设为首页
收藏本站
网站地图
|
English
|
公务邮箱
About the library
Background
History
Leadership
Organization
Readers' Guide
Opening Hours
Collections
Help Via Email
Publications
Electronic Information Resources
常用资源
电子图书
期刊论文
学位会议
外文资源
特色专题
内部出版物
Springer电子图书(1)
CNKI学位论文(7)
知网期刊论文(4)
在“
Elsevier电子期刊
”中,
命中:
10
条,耗时:小于0.01 秒
在所有数据库中总计命中:
12
条
1.
4-Aminoquinoline derivatives: Synthesis, in vitro and in vivo antiplasmodial activity against chloroquine-resistant parasites
作者:
Shailja Singh
a
;
Drishti Agarwal
a
;
c
;
Kumkum Sharma
a
;
Manish Sharma
a
;
Morten A. Nielsen
b
;
Michael Alifrangis
b
;
Ashok K. Singh
d
;
Rinkoo D. Gupta
c
;
Satish K. Awasthi
a
;
satishpna@gmail.com" class="auth_mail" title="E-mail the corresponding author
;
skawasthi@chemistry.du.ac.in" class="auth_mail" title="E-mail the corresponding author
关键词:
Antimalarial
;
Amodiaquine
;
Chloroquine
;
4-Aminoquinoline
analogues
;
Plasmodium falciparum
;
Plasmodium berghei
刊名:European Journal of Medicinal Chemistry
出版年:2016
2.
Benzoheterocyclic
amodiaquine
analogues
with potent antiplasmodial activity: Synthesis and pharmacological evaluation
作者:
Dennis S.B. Ongarora
;
Jiri Gut
;
Philip J. Rosenthal
;
Collen M. Masimirembwa
;
Kelly Chibale
关键词:
Benzothiazole
;
Benzoxazole
;
Amodiaquine
;
Benzoheterocyclic
;
Antiplasmodial
;
Reactive metabolite
;
Quinone imine
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2012
3.
Amodiaquine
analogues
containing NO-donor substructures: Synthesis and their preliminary evaluation as potential tools in the treatment of cerebral malaria
作者:
Massimo Bertinaria
;
Stefano Guglielmo
;
Barbara Rol
o ;
Marta Giorgis
;
Cristina Aragno
;
Roberta Fruttero
;
Alberto Gasco
;
Silvia Parapini
;
Donatella Taramelli
;
Yuri C. Martins
;
Leonardo J.M. Carvalho
关键词:
Amodiaquine
;
Cerebral malaria
;
Nitric oxide
;
Furoxans
;
Nitrooxy derivatives
刊名:European Journal of Medicinal Chemistry
出版年:2011
4.
Hit identification of novel heparanase inhibitors by structure- and ligand-based approaches
作者:
Rafael Gozalbes
a
;
&dagger
;
;
&Dagger
;
;
rgozalbes@cipf.es
;
Silvia Mosulé
;
n
a
;
&Dagger
;
;
Leticia Ortí
;
a
;
Jesú
;
s Rodrí
;
guez-Dí
;
az
b
;
Rodrigo J. Carbajo
a
;
Patricia Melnyk
c
;
d
;
e
;
Antonio Pineda-Lucena
a
;
apineda@cipf.es
关键词:
Drug discovery
;
Heparanase
;
Computational chemistry
;
Biophysical experiments
;
Structure&ndash
;
activity relationships
刊名:Bioorganic and Medicinal Chemistry
出版年:2013
5.
A new series of
amodiaquine
analogues
modified in the basic side chain with in vitro antileishmanial and antiplasmodial activity
作者:
Stefano Guglielmo
;
Massimo Bertinaria
;
Barbara Rol
o ;
Marco Crosetti
;
Roberta Fruttero
;
Vanessa Yardley
;
Simon L. Croft
;
Alberto Gasco
关键词:
Amodiaquine
analogues
;
Leishmania donovani
;
Plasmodium falciparum
;
Antiprotozoals
刊名:European Journal of Medicinal Chemistry
出版年:2009
6.
Synthesis and antimalarial activity of new
analogues
of
amodiaquine
作者:S ;
rine Delarue-Cochin
;
Emilia Paunescu
;
Louis Maes
;
Elisabeth Mouray
;
Christian Sergheraert
;
Philippe Grellier
;
Patricia Melnyk
关键词:
Drug design
;
Plasmodium falciparum
;
Antimalarials
;
Amodiaquine
;
4-Aminoquinolines
刊名:European Journal of Medicinal Chemistry
出版年:2008
7.
Novel
amodiaquine
congeners as potent antimalarial agents
作者:
Manolo Casagr
e ;
Nicoletta Basilico
;
Silvia Parapini
;
Sergio Romeo
;
Donatella Taramelli
;
Anna Sparatore
关键词:
4-Aminoquinoline derivatives
;
Amodiaquine
analogues
;
Chloroquine
;
Antimalarial agents
刊名:Bioorganic and Medicinal Chemistry
出版年:2008
8.
The hydroxyl functionality and a rigid proximal N are required for forming a novel non-covalent quinine-heme complex
作者:
John N. Alumasa
a
;
Alexander P. Gorka
a
;
Leah B. Casabianca
d
;
1
;
Erica Comstock
e
;
1
;
Angel C. de Dios
a
;
c
;
Paul D. Roepe
a
;
b
;
c
;
roepep@georgetown.edu
关键词:
Hemozoin
;
Antimalarial drugs
;
Ferriprotoporphyrin IX
刊名:Journal of Inorganic Biochemistry
出版年:2011
9.
Suzuki–Miyaura cross-coupling reaction as the key step for the synthesis of some new 4′-aryl and alkyl substituted
analogues
of
amodiaquine
and amopyroquine
作者:
Emilia Paunescu
;
Nicolas Matuszak
;
Patricia Melnyk
关键词:
Indol-2-yl quinoline-2-one
;
Synthesis
;
5-
endo
-
dig
-Cyclization
;
KDR kinase inhibitor
刊名:Tetrahedron
出版年:2007
10.
The Role of Drug Accumulation in 4-Aminoquinoline Antimalarial Potency: The influence of structural substitution and physicochemical properties
作者:
Hawley
;
Shaun R.
;
Bray
;
Patrick G.
;
O'Neill
;
Paul M.
;
Park
;
B. Kevin
;
Ward
;
Stephen A.
关键词:
amodiaquine
;
4-aminoquinolines
;
Plasmodium falciparum
;
accumulation
;
activity
;
physicochemical properties
刊名:Biochemical Pharmacology
出版年:1996
1
按检索点细分(10)
题名(5)
关键词(3)
文摘(7)
按出版年细分(10)
2016年(1)
2013年(1)
2012年(1)
2011年(2)
2009年(1)
2008年(2)
2007年(1)
2000年及以前(1)
NGLC 2004-2010.National Geological Library of China All Rights Reserved.
Add:29 Xueyuan Rd,Haidian District,Beijing,PRC. Mail Add: 8324 mailbox 100083
For exchange or info please contact us via
email
.