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CNKI学位论文(3)
知网期刊论文(4)
在“
Elsevier电子期刊
”中,
命中:
18
条,耗时:小于0.01 秒
在所有数据库中总计命中:
7
条
1.
Tetrahydro-¦Â-carboline derivatives targeting fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channels
作者:
Giorgio
Ortar
a
;
giorgio
.
ortar
@uniroma1.it
;
Luciano De Petrocellis
b
;
Aniello Schiano Moriello
b
;
c
;
Marco Allarà
;
c
;
Enrico Morera
a
;
Marianna Nalli
a
;
Vincenzo Di Marzo
c
关键词:
FAAH
;
Transient receptor potential channels
;
TRPV1
;
TRPA1
;
Tetrahydro-¦Â-carbolines
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2013
2.
Biaryl tetrazolyl ureas as inhibitors of endocannabinoid metabolism: Modulation at the N-portion and distal phenyl ring
作者:
Giorgio
Ortar
a
;
giorgio
.
ortar
@uniroma1.it
;
Enrico Morera
a
;
Luciano De Petrocellis
b
;
Alessia Ligresti
c
;
Aniello Schiano Moriello
b
;
Ludovica Morera
a
;
Marianna Nalli
a
;
Rino Ragno
a
;
d
;
Adele Pirolli
a
;
d
;
Vincenzo Di Marzo
c
关键词:
Endocannabinoids
;
Fatty acid amide hydrolase (FAAH)
;
Monoacylglycerol lipase (MAGL)
;
TRPV1 channel
;
TRPA1 channel
;
Biaryl tetrazolyl ureas
刊名:European Journal of Medicinal Chemistry
出版年:2013
3.
3-Ylidenephthalides as a new class of transient receptor potential channel TRPA1 and TRPM8 modulators
作者:
Giorgio
Ortar
;
Aniello Schiano Moriello
;
Enrico Morera
;
Marianna Nalli
;
Vincenzo Di Marzo
;
Luciano De Petrocellis
关键词:
Transient receptor potential channels
;
TRPA1
;
TRPM8
;
3-Ylidenephthalides
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2013
4.
Piperazinyl carbamate fatty acid amide hydrolase inhibitors and transient receptor potential channel modulators as ¡°dual-target¡± analgesics
作者:
Sabatino Maione
;
Barbara Costa
;
Fabiana Piscitelli
;
Enrico Morera
;
Maria De Chiaro
;
Francesca Comelli
;
Serena Boccella
;
Francesca Guida
;
Roberta Verde
;
Giorgio
Ortar
;
Vincenzo Di Marzo
关键词:
Cannabinoid
;
Endocannabinoid
;
Anandamide
;
FAAH
;
TRPV1
;
TRPA1
;
N-Arachidonoylserotonin
刊名:Pharmacological Research
出版年:2013
5.
Modulation of thermo-transient receptor potential (thermo-TRP) channels by thymol-based compounds
作者:
Giorgio
Ortar
a
;
giorgio
.
ortar
@uniroma1.it
;
Ludovica Morera
a
;
Aniello Schiano Moriello
b
;
Enrico Morera
a
;
Marianna Nalli
a
;
Vincenzo Di Marzo
c
;
Luciano De Petrocellis
b
关键词:
Thermo-TRP channels
;
TRPA1
;
TRPM8
;
TRPV3
;
Tymol derivatives
;
p-Cymene-3-carboxylic acid derivatives
;
3-Amino-p-cymene derivatives
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2012
6.
Development and characterization of endocannabinoid hydrolases FAAH and MAGL inhibitors bearing a benzotriazol-1-yl carboxamide scaffold
作者:
Ludovica Morera
;
Geoffray Labar
;
Giorgio
Ortar
;
Didier M. Lambert
关键词:
FAAH
;
Fatty acid amide hydrolase
;
MAGL
;
Monoacylglycerol lipase
;
FAAH and MAGL inhibitors
刊名:Bioorganic and Medicinal Chemistry
出版年:2012
7.
(−)-Menthylamine derivatives as potent and selective antagonists of transient receptor potential melastatin type-8 (TRPM8) channels
作者:
Giorgio
Ortar
;
Luciano De Petrocellis
;
Ludovica Morera
;
Aniello Schiano Moriello
;
Pierangelo Orl
o ;
Enrico Morera
;
Marianna Nalli
;
Vincenzo Di Marzo
关键词:
Transient receptor potential channels
;
TRPA1
;
TRPV1
;
TRPM8
;
(−
;
)-Menthylamine derivatives
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
8.
Development of a potent inhibitor of 2-arachidonoylglycerol hydrolysis with antinociceptive activity in vivo
作者:
Tiziana Bisogno
;
Giorgio
Ortar
;
Stefania Petrosino
;
Enrico Morera
;
Enza Palazzo
;
Marianna Nalli
;
Sabatino Maione
;
Vincenzo Di Marzo
;
Endocannabinoid Research Group
关键词:
Endocannabinoid
;
Cannabinoid receptor
;
2-arachidonoylglycerol
;
Anandamide
;
Monoacylglycerol lipase
;
Diacylglycerol lipase
;
Fatty acid amide hydrolase
;
Pain
;
Inhibitor
刊名:Biochimica et Biophysica Acta (BBA)/Molecular and Cell Biology of Lipids
出版年:2009
9.
Synthesis and biological evaluation of piperazinyl carbamates and ureas as fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channel dual ligands
作者:
Enrico Morera
;
Luciano De Petrocellis
;
Ludovica Morera
;
Aniello Schiano Moriello
;
Alessia Ligresti
;
Marianna Nalli
;
David F. Woodward
;
Vincenzo Di Marzo
;
Giorgio
Ortar
关键词:
Fatty acid amide hydrolase
;
FAAH
;
Transient receptor potential channels
;
TRPV1
;
TRPA1
;
Dual-ligands
;
Piperazinyl carbamates
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
10.
Carbamoyl tetrazoles as inhibitors of endocannabinoid inactivation: A critical revisitation
作者:
Giorgio
Ortar
;
Maria Grazia Cascio
;
Aniello Schiano Moriello
;
Mercedes Camalli
;
Enrico Morera
;
Marianna Nalli
;
Vincenzo Di Marzo
关键词:
Endocannabinoids
;
Anandamide cellular uptake inhibitors
;
Fatty acid amide hydrolase inhibitors
;
Carbamoyl tetrazoles
刊名:European Journal of Medicinal Chemistry
出版年:2008
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