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在“Elsevier电子期刊”中，命中：465条，耗时：0.0149926 秒

在所有数据库中总计命中：958条

1.Synthesis, structure and properties of N-aminosaccharin - A selective inhibitor of human carbonic anhydrase I

作者：Mikhail A. Kuznetsov^a ; ^{m.kuznetsov@spbu.ru} ; Aleksandr N. Shestakov^a ; Mikhail Zibinsky^a ; Mikhail Krasavin^a ; Claudiu T. Supuran^b ; Stanislav Kalinin^a ; Muhammet Tanç ; ^b

关键词：N-Aminosaccharin ; N-Amination ; hCA I inhibitor ; Oxidative aminoaziridination ; Ligand efficiency

刊名：Tetrahedron Letters

出版年：2017

2.Sulfonamide inhibition profile of the γ-carbonic anhydrase identified in the genome of the pathogenic bacterium Burkholderia pseudomallei the etiological agent responsible of melioidosis

作者：Sonia Del Prete^a ; Daniela Vullo^b ; Pietro Di Fonzo^a ; Sameh M. Osman^c ; Zeid AlOthman^c ; William A. Donald^d ; Claudiu T. Supuran^c ; ^d ; ^e ; ^{claudiu.supuran@unifi.it} ; Clemente Capasso^a ; ^{clemente.capasso@ibbr.cnr.it}

关键词：Carbonic anhydrase ; γ-Class ; Inhibitor ; Sulfonamide ; Sulfamate ; Acetazolamide ; Drug resistance ; Burkholderia pseudomallei

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

3.Dithiocarbamates effectively inhibit the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa

作者：Daniela Vullo^a ; Sonia Del Prete^b ; ^c ; Alessio Nocentini^b ; Sameh M. Osman^d ; Zeid AlOthman^d ; Clemente Capasso^c ; Murat Bozdag^a ; Fabrizio Carta^b ; Paola Gratteri^e ; Claudiu T. Supuran^b ; ^d ; ^{claudiu.supuran@unifi.it}

关键词：Carbonic anhydrase ; β-CA-class enzyme ; Dithiocarbamate ; Inhibitor ; Malassezia globosa

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

4.5-Substituted-benzylsulfanyl-thiophene-2-sulfonamides with effective carbonic anhydrase inhibitory activity: Solution and crystallographic investigations

作者：Jekaterīna Ivanova^a ; ^b ; Agnese Balode^a ; ^b ; Raivis Žalubovskis^a ; ^{raivis@osi.lv} ; Janis Leitans^c ; Andris Kazaks^c ; Daniela Vullo^d ; Kaspars Tars^c ; ^e ; Claudiu T. Supuran^f ; ^{claudiu.supuran@unifi.it}

关键词：Carbonic anhydrase ; Thiophene-2-sulfonamide ; Mercaptan ; Inhibitor

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

5.Novel eugenol derivatives: Potent acetylcholinesterase and carbonic anhydrase inhibitors

作者：Fevzi Topal^a ; Ilhami Gulcin^b ; ^c ; ^{igulcin@atauni.edu.tr} ; ^{igulcin@yahoo.com} ; Arif Dastan^b ; Murat Guney^d

关键词：Eugenol ; Carbonic anhydrase ; Acetylcholinesterase ; Enzyme purification ; Enzyme inhibition

刊名：International Journal of Biological Macromolecules

出版年：2017

6.Substituted (E)-2-(2-benzylidenehydrazinyl)-4-methylthiazole-5-carboxylates as dual inhibitors of 15-lipoxygenase & carbonic anhydrase II: synthesis, biochemical evaluation and docking studies

作者：Aamer Saeed^a ; ^{aamersaeed@yahoo.com} ; Shafi Ullah Khan^b ; Parvez Ali Mahesar^a ; Pervaiz Ali Channar^a ; Ghulam Shabir^a ; Jamshed Iqbal^b ; ^{drjamshed@ciit.net.pk}

关键词：Thiazoles ; 15-Lipoxygenase ; Bovine carbonic anhydrase II ; Docking studies

刊名：Biochemical and Biophysical Research Communications

出版年：2017

7.Anion inhibition profiles of the γ-carbonic anhydrase from the pathogenic bacterium Burkholderia pseudomallei responsible of melioidosis and highly drug resistant to common antibiotics

作者：Sonia Del Prete^a ; ^b ; Daniela Vullo^b ; Pietro Di Fonzo^a ; Sameh M. Osman^c ; Zeid AlOthman^c ; Claudiu T. Supuran^c ; ^d ; ^{claudiu.supuran@unifi.it} ; Clemente Capasso^a ; ^{clemente.capasso@ibbr.cnr.it}

关键词：Carbonic anhydrase ; Metalloenzymes ; γ-Class ; Inhibitor ; Anion ; Burkholderia pseudomallei

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

8.Carbonic anhydrase inhibition boosts the antitumor effects of Imatinib mesylate via potentiating the antiangiogenic and antimetastatic machineries

作者：Amal A. Abd-El Fattah^a ; Hebatallah A. Darwish^a ; ^b ; Nevine Fathy^a ; ^{nevine.abdallah@pharma.cu.edu.eg} ; Samia A. Shouman^c

关键词：AZ ; acetazolamide ; IM ; imatinib ; EAC ; Ehrlich ascites carcinoma ; PDGF-A ; platelet derived growth factor-A ; TSP-1 ; thrombospondin-1 ; VEGF ; vascular endothelial growth factor ; NO ; nitric oxide ; MMP ; matrix metalloproteinase ; MAPK ; mitogen activated protein kinase ; TIMP ; tissue inhibitor of metalloproteinase ; MVD ; microvessel density

刊名：Toxicology and Applied Pharmacology

出版年：2017

9.New approach of delivering cytotoxic drugs towards CAIX expressing cells: A concept of dual-target drugs

作者：Simon J.A. van Kuijk^a ; ¹ ; ^{s.vankuijk@maastrichtuniversity.nl} ; Nanda Kumar Parvathaneni^a ; ^b ; ¹ ; ^{nanda-kumar.parvathaneni@etu.umontpellier.fr} ; Raymon Niemans^a ; ¹ ; Marike W. van Gisbergen^a ; ¹ ; Fabrizio Carta^c ; Daniela Vullo^d ; Silvia Pastorekova^e ; Ala Yaromina^a ; Claudiu T. Supuran^c ; Ludwig J. Dubois^a ; ² ; Jean-Yves Winum^b ; ² ; Philippe Lambin^a ; ²

关键词：Tumor ; Hypoxia ; Carbonic anhydrase IX ; Dual-target drugs ; CAIX inhibitors ; Cytotoxic drugs

刊名：European Journal of Medicinal Chemistry

出版年：2017

10.Design and synthesis of a novel class of carbonic anhydrase-IX inhibitor 1-(3-(phenyl/4-fluorophenyl)-7-imino-3H-[1,2,3]triazolo[4,5d]pyrimidin 6(7H)yl)urea

作者：Shikha Kumari^a ; ¹ ; Danish Idrees^b ; ¹ ; Chandra Bhushan Mishra^a ; ¹ ; Amresh Prakash^b ; ¹ ; Wahiduzzaman^b ; Faizan Ahmad^b ; Md. Imtaiyaz Hassan^b ; ^{mihassan@jmi.ac.in" class="auth_mail" title="E-mail the corresponding author} ; Manisha Tiwari^a ; ^{mtiwari07@gmail.com" class="auth_mail" title="E-mail the corresponding author}

关键词：Hypoxia-induced cancer ; Carbonic anhydrase IX inhibitor ; Drug design and discovery ; Triazolo-pyrimidine urea ; MD simulation

刊名：Journal of Molecular Graphics and Modelling

出版年：2016

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