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内部出版物
CNKI学位论文(2)
在“
Elsevier电子期刊
”中,
命中:
7
条,耗时:小于0.01 秒
在所有数据库中总计命中:
2
条
1.
Novel highly potent serotonin 5-HT
7
receptor ligands: Structural modifications to improve pharmacokinetic properties
作者:
Enza
Lacivita
;
Pantaleo Di Pilato
;
Madia Letizia Stama
;
Nicola Antonio Colabufo
;
Francesco Berardi
;
Roberto Perrone
;
Bianca De Filippis
;
Giovanni Laviola
;
Walter Adriani
;
Mauro Niso
;
Marcello Leopoldo
关键词:
5-HT7 receptors
;
Arylpiperazines
;
Serotonin
;
Microsomial S9 fraction
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2013
2.
LP-211 is a brain penetrant selective agonist for the serotonin 5-HT
7
receptor
作者:
Peter B. Hedlund
;
Marcello Leopoldo
;
Silvio Caccia
;
Gor Sarkisyan
;
Claudia Fracasso
;
Giuliana Martelli
;
Enza
Lacivita
;
Francesco Berardi
;
Roberto Perrone
关键词:
Serotonin 5-HT
7
receptor
;
Agonist
;
LP-211
;
RA-7
;
Brain distribution
;
Body temperature
刊名:Neuroscience Letters
出版年:2010
3.
Identification of a red-emitting fluorescent ligand for in vitro visualization of human serotonin 5-HT
1A
receptors
作者:
Enza
Lacivita
;
Anna Carmela Masotti
;
Md. Jafurulla
;
Roopali Saxena
;
N
;
ini Rangaraj
;
Amitabha Chattopadhyay
;
Nicola A. Colabufo
;
Francesco Berardi
;
Roberto Perrone
;
Marcello Leopoldo
关键词:
5-HT1A receptor
;
Fluorescence
;
SAR
;
1-Arylpiperazine
;
Confocal laser scanning microscopy
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
4.
Design, synthesis, and binding affinities of potential positron emission tomography (PET) ligands with optimal lipophilicity for brain imaging of the dopamine D
3
receptor. Part II
作者:
Marcello Leopoldo
;
Enza
Lacivita
;
Paola De Giorgio
;
Marialess
;
ra Contino
;
Francesco Berardi
;
Roberto Perrone
关键词:
D
3
receptors
;
Positron emission tomography
;
Structure–
;
affinity relationships
;
Arylpiperazine
;
Lipophilicity
刊名:Bioorganic and Medicinal Chemistry
出版年:2009
5.
Determination of 1-aryl-4-propylpiperazine pK
作者:
Enza
Lacivita
;
Marcello Leopoldo
;
Paola De Giorgio
;
Francesco Berardi
;
Roberto Perrone
关键词:
1-Arylpiperazine
;
Basicity
;
p
K
a
;
Potentiometric titration
刊名:Bioorganic and Medicinal Chemistry
出版年:2009
6.
Developments in fluorescent probes for receptor research
作者:
Marcello Leopoldo
;
Enza
Lacivita
;
Francesco Berardi
;
Roberto Perrone
刊名:Drug Discovery Today
出版年:2009
7.
Bivalent ligand approach on 4-[2-(3-methoxyphenyl)ethyl]-1-(2-methoxyphenyl)piperazine: Synthesis and binding affinities for 5-HT
7
and 5-HT
1A
receptors
作者:
Marcello Leopoldo
;
Enza
Lacivita
;
Nicola A. Colabufo
;
Mauro Niso
;
Francesco Berardi
;
Roberto Perrone
关键词:
5-HT
7
receptors
;
5-HT
1A
receptors
;
Arylpiperazine
;
Structure–
;
affinity relationships
;
Bivalent ligands
刊名:Bioorganic and Medicinal Chemistry
出版年:2007
1
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