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CNKI学位论文(38)
知网期刊论文(6)
在“
Elsevier电子期刊
”中,
命中:
9
条,耗时:小于0.01 秒
在所有数据库中总计命中:
44
条
1.
Strategy for designing selective α-l-rhamnosidase inhibitors: Synthesis and biological evaluation of l-DMDP
cyclic
isothiourea
s
作者:
Shota Miyawaki
a
;
Yuki Hirokami
a
;
Kyoko Kinami
a
;
Masako Hoshino
a
;
Daisuke Minehira
a
;
Daiki Miyamoto
b
;
Robert J. Nash
c
;
George W.J. Fleet
d
;
Isao Adachi
a
;
Naoki Toyooka
b
;
Atsushi Kato
a
;
关键词:
α-l-Rhamnosidase
;
l-DMDP
cyclic
isothiourea
;
Iminosugars
;
Structure&ndash
;
activity relationships
;
Glycosidase inhibitor
;
Mycobacterium tuberculosis
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
2.
Structure-activity relationship of dihydroimidazo-, dihydropyrimido, tetrahydrodiazepino-[2,1-b]-thiazoles, and -benzothiazoles as an acylation catalyst
作者:
Sentaro Okamoto
;
okamos10@kanagawa-u.ac.jp" class="auth_mail
;
Yuzo Sakai
;
Saki Watanabe
;
Shohei Nishi
;
Aya Yoneyama
;
Hitomi Katsumata
;
Yu Kosaki
;
Rumi Sato
;
Megumi Shiratori
;
Misuzu Shibuno
;
Tsukasa Shishido
关键词:
Cyclic
isothiourea
;
Acylation
;
Catalyst
;
Substitution effect
;
Kinetic resolution
刊名:Tetrahedron Letters
出版年:12 March, 2014
3.
Discovery and SAR of
cyclic
isothiourea
s as novel NPY Y
1
receptor antagonists
作者:
Zhong-Yue Sun
;
Zhaoning Zhu
;
Yuanzan Ye
;
Brian McKittrick
;
Michael Czarniecki
;
William Greenlee
;
Deborra Mullins
;
Mario Guzzi
关键词:
NPY Y
1
receptor antagonist
;
Thioisourea
;
Thiazoline
;
Thiazine
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
4.
High throughput synthesis of 2,3,6-trisubstituted-5,6-dihydroimidazo[2,1-b]thiazole derivatives
作者:
Yangmei Li
a
;
yli@tpims.org
;
Marc Giulianotti
a
;
Richard A. Houghten
;
a
;
houghten@tpims.org
刊名:Tetrahedron Letters
出版年:2011
5.
Corrigendum to “Discovery and SAR of
cyclic
isothiourea
s as novel NPY Y
1
receptor antagonists” [Bioorg. Med. Chem. Lett. 19 (2009) 6801]
作者:
Zhong-Yue Sun
;
Zhaoning Zhu
;
Yuanzan Ye
;
Brian McKittrick
;
Michael Czarniecki
;
William Greenlee
;
Deborra Mullins
;
Mario Guzzi
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
6.
Diastereoselective
isothiourea
iodocyclization for manzacidin synthesis
作者:
Woo
;
Jacqueline C.S.
;
MacKay
;
D. Bruce
刊名:Tetrahedron Letters
出版年:2003
7.
Synthesis of C
2
-Symmetric Bis(
Cyclic
Isothiourea
s) As Potent Inhibitors of Glycosidases
作者:
Gauzy
;
Laurence
;
Le Merrer
;
Yves
;
Depezay
;
Jean-Claude
;
Damour-Barbalat
;
Dominique
;
Mignani
;
Serge
关键词:
Glycosidase
;
Isothiourea
;
Thioformamide
;
Thiazolidinethione
;
Mercuric chloride
刊名:Tetrahedron Letters
出版年:1999
8.
Synthesis of C
2
-symmetric bis(
cyclic
isothiourea
s) as potent inhibitors of glycosidases
作者:
Gauzy
;
Laurence
;
Le Merrer
;
Yves
;
Depezay
;
Jean-Claude
;
Damour-Barbalat
;
Dominique
;
Mignani
;
Serge
关键词:
Glycosidase
;
Isothiourea
;
Thioformamide
;
Thiazolidinethione
;
Mercuric chloride
刊名:Tetrahedron Letters
出版年:1999
9.
A General Route to
Cyclic
Amidines and
Isothiourea
s Based on Formal Aza Diels Alder Reactions of Aminoheterocycles
作者:
Mellor
;
John M.
;
Rataj
;
Helen
刊名:Tetrahedron Letters
出版年:1996
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