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Springer电子图书(9)
CNKI会议论文(23)
CNKI学位论文(21306)
CNKI期刊论文0611(10)
知网期刊论文(10082)
在“
Elsevier电子期刊
”中,
命中:
10,929
条,耗时:0.0539749 秒
在所有数据库中总计命中:
31,430
条
1.
Design, synthesis and analgesic/anti-inflammatory evaluation of novel diarylthiazole and diarylimidazole derivatives towards
selective
COX-1
inhibitors
with better gastric profile
作者:
Ahmed H. Abdelazeem
a
;
b
;
ahmed.abdelazeem@pharm.bsu.edu.eg
;
ahmed.pharm@yahoo.com
;
Mohammed T. El-Saadi
a
;
Asmaa G. Safi El-Din
a
;
Hany A. Omar
c
;
d
;
Samir M. El-Moghazy
e
;
samirelmoghazy@gmail.com
关键词:
Selective
COX-1
;
Mofezolac
;
Diarylthiazole
;
Diarylimidazole
;
Analgesic
;
Anti-inflammatory
;
Ulcerogenicity
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
2.
Selective
Serotonin Reuptake
Inhibitors
and Poststroke Epilepsy: A Population-Based Nationwide Study
作者:
Chien-Chen Chou
;
MD
a
;
b
;
Der-Jen Yen
;
MD
a
;
b
;
Yung-Yang Lin
;
MD
;
PhD
a
;
c
;
d
;
Yu-Chiao Wang
;
MSc
e
;
g
;
Cheng-Li Lin
;
MSc
e
;
g
;
Chia-Hung Kao
;
MD
f
;
h
;
i
;
d10040@mail.cmuh.org.tw
关键词:
aHR
;
adjusted hazard ratio
;
DDD
;
defined daily dose
;
HR
;
hazard ratio
;
ICD-9-CM
;
International Classification of Diseases
;
Ninth Revision
;
Clinical Modification
;
IQR
;
interquartile range
;
LHID2000
;
Longitudinal Health Insurance Database 2000
;
NHI
;
National Health Insurance
;
NHIRD
;
National Health Insurance Research Database
;
PY
;
person-year
;
SSRI
;
selective
serotonin reuptake inhibitor
刊名:Mayo Clinic Proceedings
出版年:2017
3.
Crystal structures, binding interactions, and ADME evaluation of brain penetrant N-substituted indazole-5-carboxamides as subnanomolar,
selective
monoamine oxidase B and dual MAO-A/B
inhibitors
作者:
Nikolay T. Tzvetkov
a
;
ntzvetkov@ntzlab.com
;
Hans-Georg Stammler
b
;
Beate Neumann
b
;
Silvia Hristova
c
;
Liudmil Antonov
c
;
Marcus Gastreich
d
关键词:
ADME
;
MAO
inhibitors
;
Molecular modeling
;
Indazole-5-carboxamides
;
Parkinson's disease
;
X-ray
刊名:European Journal of Medicinal Chemistry
出版年:2017
4.
Discovery of triazole aminopyrazines as a highly potent and
selective
series of PI3Kδ
inhibitors
作者:
Ina Terstiege
a
;
Ina.Terstiege@astrazeneca.com
;
Matthew Perry
a
;
Jens Petersen
b
;
Christian Tyrchan
a
;
Tor Svensson
a
;
Helena Lindmark
b
;
Linda Ö
;
ster
b
关键词:
Phosphoinositide 3-kinase
;
PI3Kδ inhibitor
;
Aminopyrazine
;
Inflammation
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
5.
In silico receptor-based drug design of X,Y-benzenesulfonamide derivatives as
selective
COX-2
inhibitors
作者:
David J. Pé
;
rez
a
;
Orlando Sarabia
a
;
Manuel Villanueva-Garcí
;
a
b
;
Kayim Pineda-Urbina
a
;
Á
;
ngel Ramos-Organillo
a
;
Jorge Gonzalez-Gonzalez
a
;
Zeferino Gó
;
mez-Sandoval
a
;
zgomez@ucol.com
;
Rodrigo Said Razo-Herná
;
ndez
a
;
c
;
rrazo@ucol.mx
关键词:
QSAR
;
Docking
;
Cyclooxygenase
;
Benzenesulfonamides
;
Drug design
;
Artificial neural networks
刊名:Comptes Rendus Chimie
出版年:2017
6.
2-Oxoamides based on dipeptides as
selective
calcium-independent phospholipase A
2
inhibitors
作者:
Anneta Smyrniotou
a
;
Maroula G. Kokotou
b
;
c
;
Varnavas D. Mouchlis
c
;
Efrosini Barbayianni
b
;
George Kokotos
b
;
Edward A. Dennis
c
;
edennis@ucsd.edu
;
Violetta Constantinou-Kokotou
a
;
vikon@aua.gr
关键词:
Dipeptides
;
Inhibitors
;
Oxoamides
;
Phospholipase A2
;
Pseudodipeptides
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
7.
Discovery of novel 3-hydroxypicolinamides as
selective
inhibitors
of HIV-1 integrase-LEDGF/p75 interaction
作者:
Feng-Hua Zhang
a
;
Bikash Debnath
b
;
Zhong-Liang Xu
a
;
Liu-Meng Yang
c
;
Li-Rui Song
a
;
Yong-Tang Zheng
c
;
Nouri Neamati
b
;
neamati@umich.edu
;
Ya-Qiu Long
a
;
yqlong@simm.ac.cn
关键词:
HIV-1 integrase
;
Allosteric inhibitor
;
LEDGF/p75
;
Dimerization
;
3-Hydroxypicolinamide
刊名:European Journal of Medicinal Chemistry
出版年:2017
8.
Strategy for designing
selective
α-l-rhamnosidase
inhibitors
: Synthesis and biological evaluation of l-DMDP cyclic isothioureas
作者:
Shota Miyawaki
a
;
Yuki Hirokami
a
;
Kyoko Kinami
a
;
Masako Hoshino
a
;
Daisuke Minehira
a
;
Daiki Miyamoto
b
;
Robert J. Nash
c
;
George W.J. Fleet
d
;
Isao Adachi
a
;
Naoki Toyooka
b
;
Atsushi Kato
a
;
关键词:
α-l-Rhamnosidase
;
l-DMDP cyclic isothiourea
;
Iminosugars
;
Structure&ndash
;
activity relationships
;
Glycosidase inhibitor
;
Mycobacterium tuberculosis
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
9.
Selective
Substrates and
Inhibitors
for Kallikrein-Related Peptidase 7 (KLK7) Shed Light on KLK Proteolytic Activity in the Stratum Corneum
作者:
Simon J. de Veer
1
;
2
;
3
;
Laetitia Furio
2
;
3
;
Joakim E. Swedberg
4
;
Christopher A. Munro
1
;
Maria Brattsand
5
;
Judith A. Clements
1
;
6
;
Alain Hovnanian
2
;
3
;
7
;
Jonathan M. Harris
1
;
j2.harris@qut.edu.au
关键词:
AD
;
atopic dermatitis
;
KLK
;
kallikrein-related peptidase
;
LEKTI
;
lymphoepithelial Kazal-type-related inhibitor
;
NS
;
Netherton syndrome
;
pNA
;
para-nitroanilide
;
SFTI-1
;
sunflower trypsin inhibitor-1
;
SPINK
;
serine protease inhibitor Kazal-type
刊名:Journal of Investigative Dermatology
出版年:2017
10.
Multitarget drug design strategy against Alzheimer’s disease: Homoisoflavonoid Mannich base derivatives serve as acetylcholinesterase and monoamine oxidase B dual
inhibitors
with multifunctional properties
作者:
Yan Li
a
;
Xiaoming Qiang
a
;
Li Luo
a
;
Xia Yang
a
;
Ganyuan Xiao
a
;
Yunxiaozhu Zheng
a
;
Zhongcheng Cao
a
;
Zhipei Sang
b
;
Fu Su
a
;
sufu@scu.edu.cn
;
Yong Deng
a
;
dengyong@scu.edu.cn
关键词:
Alzheimer&rsquo
;
s disease
;
Homoisoflavonoid
;
Mannich base derivatives
;
Acetylcholinesterase
inhibitors
;
Monoamine oxidase B
inhibitors
;
Multifunctional properties
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
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