori
;
Keiji Kamiyama
;
Shinichi Imamura
关键词:
VEGFR
;
Type-II inhibitor
;
Pyrrolo[3
;
2-
d
]pyrimidine
;
diphenylurea
刊名:Bioorganic and Medicinal Chemistry
出版年:2010
7.
Synthesis and biological evaluation of the metabolites of 2-(1-{3-[(6-chloronaphthalen-2-yl)sulfonyl]propanoyl}piperidin-4-yl)-5-methyl-1,2-dihydro-3H-imidazo[1,5-c]imidazol-3-one
作者:
Takuya Fujimoto
;
Mamoru Tobisu
;
Noriko Konishi
;
Masaki Kawamura
;
Norio Tada
;
Terufumi
Takagi
;
Keiji Kubo
关键词:
Factor Xa inhibitor
;
Antithrombotic agent
;
Active metabolite
刊名:Bioorganic and Medicinal Chemistry
出版年:2009
1
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